Index by author
December 01, 2005; Volume 33,Issue 12
A
Anbazhagan, Mariappan
- You have accessUNUSUAL DEHYDROXYLATION OF ANTIMICROBIAL AMIDOXIME PRODRUGS BY CYTOCHROME b5 AND NADH CYTOCHROME b5 REDUCTASEJanelle Y. Saulter, Joseph R. Kurian, Lauren A. Trepanier, Richard R. Tidwell, Arlene S. Bridges, David W. Boykin, Chad E. Stephens, Mariappan Anbazhagan and James Edwin HallDrug Metabolism and Disposition December 2005, 33 (12) 1886-1893; DOI: https://doi.org/10.1124/dmd.105.005017
Ando, Yuichi
- You have accessGEFITINIB (IRESSA) INHIBITS THE CYP3A4-MEDIATED FORMATION OF 7-ETHYL-10-(4-AMINO-1-PIPERIDINO)CARBONYLOXYCAMPTOTHECIN BUT ACTIVATES THAT OF 7-ETHYL-10-[4-N-(5-AMINOPENTANOIC ACID)-1-PIPERIDINO]CARBONYLOXYCAMPTOTHECIN FROM IRINOTECANKen-ichi Fujita, Yuichi Ando, Masaru Narabayashi, Toshimichi Miya, Fumio Nagashima, Wataru Yamamoto, Keiji Kodama, Kazuhiro Araki, Hisashi Endo and Yasutsuna SasakiDrug Metabolism and Disposition December 2005, 33 (12) 1785-1790; DOI: https://doi.org/10.1124/dmd.105.006205
Anraku, Makoto
- You have accessHYDROLYSIS OF ANGIOTENSIN II RECEPTOR BLOCKER PRODRUG OLMESARTAN MEDOXOMIL BY HUMAN SERUM ALBUMIN AND IDENTIFICATION OF ITS CATALYTIC ACTIVE SITESShen-Feng Ma, Makoto Anraku, Yasunori Iwao, Keishi Yamasaki, Ulrich Kragh-Hansen, Noriyuki Yamaotsu, Shuichi Hirono, Toshihiko Ikeda and Masaki OtagiriDrug Metabolism and Disposition December 2005, 33 (12) 1911-1919; DOI: https://doi.org/10.1124/dmd.105.006163
Aoki, Yasuhiro
- You have accessCYP2A6 AND CYP2B6 ARE INVOLVED IN NORNICOTINE FORMATION FROM NICOTINE IN HUMANS: INTERINDIVIDUAL DIFFERENCES IN THESE CONTRIBUTIONSHiroyuki Yamanaka, Miki Nakajima, Tatsuki Fukami, Haruko Sakai, Akiko Nakamura, Miki Katoh, Masataka Takamiya, Yasuhiro Aoki and Tsuyoshi YokoiDrug Metabolism and Disposition December 2005, 33 (12) 1811-1818; DOI: https://doi.org/10.1124/dmd.105.006254
Araki, Kazuhiro
- You have accessGEFITINIB (IRESSA) INHIBITS THE CYP3A4-MEDIATED FORMATION OF 7-ETHYL-10-(4-AMINO-1-PIPERIDINO)CARBONYLOXYCAMPTOTHECIN BUT ACTIVATES THAT OF 7-ETHYL-10-[4-N-(5-AMINOPENTANOIC ACID)-1-PIPERIDINO]CARBONYLOXYCAMPTOTHECIN FROM IRINOTECANKen-ichi Fujita, Yuichi Ando, Masaru Narabayashi, Toshimichi Miya, Fumio Nagashima, Wataru Yamamoto, Keiji Kodama, Kazuhiro Araki, Hisashi Endo and Yasutsuna SasakiDrug Metabolism and Disposition December 2005, 33 (12) 1785-1790; DOI: https://doi.org/10.1124/dmd.105.006205
B
Bajimaya, Susan
- You have accessDISPOSITION OF FLAVONOIDS VIA RECYCLING: COMPARISON OF INTESTINAL VERSUS HEPATIC DISPOSITIONJun Chen, Stephen Wang, Xiaobin Jia, Susan Bajimaya, Huimin Lin, Vincent H. Tam and Ming HuDrug Metabolism and Disposition December 2005, 33 (12) 1777-1784; DOI: https://doi.org/10.1124/dmd.105.003673
Beaune, Philippe
- You have accessSIMULTANEOUS MEASUREMENT OF 23 ISOFORMS FROM THE HUMAN CYTOCHROME P450 FAMILIES 1 TO 3 BY QUANTITATIVE REVERSE TRANSCRIPTASE-POLYMERASE CHAIN REACTIONIgor Girault, Nathalie Rougier, Christophe Chesné, Rosette Lidereau, Philippe Beaune, Ivan Bieche and Isabelle de WaziersDrug Metabolism and Disposition December 2005, 33 (12) 1803-1810; DOI: https://doi.org/10.1124/dmd.105.005173
Bieche, Ivan
- You have accessSIMULTANEOUS MEASUREMENT OF 23 ISOFORMS FROM THE HUMAN CYTOCHROME P450 FAMILIES 1 TO 3 BY QUANTITATIVE REVERSE TRANSCRIPTASE-POLYMERASE CHAIN REACTIONIgor Girault, Nathalie Rougier, Christophe Chesné, Rosette Lidereau, Philippe Beaune, Ivan Bieche and Isabelle de WaziersDrug Metabolism and Disposition December 2005, 33 (12) 1803-1810; DOI: https://doi.org/10.1124/dmd.105.005173
Boykin, David W.
- You have accessUNUSUAL DEHYDROXYLATION OF ANTIMICROBIAL AMIDOXIME PRODRUGS BY CYTOCHROME b5 AND NADH CYTOCHROME b5 REDUCTASEJanelle Y. Saulter, Joseph R. Kurian, Lauren A. Trepanier, Richard R. Tidwell, Arlene S. Bridges, David W. Boykin, Chad E. Stephens, Mariappan Anbazhagan and James Edwin HallDrug Metabolism and Disposition December 2005, 33 (12) 1886-1893; DOI: https://doi.org/10.1124/dmd.105.005017
Bräter, M.
- You have accessEFFECT OF PROPIVERINE ON CYTOCHROME P450 ENZYMES: A COCKTAIL INTERACTION STUDY IN HEALTHY VOLUNTEERSD. Tomalik-Scharte, A. Jetter, M. Kinzig-Schippers, A. Skott, F. Sörgel, T. Klaassen, D. Kasel, S. Harlfinger, O. Doroshyenko, D. Frank, J. Kirchheiner, M. Bräter, K. Richter, T. Gramatté and U. FuhrDrug Metabolism and Disposition December 2005, 33 (12) 1859-1866; DOI: https://doi.org/10.1124/dmd.105.005272
Bridges, Arlene S.
- You have accessUNUSUAL DEHYDROXYLATION OF ANTIMICROBIAL AMIDOXIME PRODRUGS BY CYTOCHROME b5 AND NADH CYTOCHROME b5 REDUCTASEJanelle Y. Saulter, Joseph R. Kurian, Lauren A. Trepanier, Richard R. Tidwell, Arlene S. Bridges, David W. Boykin, Chad E. Stephens, Mariappan Anbazhagan and James Edwin HallDrug Metabolism and Disposition December 2005, 33 (12) 1886-1893; DOI: https://doi.org/10.1124/dmd.105.005017
Bu, Hai-Zhi
- You have accessHUMAN IN VITRO GLUTATHIONYL AND PROTEIN ADDUCTS OF CARBAMAZEPINE-10,11-EPOXIDE, A STABLE AND PHARMACOLOGICALLY ACTIVE METABOLITE OF CARBAMAZEPINEHai-Zhi Bu, Ping Kang, Alan J. Deese, Ping Zhao and William F. PoolDrug Metabolism and Disposition December 2005, 33 (12) 1920-1924; DOI: https://doi.org/10.1124/dmd.105.006866
C
Caldwell, Gary W.
- You have accessBIOACTIVATION OF 4-METHYLPHENOL (p-CRESOL) VIA CYTOCHROME P450-MEDIATED AROMATIC OXIDATION IN HUMAN LIVER MICROSOMESZhengyin Yan, H. Marlon Zhong, Noureddine Maher, Rhoda Torres, Gregory C. Leo, Gary W. Caldwell and Norman HuebertDrug Metabolism and Disposition December 2005, 33 (12) 1867-1876; DOI: https://doi.org/10.1124/dmd.105.006387
Cato, Brian
- You have accessSPECIES DIFFERENCES IN THE ELIMINATION OF A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR AGONIST HIGHLIGHTED BY OXIDATIVE METABOLISM OF ITS ACYL GLUCURONIDEChristopher J. Kochansky, Yuan-Qing Xia, Sui Wang, Brian Cato, Mellissa Creighton, Stella H. Vincent, Ronald B. Franklin and James R. ReedDrug Metabolism and Disposition December 2005, 33 (12) 1894-1904; DOI: https://doi.org/10.1124/dmd.105.004010
Chen, Jun
- You have accessDISPOSITION OF FLAVONOIDS VIA RECYCLING: COMPARISON OF INTESTINAL VERSUS HEPATIC DISPOSITIONJun Chen, Stephen Wang, Xiaobin Jia, Susan Bajimaya, Huimin Lin, Vincent H. Tam and Ming HuDrug Metabolism and Disposition December 2005, 33 (12) 1777-1784; DOI: https://doi.org/10.1124/dmd.105.003673
Chesné, Christophe
- You have accessSIMULTANEOUS MEASUREMENT OF 23 ISOFORMS FROM THE HUMAN CYTOCHROME P450 FAMILIES 1 TO 3 BY QUANTITATIVE REVERSE TRANSCRIPTASE-POLYMERASE CHAIN REACTIONIgor Girault, Nathalie Rougier, Christophe Chesné, Rosette Lidereau, Philippe Beaune, Ivan Bieche and Isabelle de WaziersDrug Metabolism and Disposition December 2005, 33 (12) 1803-1810; DOI: https://doi.org/10.1124/dmd.105.005173
Chilakapati, Jaya
- You have accessSATURATION TOXICOKINETICS OF THIOACETAMIDE: ROLE IN INITIATION OF LIVER INJURYJaya Chilakapati, Kartik Shankar, Midhun C. Korrapati, Ronald A. Hill and Harihara M. MehendaleDrug Metabolism and Disposition December 2005, 33 (12) 1877-1885; DOI: https://doi.org/10.1124/dmd.105.005520
Chun, Young-Jin
- You have accessMODULATION OF HUMAN CYTOCHROME P450 1B1 EXPRESSION BY 2,4,3′,5′-TETRAMETHOXYSTILBENEYoung-Jin Chun, Sang-Kwang Lee and Mie Young KimDrug Metabolism and Disposition December 2005, 33 (12) 1771-1776; DOI: https://doi.org/10.1124/dmd.105.006502
Court, Michael H.
- You have accessROLE OF THE NUCLEAR RECEPTOR PREGNANE X RECEPTOR IN ACETAMINOPHEN HEPATOTOXICITYKristina K. Wolf, Sheryl G. Wood, Jane A. Hunt, Brooke W. Walton-Strong, Kazuto Yasuda, Lubin Lan, Su X. Duan, Qin Hao, Steven A. Wrighton, Elizabeth H. Jeffery, Ronald M. Evans, Juliana G. Szakacs, Lisa L. von Moltke, David J. Greenblatt, Michael H. Court, Erin G. Schuetz, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition December 2005, 33 (12) 1827-1836; DOI: https://doi.org/10.1124/dmd.105.005256
Creighton, Mellissa
- You have accessSPECIES DIFFERENCES IN THE ELIMINATION OF A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR AGONIST HIGHLIGHTED BY OXIDATIVE METABOLISM OF ITS ACYL GLUCURONIDEChristopher J. Kochansky, Yuan-Qing Xia, Sui Wang, Brian Cato, Mellissa Creighton, Stella H. Vincent, Ronald B. Franklin and James R. ReedDrug Metabolism and Disposition December 2005, 33 (12) 1894-1904; DOI: https://doi.org/10.1124/dmd.105.004010
Cui, Donghui
- You have accessTRANSAMINATION IN THE METABOLISM OF THE NEPHROTOXICANT N-(3,5-DICHLOROPHENYL)SUCCINIMIDE IN RATSDonghui Cui, Gary O. Rankin and Peter J. HarvisonDrug Metabolism and Disposition December 2005, 33 (12) 1765-1770; DOI: https://doi.org/10.1124/dmd.105.006593
D
Deese, Alan J.
- You have accessHUMAN IN VITRO GLUTATHIONYL AND PROTEIN ADDUCTS OF CARBAMAZEPINE-10,11-EPOXIDE, A STABLE AND PHARMACOLOGICALLY ACTIVE METABOLITE OF CARBAMAZEPINEHai-Zhi Bu, Ping Kang, Alan J. Deese, Ping Zhao and William F. PoolDrug Metabolism and Disposition December 2005, 33 (12) 1920-1924; DOI: https://doi.org/10.1124/dmd.105.006866
de Waziers, Isabelle
- You have accessSIMULTANEOUS MEASUREMENT OF 23 ISOFORMS FROM THE HUMAN CYTOCHROME P450 FAMILIES 1 TO 3 BY QUANTITATIVE REVERSE TRANSCRIPTASE-POLYMERASE CHAIN REACTIONIgor Girault, Nathalie Rougier, Christophe Chesné, Rosette Lidereau, Philippe Beaune, Ivan Bieche and Isabelle de WaziersDrug Metabolism and Disposition December 2005, 33 (12) 1803-1810; DOI: https://doi.org/10.1124/dmd.105.005173
Dicke, Kari E.
- You have accessNICOTINE AND 4-(METHYLNITROSAMINO)-1-(3-PYRIDYL)-BUTANONE METABOLISM BY CYTOCHROME P450 2B6Kari E. Dicke, Sara M. Skrlin and Sharon E. MurphyDrug Metabolism and Disposition December 2005, 33 (12) 1760-1764; DOI: https://doi.org/10.1124/dmd.105.006718
Doroshyenko, O.
- You have accessEFFECT OF PROPIVERINE ON CYTOCHROME P450 ENZYMES: A COCKTAIL INTERACTION STUDY IN HEALTHY VOLUNTEERSD. Tomalik-Scharte, A. Jetter, M. Kinzig-Schippers, A. Skott, F. Sörgel, T. Klaassen, D. Kasel, S. Harlfinger, O. Doroshyenko, D. Frank, J. Kirchheiner, M. Bräter, K. Richter, T. Gramatté and U. FuhrDrug Metabolism and Disposition December 2005, 33 (12) 1859-1866; DOI: https://doi.org/10.1124/dmd.105.005272
Duan, Su X.
- You have accessROLE OF THE NUCLEAR RECEPTOR PREGNANE X RECEPTOR IN ACETAMINOPHEN HEPATOTOXICITYKristina K. Wolf, Sheryl G. Wood, Jane A. Hunt, Brooke W. Walton-Strong, Kazuto Yasuda, Lubin Lan, Su X. Duan, Qin Hao, Steven A. Wrighton, Elizabeth H. Jeffery, Ronald M. Evans, Juliana G. Szakacs, Lisa L. von Moltke, David J. Greenblatt, Michael H. Court, Erin G. Schuetz, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition December 2005, 33 (12) 1827-1836; DOI: https://doi.org/10.1124/dmd.105.005256
E
Endo, Hisashi
- You have accessGEFITINIB (IRESSA) INHIBITS THE CYP3A4-MEDIATED FORMATION OF 7-ETHYL-10-(4-AMINO-1-PIPERIDINO)CARBONYLOXYCAMPTOTHECIN BUT ACTIVATES THAT OF 7-ETHYL-10-[4-N-(5-AMINOPENTANOIC ACID)-1-PIPERIDINO]CARBONYLOXYCAMPTOTHECIN FROM IRINOTECANKen-ichi Fujita, Yuichi Ando, Masaru Narabayashi, Toshimichi Miya, Fumio Nagashima, Wataru Yamamoto, Keiji Kodama, Kazuhiro Araki, Hisashi Endo and Yasutsuna SasakiDrug Metabolism and Disposition December 2005, 33 (12) 1785-1790; DOI: https://doi.org/10.1124/dmd.105.006205
Evans, Ronald M.
- You have accessROLE OF THE NUCLEAR RECEPTOR PREGNANE X RECEPTOR IN ACETAMINOPHEN HEPATOTOXICITYKristina K. Wolf, Sheryl G. Wood, Jane A. Hunt, Brooke W. Walton-Strong, Kazuto Yasuda, Lubin Lan, Su X. Duan, Qin Hao, Steven A. Wrighton, Elizabeth H. Jeffery, Ronald M. Evans, Juliana G. Szakacs, Lisa L. von Moltke, David J. Greenblatt, Michael H. Court, Erin G. Schuetz, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition December 2005, 33 (12) 1827-1836; DOI: https://doi.org/10.1124/dmd.105.005256
F
Frank, D.
- You have accessEFFECT OF PROPIVERINE ON CYTOCHROME P450 ENZYMES: A COCKTAIL INTERACTION STUDY IN HEALTHY VOLUNTEERSD. Tomalik-Scharte, A. Jetter, M. Kinzig-Schippers, A. Skott, F. Sörgel, T. Klaassen, D. Kasel, S. Harlfinger, O. Doroshyenko, D. Frank, J. Kirchheiner, M. Bräter, K. Richter, T. Gramatté and U. FuhrDrug Metabolism and Disposition December 2005, 33 (12) 1859-1866; DOI: https://doi.org/10.1124/dmd.105.005272
Franklin, Ronald B.
- You have accessSPECIES DIFFERENCES IN THE ELIMINATION OF A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR AGONIST HIGHLIGHTED BY OXIDATIVE METABOLISM OF ITS ACYL GLUCURONIDEChristopher J. Kochansky, Yuan-Qing Xia, Sui Wang, Brian Cato, Mellissa Creighton, Stella H. Vincent, Ronald B. Franklin and James R. ReedDrug Metabolism and Disposition December 2005, 33 (12) 1894-1904; DOI: https://doi.org/10.1124/dmd.105.004010
Fuhr, U.
- You have accessEFFECT OF PROPIVERINE ON CYTOCHROME P450 ENZYMES: A COCKTAIL INTERACTION STUDY IN HEALTHY VOLUNTEERSD. Tomalik-Scharte, A. Jetter, M. Kinzig-Schippers, A. Skott, F. Sörgel, T. Klaassen, D. Kasel, S. Harlfinger, O. Doroshyenko, D. Frank, J. Kirchheiner, M. Bräter, K. Richter, T. Gramatté and U. FuhrDrug Metabolism and Disposition December 2005, 33 (12) 1859-1866; DOI: https://doi.org/10.1124/dmd.105.005272
Fujita, Ken-ichi
- You have accessGEFITINIB (IRESSA) INHIBITS THE CYP3A4-MEDIATED FORMATION OF 7-ETHYL-10-(4-AMINO-1-PIPERIDINO)CARBONYLOXYCAMPTOTHECIN BUT ACTIVATES THAT OF 7-ETHYL-10-[4-N-(5-AMINOPENTANOIC ACID)-1-PIPERIDINO]CARBONYLOXYCAMPTOTHECIN FROM IRINOTECANKen-ichi Fujita, Yuichi Ando, Masaru Narabayashi, Toshimichi Miya, Fumio Nagashima, Wataru Yamamoto, Keiji Kodama, Kazuhiro Araki, Hisashi Endo and Yasutsuna SasakiDrug Metabolism and Disposition December 2005, 33 (12) 1785-1790; DOI: https://doi.org/10.1124/dmd.105.006205
Fukami, Tatsuki
- You have accessCYP2A6 AND CYP2B6 ARE INVOLVED IN NORNICOTINE FORMATION FROM NICOTINE IN HUMANS: INTERINDIVIDUAL DIFFERENCES IN THESE CONTRIBUTIONSHiroyuki Yamanaka, Miki Nakajima, Tatsuki Fukami, Haruko Sakai, Akiko Nakamura, Miki Katoh, Masataka Takamiya, Yasuhiro Aoki and Tsuyoshi YokoiDrug Metabolism and Disposition December 2005, 33 (12) 1811-1818; DOI: https://doi.org/10.1124/dmd.105.006254
G
Girault, Igor
- You have accessSIMULTANEOUS MEASUREMENT OF 23 ISOFORMS FROM THE HUMAN CYTOCHROME P450 FAMILIES 1 TO 3 BY QUANTITATIVE REVERSE TRANSCRIPTASE-POLYMERASE CHAIN REACTIONIgor Girault, Nathalie Rougier, Christophe Chesné, Rosette Lidereau, Philippe Beaune, Ivan Bieche and Isabelle de WaziersDrug Metabolism and Disposition December 2005, 33 (12) 1803-1810; DOI: https://doi.org/10.1124/dmd.105.005173
Gramatté, T.
- You have accessEFFECT OF PROPIVERINE ON CYTOCHROME P450 ENZYMES: A COCKTAIL INTERACTION STUDY IN HEALTHY VOLUNTEERSD. Tomalik-Scharte, A. Jetter, M. Kinzig-Schippers, A. Skott, F. Sörgel, T. Klaassen, D. Kasel, S. Harlfinger, O. Doroshyenko, D. Frank, J. Kirchheiner, M. Bräter, K. Richter, T. Gramatté and U. FuhrDrug Metabolism and Disposition December 2005, 33 (12) 1859-1866; DOI: https://doi.org/10.1124/dmd.105.005272
Greenblatt, David J.
- You have accessROLE OF THE NUCLEAR RECEPTOR PREGNANE X RECEPTOR IN ACETAMINOPHEN HEPATOTOXICITYKristina K. Wolf, Sheryl G. Wood, Jane A. Hunt, Brooke W. Walton-Strong, Kazuto Yasuda, Lubin Lan, Su X. Duan, Qin Hao, Steven A. Wrighton, Elizabeth H. Jeffery, Ronald M. Evans, Juliana G. Szakacs, Lisa L. von Moltke, David J. Greenblatt, Michael H. Court, Erin G. Schuetz, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition December 2005, 33 (12) 1827-1836; DOI: https://doi.org/10.1124/dmd.105.005256
H
Hakooz, Nancy
- You have accessPREDICTION OF METABOLIC CLEARANCE USING CRYOPRESERVED HUMAN HEPATOCYTES: KINETIC CHARACTERISTICS FOR FIVE BENZODIAZEPINESDavid Hallifax, Helen C. Rawden, Nancy Hakooz and J. Brian HoustonDrug Metabolism and Disposition December 2005, 33 (12) 1852-1858; DOI: https://doi.org/10.1124/dmd.105.005389
Hall, James Edwin
- You have accessUNUSUAL DEHYDROXYLATION OF ANTIMICROBIAL AMIDOXIME PRODRUGS BY CYTOCHROME b5 AND NADH CYTOCHROME b5 REDUCTASEJanelle Y. Saulter, Joseph R. Kurian, Lauren A. Trepanier, Richard R. Tidwell, Arlene S. Bridges, David W. Boykin, Chad E. Stephens, Mariappan Anbazhagan and James Edwin HallDrug Metabolism and Disposition December 2005, 33 (12) 1886-1893; DOI: https://doi.org/10.1124/dmd.105.005017
Hallifax, David
- You have accessPREDICTION OF METABOLIC CLEARANCE USING CRYOPRESERVED HUMAN HEPATOCYTES: KINETIC CHARACTERISTICS FOR FIVE BENZODIAZEPINESDavid Hallifax, Helen C. Rawden, Nancy Hakooz and J. Brian HoustonDrug Metabolism and Disposition December 2005, 33 (12) 1852-1858; DOI: https://doi.org/10.1124/dmd.105.005389
Halpert, James R.
- You have accessJames R. HalpertDrug Metabolism and Disposition December 2005, 33 (12) 1759; DOI: https://doi.org/10.1124/dmd.33.12.1759
Hanioka, Nobumitsu
- You have accessFUNCTIONAL ANALYSIS OF THREE CYP1A2 VARIANTS FOUND IN A JAPANESE POPULATIONYoshiro Saito, Nobumitsu Hanioka, Keiko Maekawa, Takashi Isobe, Yumi Tsuneto, Ryosuke Nakamura, Akiko Soyama, Shogo Ozawa, Toshiko Tanaka-Kagawa, Hideto Jinno, Shizuo Narimatsu and Jun-ichi SawadaDrug Metabolism and Disposition December 2005, 33 (12) 1905-1910; DOI: https://doi.org/10.1124/dmd.105.005819
Hao, Qin
- You have accessROLE OF THE NUCLEAR RECEPTOR PREGNANE X RECEPTOR IN ACETAMINOPHEN HEPATOTOXICITYKristina K. Wolf, Sheryl G. Wood, Jane A. Hunt, Brooke W. Walton-Strong, Kazuto Yasuda, Lubin Lan, Su X. Duan, Qin Hao, Steven A. Wrighton, Elizabeth H. Jeffery, Ronald M. Evans, Juliana G. Szakacs, Lisa L. von Moltke, David J. Greenblatt, Michael H. Court, Erin G. Schuetz, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition December 2005, 33 (12) 1827-1836; DOI: https://doi.org/10.1124/dmd.105.005256
Harlfinger, S.
- You have accessEFFECT OF PROPIVERINE ON CYTOCHROME P450 ENZYMES: A COCKTAIL INTERACTION STUDY IN HEALTHY VOLUNTEERSD. Tomalik-Scharte, A. Jetter, M. Kinzig-Schippers, A. Skott, F. Sörgel, T. Klaassen, D. Kasel, S. Harlfinger, O. Doroshyenko, D. Frank, J. Kirchheiner, M. Bräter, K. Richter, T. Gramatté and U. FuhrDrug Metabolism and Disposition December 2005, 33 (12) 1859-1866; DOI: https://doi.org/10.1124/dmd.105.005272
Harvison, Peter J.
- You have accessTRANSAMINATION IN THE METABOLISM OF THE NEPHROTOXICANT N-(3,5-DICHLOROPHENYL)SUCCINIMIDE IN RATSDonghui Cui, Gary O. Rankin and Peter J. HarvisonDrug Metabolism and Disposition December 2005, 33 (12) 1765-1770; DOI: https://doi.org/10.1124/dmd.105.006593
Hill, Ronald A.
- You have accessSATURATION TOXICOKINETICS OF THIOACETAMIDE: ROLE IN INITIATION OF LIVER INJURYJaya Chilakapati, Kartik Shankar, Midhun C. Korrapati, Ronald A. Hill and Harihara M. MehendaleDrug Metabolism and Disposition December 2005, 33 (12) 1877-1885; DOI: https://doi.org/10.1124/dmd.105.005520
Hirayama, Masamichi
- You have accessINVOLVEMENT OF URIC ACID TRANSPORTER IN INCREASED RENAL CLEARANCE OF THE XANTHINE OXIDASE INHIBITOR OXYPURINOL INDUCED BY A URICOSURIC AGENT, BENZBROMARONETakashi Iwanaga, Daisuke Kobayashi, Masamichi Hirayama, Tomoji Maeda and Ikumi TamaiDrug Metabolism and Disposition December 2005, 33 (12) 1791-1795; DOI: https://doi.org/10.1124/dmd.105.006056
Hirono, Shuichi
- You have accessHYDROLYSIS OF ANGIOTENSIN II RECEPTOR BLOCKER PRODRUG OLMESARTAN MEDOXOMIL BY HUMAN SERUM ALBUMIN AND IDENTIFICATION OF ITS CATALYTIC ACTIVE SITESShen-Feng Ma, Makoto Anraku, Yasunori Iwao, Keishi Yamasaki, Ulrich Kragh-Hansen, Noriyuki Yamaotsu, Shuichi Hirono, Toshihiko Ikeda and Masaki OtagiriDrug Metabolism and Disposition December 2005, 33 (12) 1911-1919; DOI: https://doi.org/10.1124/dmd.105.006163
Houston, J. Brian
- You have accessPREDICTION OF METABOLIC CLEARANCE USING CRYOPRESERVED HUMAN HEPATOCYTES: KINETIC CHARACTERISTICS FOR FIVE BENZODIAZEPINESDavid Hallifax, Helen C. Rawden, Nancy Hakooz and J. Brian HoustonDrug Metabolism and Disposition December 2005, 33 (12) 1852-1858; DOI: https://doi.org/10.1124/dmd.105.005389
Hu, Ming
- You have accessDISPOSITION OF FLAVONOIDS VIA RECYCLING: COMPARISON OF INTESTINAL VERSUS HEPATIC DISPOSITIONJun Chen, Stephen Wang, Xiaobin Jia, Susan Bajimaya, Huimin Lin, Vincent H. Tam and Ming HuDrug Metabolism and Disposition December 2005, 33 (12) 1777-1784; DOI: https://doi.org/10.1124/dmd.105.003673
Huebert, Norman
- You have accessBIOACTIVATION OF 4-METHYLPHENOL (p-CRESOL) VIA CYTOCHROME P450-MEDIATED AROMATIC OXIDATION IN HUMAN LIVER MICROSOMESZhengyin Yan, H. Marlon Zhong, Noureddine Maher, Rhoda Torres, Gregory C. Leo, Gary W. Caldwell and Norman HuebertDrug Metabolism and Disposition December 2005, 33 (12) 1867-1876; DOI: https://doi.org/10.1124/dmd.105.006387
Hunt, Jane A.
- You have accessROLE OF THE NUCLEAR RECEPTOR PREGNANE X RECEPTOR IN ACETAMINOPHEN HEPATOTOXICITYKristina K. Wolf, Sheryl G. Wood, Jane A. Hunt, Brooke W. Walton-Strong, Kazuto Yasuda, Lubin Lan, Su X. Duan, Qin Hao, Steven A. Wrighton, Elizabeth H. Jeffery, Ronald M. Evans, Juliana G. Szakacs, Lisa L. von Moltke, David J. Greenblatt, Michael H. Court, Erin G. Schuetz, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition December 2005, 33 (12) 1827-1836; DOI: https://doi.org/10.1124/dmd.105.005256
I
Ikeda, Toshihiko
- You have accessHYDROLYSIS OF ANGIOTENSIN II RECEPTOR BLOCKER PRODRUG OLMESARTAN MEDOXOMIL BY HUMAN SERUM ALBUMIN AND IDENTIFICATION OF ITS CATALYTIC ACTIVE SITESShen-Feng Ma, Makoto Anraku, Yasunori Iwao, Keishi Yamasaki, Ulrich Kragh-Hansen, Noriyuki Yamaotsu, Shuichi Hirono, Toshihiko Ikeda and Masaki OtagiriDrug Metabolism and Disposition December 2005, 33 (12) 1911-1919; DOI: https://doi.org/10.1124/dmd.105.006163
Isobe, Takashi
- You have accessFUNCTIONAL ANALYSIS OF THREE CYP1A2 VARIANTS FOUND IN A JAPANESE POPULATIONYoshiro Saito, Nobumitsu Hanioka, Keiko Maekawa, Takashi Isobe, Yumi Tsuneto, Ryosuke Nakamura, Akiko Soyama, Shogo Ozawa, Toshiko Tanaka-Kagawa, Hideto Jinno, Shizuo Narimatsu and Jun-ichi SawadaDrug Metabolism and Disposition December 2005, 33 (12) 1905-1910; DOI: https://doi.org/10.1124/dmd.105.005819
Iwanaga, Takashi
- You have accessINVOLVEMENT OF URIC ACID TRANSPORTER IN INCREASED RENAL CLEARANCE OF THE XANTHINE OXIDASE INHIBITOR OXYPURINOL INDUCED BY A URICOSURIC AGENT, BENZBROMARONETakashi Iwanaga, Daisuke Kobayashi, Masamichi Hirayama, Tomoji Maeda and Ikumi TamaiDrug Metabolism and Disposition December 2005, 33 (12) 1791-1795; DOI: https://doi.org/10.1124/dmd.105.006056
Iwao, Yasunori
- You have accessHYDROLYSIS OF ANGIOTENSIN II RECEPTOR BLOCKER PRODRUG OLMESARTAN MEDOXOMIL BY HUMAN SERUM ALBUMIN AND IDENTIFICATION OF ITS CATALYTIC ACTIVE SITESShen-Feng Ma, Makoto Anraku, Yasunori Iwao, Keishi Yamasaki, Ulrich Kragh-Hansen, Noriyuki Yamaotsu, Shuichi Hirono, Toshihiko Ikeda and Masaki OtagiriDrug Metabolism and Disposition December 2005, 33 (12) 1911-1919; DOI: https://doi.org/10.1124/dmd.105.006163
J
Jeffery, Elizabeth H.
- You have accessROLE OF THE NUCLEAR RECEPTOR PREGNANE X RECEPTOR IN ACETAMINOPHEN HEPATOTOXICITYKristina K. Wolf, Sheryl G. Wood, Jane A. Hunt, Brooke W. Walton-Strong, Kazuto Yasuda, Lubin Lan, Su X. Duan, Qin Hao, Steven A. Wrighton, Elizabeth H. Jeffery, Ronald M. Evans, Juliana G. Szakacs, Lisa L. von Moltke, David J. Greenblatt, Michael H. Court, Erin G. Schuetz, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition December 2005, 33 (12) 1827-1836; DOI: https://doi.org/10.1124/dmd.105.005256
Jetter, A.
- You have accessEFFECT OF PROPIVERINE ON CYTOCHROME P450 ENZYMES: A COCKTAIL INTERACTION STUDY IN HEALTHY VOLUNTEERSD. Tomalik-Scharte, A. Jetter, M. Kinzig-Schippers, A. Skott, F. Sörgel, T. Klaassen, D. Kasel, S. Harlfinger, O. Doroshyenko, D. Frank, J. Kirchheiner, M. Bräter, K. Richter, T. Gramatté and U. FuhrDrug Metabolism and Disposition December 2005, 33 (12) 1859-1866; DOI: https://doi.org/10.1124/dmd.105.005272
Jia, Xiaobin
- You have accessDISPOSITION OF FLAVONOIDS VIA RECYCLING: COMPARISON OF INTESTINAL VERSUS HEPATIC DISPOSITIONJun Chen, Stephen Wang, Xiaobin Jia, Susan Bajimaya, Huimin Lin, Vincent H. Tam and Ming HuDrug Metabolism and Disposition December 2005, 33 (12) 1777-1784; DOI: https://doi.org/10.1124/dmd.105.003673
Jinno, Hideto
- You have accessFUNCTIONAL ANALYSIS OF THREE CYP1A2 VARIANTS FOUND IN A JAPANESE POPULATIONYoshiro Saito, Nobumitsu Hanioka, Keiko Maekawa, Takashi Isobe, Yumi Tsuneto, Ryosuke Nakamura, Akiko Soyama, Shogo Ozawa, Toshiko Tanaka-Kagawa, Hideto Jinno, Shizuo Narimatsu and Jun-ichi SawadaDrug Metabolism and Disposition December 2005, 33 (12) 1905-1910; DOI: https://doi.org/10.1124/dmd.105.005819
K
Kang, Ping
- You have accessHUMAN IN VITRO GLUTATHIONYL AND PROTEIN ADDUCTS OF CARBAMAZEPINE-10,11-EPOXIDE, A STABLE AND PHARMACOLOGICALLY ACTIVE METABOLITE OF CARBAMAZEPINEHai-Zhi Bu, Ping Kang, Alan J. Deese, Ping Zhao and William F. PoolDrug Metabolism and Disposition December 2005, 33 (12) 1920-1924; DOI: https://doi.org/10.1124/dmd.105.006866
Kasel, D.
- You have accessEFFECT OF PROPIVERINE ON CYTOCHROME P450 ENZYMES: A COCKTAIL INTERACTION STUDY IN HEALTHY VOLUNTEERSD. Tomalik-Scharte, A. Jetter, M. Kinzig-Schippers, A. Skott, F. Sörgel, T. Klaassen, D. Kasel, S. Harlfinger, O. Doroshyenko, D. Frank, J. Kirchheiner, M. Bräter, K. Richter, T. Gramatté and U. FuhrDrug Metabolism and Disposition December 2005, 33 (12) 1859-1866; DOI: https://doi.org/10.1124/dmd.105.005272
Katoh, Miki
- You have accessCYP2A6 AND CYP2B6 ARE INVOLVED IN NORNICOTINE FORMATION FROM NICOTINE IN HUMANS: INTERINDIVIDUAL DIFFERENCES IN THESE CONTRIBUTIONSHiroyuki Yamanaka, Miki Nakajima, Tatsuki Fukami, Haruko Sakai, Akiko Nakamura, Miki Katoh, Masataka Takamiya, Yasuhiro Aoki and Tsuyoshi YokoiDrug Metabolism and Disposition December 2005, 33 (12) 1811-1818; DOI: https://doi.org/10.1124/dmd.105.006254
Kim, Mie Young
- You have accessMODULATION OF HUMAN CYTOCHROME P450 1B1 EXPRESSION BY 2,4,3′,5′-TETRAMETHOXYSTILBENEYoung-Jin Chun, Sang-Kwang Lee and Mie Young KimDrug Metabolism and Disposition December 2005, 33 (12) 1771-1776; DOI: https://doi.org/10.1124/dmd.105.006502
Kinzig-Schippers, M.
- You have accessEFFECT OF PROPIVERINE ON CYTOCHROME P450 ENZYMES: A COCKTAIL INTERACTION STUDY IN HEALTHY VOLUNTEERSD. Tomalik-Scharte, A. Jetter, M. Kinzig-Schippers, A. Skott, F. Sörgel, T. Klaassen, D. Kasel, S. Harlfinger, O. Doroshyenko, D. Frank, J. Kirchheiner, M. Bräter, K. Richter, T. Gramatté and U. FuhrDrug Metabolism and Disposition December 2005, 33 (12) 1859-1866; DOI: https://doi.org/10.1124/dmd.105.005272
Kirchheiner, J.
- You have accessEFFECT OF PROPIVERINE ON CYTOCHROME P450 ENZYMES: A COCKTAIL INTERACTION STUDY IN HEALTHY VOLUNTEERSD. Tomalik-Scharte, A. Jetter, M. Kinzig-Schippers, A. Skott, F. Sörgel, T. Klaassen, D. Kasel, S. Harlfinger, O. Doroshyenko, D. Frank, J. Kirchheiner, M. Bräter, K. Richter, T. Gramatté and U. FuhrDrug Metabolism and Disposition December 2005, 33 (12) 1859-1866; DOI: https://doi.org/10.1124/dmd.105.005272
Klaassen, T.
- You have accessEFFECT OF PROPIVERINE ON CYTOCHROME P450 ENZYMES: A COCKTAIL INTERACTION STUDY IN HEALTHY VOLUNTEERSD. Tomalik-Scharte, A. Jetter, M. Kinzig-Schippers, A. Skott, F. Sörgel, T. Klaassen, D. Kasel, S. Harlfinger, O. Doroshyenko, D. Frank, J. Kirchheiner, M. Bräter, K. Richter, T. Gramatté and U. FuhrDrug Metabolism and Disposition December 2005, 33 (12) 1859-1866; DOI: https://doi.org/10.1124/dmd.105.005272
Kobayashi, Daisuke
- You have accessINVOLVEMENT OF URIC ACID TRANSPORTER IN INCREASED RENAL CLEARANCE OF THE XANTHINE OXIDASE INHIBITOR OXYPURINOL INDUCED BY A URICOSURIC AGENT, BENZBROMARONETakashi Iwanaga, Daisuke Kobayashi, Masamichi Hirayama, Tomoji Maeda and Ikumi TamaiDrug Metabolism and Disposition December 2005, 33 (12) 1791-1795; DOI: https://doi.org/10.1124/dmd.105.006056
Kobayashi, Yasuna
- You have accessFUNCTIONAL CHARACTERIZATION OF HUMAN MONOCARBOXYLATE TRANSPORTER 6 (SLC16A5)Yuichi Murakami, Noriko Kohyama, Yasuna Kobayashi, Masayuki Ohbayashi, Hisakazu Ohtani, Yasufumi Sawada and Toshinori YamamotoDrug Metabolism and Disposition December 2005, 33 (12) 1845-1851; DOI: https://doi.org/10.1124/dmd.105.005264
Kochansky, Christopher J.
- You have accessSPECIES DIFFERENCES IN THE ELIMINATION OF A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR AGONIST HIGHLIGHTED BY OXIDATIVE METABOLISM OF ITS ACYL GLUCURONIDEChristopher J. Kochansky, Yuan-Qing Xia, Sui Wang, Brian Cato, Mellissa Creighton, Stella H. Vincent, Ronald B. Franklin and James R. ReedDrug Metabolism and Disposition December 2005, 33 (12) 1894-1904; DOI: https://doi.org/10.1124/dmd.105.004010
Kodama, Keiji
- You have accessGEFITINIB (IRESSA) INHIBITS THE CYP3A4-MEDIATED FORMATION OF 7-ETHYL-10-(4-AMINO-1-PIPERIDINO)CARBONYLOXYCAMPTOTHECIN BUT ACTIVATES THAT OF 7-ETHYL-10-[4-N-(5-AMINOPENTANOIC ACID)-1-PIPERIDINO]CARBONYLOXYCAMPTOTHECIN FROM IRINOTECANKen-ichi Fujita, Yuichi Ando, Masaru Narabayashi, Toshimichi Miya, Fumio Nagashima, Wataru Yamamoto, Keiji Kodama, Kazuhiro Araki, Hisashi Endo and Yasutsuna SasakiDrug Metabolism and Disposition December 2005, 33 (12) 1785-1790; DOI: https://doi.org/10.1124/dmd.105.006205
Kohyama, Noriko
- You have accessFUNCTIONAL CHARACTERIZATION OF HUMAN MONOCARBOXYLATE TRANSPORTER 6 (SLC16A5)Yuichi Murakami, Noriko Kohyama, Yasuna Kobayashi, Masayuki Ohbayashi, Hisakazu Ohtani, Yasufumi Sawada and Toshinori YamamotoDrug Metabolism and Disposition December 2005, 33 (12) 1845-1851; DOI: https://doi.org/10.1124/dmd.105.005264
Korrapati, Midhun C.
- You have accessSATURATION TOXICOKINETICS OF THIOACETAMIDE: ROLE IN INITIATION OF LIVER INJURYJaya Chilakapati, Kartik Shankar, Midhun C. Korrapati, Ronald A. Hill and Harihara M. MehendaleDrug Metabolism and Disposition December 2005, 33 (12) 1877-1885; DOI: https://doi.org/10.1124/dmd.105.005520
Kragh-Hansen, Ulrich
- You have accessHYDROLYSIS OF ANGIOTENSIN II RECEPTOR BLOCKER PRODRUG OLMESARTAN MEDOXOMIL BY HUMAN SERUM ALBUMIN AND IDENTIFICATION OF ITS CATALYTIC ACTIVE SITESShen-Feng Ma, Makoto Anraku, Yasunori Iwao, Keishi Yamasaki, Ulrich Kragh-Hansen, Noriyuki Yamaotsu, Shuichi Hirono, Toshihiko Ikeda and Masaki OtagiriDrug Metabolism and Disposition December 2005, 33 (12) 1911-1919; DOI: https://doi.org/10.1124/dmd.105.006163
Kunze, Kent L.
- You have accessOXIDATION OF CAFFEINE BY CYP1A2: ISOTOPE EFFECTS AND METABOLIC SWITCHINGKelly A. Regal, Kent L. Kunze, Raimund M. Peter and Sidney D. NelsonDrug Metabolism and Disposition December 2005, 33 (12) 1837-1844; DOI: https://doi.org/10.1124/dmd.105.006031
Kurian, Joseph R.
- You have accessUNUSUAL DEHYDROXYLATION OF ANTIMICROBIAL AMIDOXIME PRODRUGS BY CYTOCHROME b5 AND NADH CYTOCHROME b5 REDUCTASEJanelle Y. Saulter, Joseph R. Kurian, Lauren A. Trepanier, Richard R. Tidwell, Arlene S. Bridges, David W. Boykin, Chad E. Stephens, Mariappan Anbazhagan and James Edwin HallDrug Metabolism and Disposition December 2005, 33 (12) 1886-1893; DOI: https://doi.org/10.1124/dmd.105.005017
L
Lan, Lubin
- You have accessROLE OF THE NUCLEAR RECEPTOR PREGNANE X RECEPTOR IN ACETAMINOPHEN HEPATOTOXICITYKristina K. Wolf, Sheryl G. Wood, Jane A. Hunt, Brooke W. Walton-Strong, Kazuto Yasuda, Lubin Lan, Su X. Duan, Qin Hao, Steven A. Wrighton, Elizabeth H. Jeffery, Ronald M. Evans, Juliana G. Szakacs, Lisa L. von Moltke, David J. Greenblatt, Michael H. Court, Erin G. Schuetz, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition December 2005, 33 (12) 1827-1836; DOI: https://doi.org/10.1124/dmd.105.005256
Lee, Sang-Kwang
- You have accessMODULATION OF HUMAN CYTOCHROME P450 1B1 EXPRESSION BY 2,4,3′,5′-TETRAMETHOXYSTILBENEYoung-Jin Chun, Sang-Kwang Lee and Mie Young KimDrug Metabolism and Disposition December 2005, 33 (12) 1771-1776; DOI: https://doi.org/10.1124/dmd.105.006502
Leeder, J. Steven
- You have accessPATHWAYS OF CARBAMAZEPINE BIOACTIVATION IN VITRO: II. THE ROLE OF HUMAN CYTOCHROME P450 ENZYMES IN THE FORMATION OF 2-HYDROXYIMINOSTILBENERobin E. Pearce, Jack P. Uetrecht and J. Steven LeederDrug Metabolism and Disposition December 2005, 33 (12) 1819-1826; DOI: https://doi.org/10.1124/dmd.105.004861
Leo, Gregory C.
- You have accessBIOACTIVATION OF 4-METHYLPHENOL (p-CRESOL) VIA CYTOCHROME P450-MEDIATED AROMATIC OXIDATION IN HUMAN LIVER MICROSOMESZhengyin Yan, H. Marlon Zhong, Noureddine Maher, Rhoda Torres, Gregory C. Leo, Gary W. Caldwell and Norman HuebertDrug Metabolism and Disposition December 2005, 33 (12) 1867-1876; DOI: https://doi.org/10.1124/dmd.105.006387
Lidereau, Rosette
- You have accessSIMULTANEOUS MEASUREMENT OF 23 ISOFORMS FROM THE HUMAN CYTOCHROME P450 FAMILIES 1 TO 3 BY QUANTITATIVE REVERSE TRANSCRIPTASE-POLYMERASE CHAIN REACTIONIgor Girault, Nathalie Rougier, Christophe Chesné, Rosette Lidereau, Philippe Beaune, Ivan Bieche and Isabelle de WaziersDrug Metabolism and Disposition December 2005, 33 (12) 1803-1810; DOI: https://doi.org/10.1124/dmd.105.005173
Lin, Huimin
- You have accessDISPOSITION OF FLAVONOIDS VIA RECYCLING: COMPARISON OF INTESTINAL VERSUS HEPATIC DISPOSITIONJun Chen, Stephen Wang, Xiaobin Jia, Susan Bajimaya, Huimin Lin, Vincent H. Tam and Ming HuDrug Metabolism and Disposition December 2005, 33 (12) 1777-1784; DOI: https://doi.org/10.1124/dmd.105.003673
M
Ma, Bennett
- You have accessGLYCOSIDATION OF AN ENDOTHELIN ETA RECEPTOR ANTAGONIST AND DICLOFENAC IN HUMAN LIVER MICROSOMES: AGLYCONE-DEPENDENT UDP-SUGAR SELECTIVITYCuyue Tang and Bennett MaDrug Metabolism and Disposition December 2005, 33 (12) 1796-1802; DOI: https://doi.org/10.1124/dmd.105.005801
Ma, Shen-Feng
- You have accessHYDROLYSIS OF ANGIOTENSIN II RECEPTOR BLOCKER PRODRUG OLMESARTAN MEDOXOMIL BY HUMAN SERUM ALBUMIN AND IDENTIFICATION OF ITS CATALYTIC ACTIVE SITESShen-Feng Ma, Makoto Anraku, Yasunori Iwao, Keishi Yamasaki, Ulrich Kragh-Hansen, Noriyuki Yamaotsu, Shuichi Hirono, Toshihiko Ikeda and Masaki OtagiriDrug Metabolism and Disposition December 2005, 33 (12) 1911-1919; DOI: https://doi.org/10.1124/dmd.105.006163
Maeda, Tomoji
- You have accessINVOLVEMENT OF URIC ACID TRANSPORTER IN INCREASED RENAL CLEARANCE OF THE XANTHINE OXIDASE INHIBITOR OXYPURINOL INDUCED BY A URICOSURIC AGENT, BENZBROMARONETakashi Iwanaga, Daisuke Kobayashi, Masamichi Hirayama, Tomoji Maeda and Ikumi TamaiDrug Metabolism and Disposition December 2005, 33 (12) 1791-1795; DOI: https://doi.org/10.1124/dmd.105.006056
Maekawa, Keiko
- You have accessFUNCTIONAL ANALYSIS OF THREE CYP1A2 VARIANTS FOUND IN A JAPANESE POPULATIONYoshiro Saito, Nobumitsu Hanioka, Keiko Maekawa, Takashi Isobe, Yumi Tsuneto, Ryosuke Nakamura, Akiko Soyama, Shogo Ozawa, Toshiko Tanaka-Kagawa, Hideto Jinno, Shizuo Narimatsu and Jun-ichi SawadaDrug Metabolism and Disposition December 2005, 33 (12) 1905-1910; DOI: https://doi.org/10.1124/dmd.105.005819
Maher, Noureddine
- You have accessBIOACTIVATION OF 4-METHYLPHENOL (p-CRESOL) VIA CYTOCHROME P450-MEDIATED AROMATIC OXIDATION IN HUMAN LIVER MICROSOMESZhengyin Yan, H. Marlon Zhong, Noureddine Maher, Rhoda Torres, Gregory C. Leo, Gary W. Caldwell and Norman HuebertDrug Metabolism and Disposition December 2005, 33 (12) 1867-1876; DOI: https://doi.org/10.1124/dmd.105.006387
Mehendale, Harihara M.
- You have accessSATURATION TOXICOKINETICS OF THIOACETAMIDE: ROLE IN INITIATION OF LIVER INJURYJaya Chilakapati, Kartik Shankar, Midhun C. Korrapati, Ronald A. Hill and Harihara M. MehendaleDrug Metabolism and Disposition December 2005, 33 (12) 1877-1885; DOI: https://doi.org/10.1124/dmd.105.005520
Miya, Toshimichi
- You have accessGEFITINIB (IRESSA) INHIBITS THE CYP3A4-MEDIATED FORMATION OF 7-ETHYL-10-(4-AMINO-1-PIPERIDINO)CARBONYLOXYCAMPTOTHECIN BUT ACTIVATES THAT OF 7-ETHYL-10-[4-N-(5-AMINOPENTANOIC ACID)-1-PIPERIDINO]CARBONYLOXYCAMPTOTHECIN FROM IRINOTECANKen-ichi Fujita, Yuichi Ando, Masaru Narabayashi, Toshimichi Miya, Fumio Nagashima, Wataru Yamamoto, Keiji Kodama, Kazuhiro Araki, Hisashi Endo and Yasutsuna SasakiDrug Metabolism and Disposition December 2005, 33 (12) 1785-1790; DOI: https://doi.org/10.1124/dmd.105.006205
Murakami, Yuichi
- You have accessFUNCTIONAL CHARACTERIZATION OF HUMAN MONOCARBOXYLATE TRANSPORTER 6 (SLC16A5)Yuichi Murakami, Noriko Kohyama, Yasuna Kobayashi, Masayuki Ohbayashi, Hisakazu Ohtani, Yasufumi Sawada and Toshinori YamamotoDrug Metabolism and Disposition December 2005, 33 (12) 1845-1851; DOI: https://doi.org/10.1124/dmd.105.005264
Murphy, Sharon E.
- You have accessNICOTINE AND 4-(METHYLNITROSAMINO)-1-(3-PYRIDYL)-BUTANONE METABOLISM BY CYTOCHROME P450 2B6Kari E. Dicke, Sara M. Skrlin and Sharon E. MurphyDrug Metabolism and Disposition December 2005, 33 (12) 1760-1764; DOI: https://doi.org/10.1124/dmd.105.006718
N
Nagashima, Fumio
- You have accessGEFITINIB (IRESSA) INHIBITS THE CYP3A4-MEDIATED FORMATION OF 7-ETHYL-10-(4-AMINO-1-PIPERIDINO)CARBONYLOXYCAMPTOTHECIN BUT ACTIVATES THAT OF 7-ETHYL-10-[4-N-(5-AMINOPENTANOIC ACID)-1-PIPERIDINO]CARBONYLOXYCAMPTOTHECIN FROM IRINOTECANKen-ichi Fujita, Yuichi Ando, Masaru Narabayashi, Toshimichi Miya, Fumio Nagashima, Wataru Yamamoto, Keiji Kodama, Kazuhiro Araki, Hisashi Endo and Yasutsuna SasakiDrug Metabolism and Disposition December 2005, 33 (12) 1785-1790; DOI: https://doi.org/10.1124/dmd.105.006205
Nakajima, Miki
- You have accessCYP2A6 AND CYP2B6 ARE INVOLVED IN NORNICOTINE FORMATION FROM NICOTINE IN HUMANS: INTERINDIVIDUAL DIFFERENCES IN THESE CONTRIBUTIONSHiroyuki Yamanaka, Miki Nakajima, Tatsuki Fukami, Haruko Sakai, Akiko Nakamura, Miki Katoh, Masataka Takamiya, Yasuhiro Aoki and Tsuyoshi YokoiDrug Metabolism and Disposition December 2005, 33 (12) 1811-1818; DOI: https://doi.org/10.1124/dmd.105.006254
Nakamura, Akiko
- You have accessCYP2A6 AND CYP2B6 ARE INVOLVED IN NORNICOTINE FORMATION FROM NICOTINE IN HUMANS: INTERINDIVIDUAL DIFFERENCES IN THESE CONTRIBUTIONSHiroyuki Yamanaka, Miki Nakajima, Tatsuki Fukami, Haruko Sakai, Akiko Nakamura, Miki Katoh, Masataka Takamiya, Yasuhiro Aoki and Tsuyoshi YokoiDrug Metabolism and Disposition December 2005, 33 (12) 1811-1818; DOI: https://doi.org/10.1124/dmd.105.006254
Nakamura, Ryosuke
- You have accessFUNCTIONAL ANALYSIS OF THREE CYP1A2 VARIANTS FOUND IN A JAPANESE POPULATIONYoshiro Saito, Nobumitsu Hanioka, Keiko Maekawa, Takashi Isobe, Yumi Tsuneto, Ryosuke Nakamura, Akiko Soyama, Shogo Ozawa, Toshiko Tanaka-Kagawa, Hideto Jinno, Shizuo Narimatsu and Jun-ichi SawadaDrug Metabolism and Disposition December 2005, 33 (12) 1905-1910; DOI: https://doi.org/10.1124/dmd.105.005819
Narabayashi, Masaru
- You have accessGEFITINIB (IRESSA) INHIBITS THE CYP3A4-MEDIATED FORMATION OF 7-ETHYL-10-(4-AMINO-1-PIPERIDINO)CARBONYLOXYCAMPTOTHECIN BUT ACTIVATES THAT OF 7-ETHYL-10-[4-N-(5-AMINOPENTANOIC ACID)-1-PIPERIDINO]CARBONYLOXYCAMPTOTHECIN FROM IRINOTECANKen-ichi Fujita, Yuichi Ando, Masaru Narabayashi, Toshimichi Miya, Fumio Nagashima, Wataru Yamamoto, Keiji Kodama, Kazuhiro Araki, Hisashi Endo and Yasutsuna SasakiDrug Metabolism and Disposition December 2005, 33 (12) 1785-1790; DOI: https://doi.org/10.1124/dmd.105.006205
Narimatsu, Shizuo
- You have accessFUNCTIONAL ANALYSIS OF THREE CYP1A2 VARIANTS FOUND IN A JAPANESE POPULATIONYoshiro Saito, Nobumitsu Hanioka, Keiko Maekawa, Takashi Isobe, Yumi Tsuneto, Ryosuke Nakamura, Akiko Soyama, Shogo Ozawa, Toshiko Tanaka-Kagawa, Hideto Jinno, Shizuo Narimatsu and Jun-ichi SawadaDrug Metabolism and Disposition December 2005, 33 (12) 1905-1910; DOI: https://doi.org/10.1124/dmd.105.005819
Nelson, Sidney D.
- You have accessOXIDATION OF CAFFEINE BY CYP1A2: ISOTOPE EFFECTS AND METABOLIC SWITCHINGKelly A. Regal, Kent L. Kunze, Raimund M. Peter and Sidney D. NelsonDrug Metabolism and Disposition December 2005, 33 (12) 1837-1844; DOI: https://doi.org/10.1124/dmd.105.006031
O
Ohbayashi, Masayuki
- You have accessFUNCTIONAL CHARACTERIZATION OF HUMAN MONOCARBOXYLATE TRANSPORTER 6 (SLC16A5)Yuichi Murakami, Noriko Kohyama, Yasuna Kobayashi, Masayuki Ohbayashi, Hisakazu Ohtani, Yasufumi Sawada and Toshinori YamamotoDrug Metabolism and Disposition December 2005, 33 (12) 1845-1851; DOI: https://doi.org/10.1124/dmd.105.005264
Ohtani, Hisakazu
- You have accessFUNCTIONAL CHARACTERIZATION OF HUMAN MONOCARBOXYLATE TRANSPORTER 6 (SLC16A5)Yuichi Murakami, Noriko Kohyama, Yasuna Kobayashi, Masayuki Ohbayashi, Hisakazu Ohtani, Yasufumi Sawada and Toshinori YamamotoDrug Metabolism and Disposition December 2005, 33 (12) 1845-1851; DOI: https://doi.org/10.1124/dmd.105.005264
Otagiri, Masaki
- You have accessHYDROLYSIS OF ANGIOTENSIN II RECEPTOR BLOCKER PRODRUG OLMESARTAN MEDOXOMIL BY HUMAN SERUM ALBUMIN AND IDENTIFICATION OF ITS CATALYTIC ACTIVE SITESShen-Feng Ma, Makoto Anraku, Yasunori Iwao, Keishi Yamasaki, Ulrich Kragh-Hansen, Noriyuki Yamaotsu, Shuichi Hirono, Toshihiko Ikeda and Masaki OtagiriDrug Metabolism and Disposition December 2005, 33 (12) 1911-1919; DOI: https://doi.org/10.1124/dmd.105.006163
Ozawa, Shogo
- You have accessFUNCTIONAL ANALYSIS OF THREE CYP1A2 VARIANTS FOUND IN A JAPANESE POPULATIONYoshiro Saito, Nobumitsu Hanioka, Keiko Maekawa, Takashi Isobe, Yumi Tsuneto, Ryosuke Nakamura, Akiko Soyama, Shogo Ozawa, Toshiko Tanaka-Kagawa, Hideto Jinno, Shizuo Narimatsu and Jun-ichi SawadaDrug Metabolism and Disposition December 2005, 33 (12) 1905-1910; DOI: https://doi.org/10.1124/dmd.105.005819
P
Pearce, Robin E.
- You have accessPATHWAYS OF CARBAMAZEPINE BIOACTIVATION IN VITRO: II. THE ROLE OF HUMAN CYTOCHROME P450 ENZYMES IN THE FORMATION OF 2-HYDROXYIMINOSTILBENERobin E. Pearce, Jack P. Uetrecht and J. Steven LeederDrug Metabolism and Disposition December 2005, 33 (12) 1819-1826; DOI: https://doi.org/10.1124/dmd.105.004861
Peter, Raimund M.
- You have accessOXIDATION OF CAFFEINE BY CYP1A2: ISOTOPE EFFECTS AND METABOLIC SWITCHINGKelly A. Regal, Kent L. Kunze, Raimund M. Peter and Sidney D. NelsonDrug Metabolism and Disposition December 2005, 33 (12) 1837-1844; DOI: https://doi.org/10.1124/dmd.105.006031
Pool, William F.
- You have accessHUMAN IN VITRO GLUTATHIONYL AND PROTEIN ADDUCTS OF CARBAMAZEPINE-10,11-EPOXIDE, A STABLE AND PHARMACOLOGICALLY ACTIVE METABOLITE OF CARBAMAZEPINEHai-Zhi Bu, Ping Kang, Alan J. Deese, Ping Zhao and William F. PoolDrug Metabolism and Disposition December 2005, 33 (12) 1920-1924; DOI: https://doi.org/10.1124/dmd.105.006866
R
Rankin, Gary O.
- You have accessTRANSAMINATION IN THE METABOLISM OF THE NEPHROTOXICANT N-(3,5-DICHLOROPHENYL)SUCCINIMIDE IN RATSDonghui Cui, Gary O. Rankin and Peter J. HarvisonDrug Metabolism and Disposition December 2005, 33 (12) 1765-1770; DOI: https://doi.org/10.1124/dmd.105.006593
Rawden, Helen C.
- You have accessPREDICTION OF METABOLIC CLEARANCE USING CRYOPRESERVED HUMAN HEPATOCYTES: KINETIC CHARACTERISTICS FOR FIVE BENZODIAZEPINESDavid Hallifax, Helen C. Rawden, Nancy Hakooz and J. Brian HoustonDrug Metabolism and Disposition December 2005, 33 (12) 1852-1858; DOI: https://doi.org/10.1124/dmd.105.005389
Reed, James R.
- You have accessSPECIES DIFFERENCES IN THE ELIMINATION OF A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR AGONIST HIGHLIGHTED BY OXIDATIVE METABOLISM OF ITS ACYL GLUCURONIDEChristopher J. Kochansky, Yuan-Qing Xia, Sui Wang, Brian Cato, Mellissa Creighton, Stella H. Vincent, Ronald B. Franklin and James R. ReedDrug Metabolism and Disposition December 2005, 33 (12) 1894-1904; DOI: https://doi.org/10.1124/dmd.105.004010
Regal, Kelly A.
- You have accessOXIDATION OF CAFFEINE BY CYP1A2: ISOTOPE EFFECTS AND METABOLIC SWITCHINGKelly A. Regal, Kent L. Kunze, Raimund M. Peter and Sidney D. NelsonDrug Metabolism and Disposition December 2005, 33 (12) 1837-1844; DOI: https://doi.org/10.1124/dmd.105.006031
Richter, K.
- You have accessEFFECT OF PROPIVERINE ON CYTOCHROME P450 ENZYMES: A COCKTAIL INTERACTION STUDY IN HEALTHY VOLUNTEERSD. Tomalik-Scharte, A. Jetter, M. Kinzig-Schippers, A. Skott, F. Sörgel, T. Klaassen, D. Kasel, S. Harlfinger, O. Doroshyenko, D. Frank, J. Kirchheiner, M. Bräter, K. Richter, T. Gramatté and U. FuhrDrug Metabolism and Disposition December 2005, 33 (12) 1859-1866; DOI: https://doi.org/10.1124/dmd.105.005272
Rougier, Nathalie
- You have accessSIMULTANEOUS MEASUREMENT OF 23 ISOFORMS FROM THE HUMAN CYTOCHROME P450 FAMILIES 1 TO 3 BY QUANTITATIVE REVERSE TRANSCRIPTASE-POLYMERASE CHAIN REACTIONIgor Girault, Nathalie Rougier, Christophe Chesné, Rosette Lidereau, Philippe Beaune, Ivan Bieche and Isabelle de WaziersDrug Metabolism and Disposition December 2005, 33 (12) 1803-1810; DOI: https://doi.org/10.1124/dmd.105.005173
S
Saito, Yoshiro
- You have accessFUNCTIONAL ANALYSIS OF THREE CYP1A2 VARIANTS FOUND IN A JAPANESE POPULATIONYoshiro Saito, Nobumitsu Hanioka, Keiko Maekawa, Takashi Isobe, Yumi Tsuneto, Ryosuke Nakamura, Akiko Soyama, Shogo Ozawa, Toshiko Tanaka-Kagawa, Hideto Jinno, Shizuo Narimatsu and Jun-ichi SawadaDrug Metabolism and Disposition December 2005, 33 (12) 1905-1910; DOI: https://doi.org/10.1124/dmd.105.005819
Sakai, Haruko
- You have accessCYP2A6 AND CYP2B6 ARE INVOLVED IN NORNICOTINE FORMATION FROM NICOTINE IN HUMANS: INTERINDIVIDUAL DIFFERENCES IN THESE CONTRIBUTIONSHiroyuki Yamanaka, Miki Nakajima, Tatsuki Fukami, Haruko Sakai, Akiko Nakamura, Miki Katoh, Masataka Takamiya, Yasuhiro Aoki and Tsuyoshi YokoiDrug Metabolism and Disposition December 2005, 33 (12) 1811-1818; DOI: https://doi.org/10.1124/dmd.105.006254
Sasaki, Yasutsuna
- You have accessGEFITINIB (IRESSA) INHIBITS THE CYP3A4-MEDIATED FORMATION OF 7-ETHYL-10-(4-AMINO-1-PIPERIDINO)CARBONYLOXYCAMPTOTHECIN BUT ACTIVATES THAT OF 7-ETHYL-10-[4-N-(5-AMINOPENTANOIC ACID)-1-PIPERIDINO]CARBONYLOXYCAMPTOTHECIN FROM IRINOTECANKen-ichi Fujita, Yuichi Ando, Masaru Narabayashi, Toshimichi Miya, Fumio Nagashima, Wataru Yamamoto, Keiji Kodama, Kazuhiro Araki, Hisashi Endo and Yasutsuna SasakiDrug Metabolism and Disposition December 2005, 33 (12) 1785-1790; DOI: https://doi.org/10.1124/dmd.105.006205
Saulter, Janelle Y.
- You have accessUNUSUAL DEHYDROXYLATION OF ANTIMICROBIAL AMIDOXIME PRODRUGS BY CYTOCHROME b5 AND NADH CYTOCHROME b5 REDUCTASEJanelle Y. Saulter, Joseph R. Kurian, Lauren A. Trepanier, Richard R. Tidwell, Arlene S. Bridges, David W. Boykin, Chad E. Stephens, Mariappan Anbazhagan and James Edwin HallDrug Metabolism and Disposition December 2005, 33 (12) 1886-1893; DOI: https://doi.org/10.1124/dmd.105.005017
Sawada, Jun-ichi
- You have accessFUNCTIONAL ANALYSIS OF THREE CYP1A2 VARIANTS FOUND IN A JAPANESE POPULATIONYoshiro Saito, Nobumitsu Hanioka, Keiko Maekawa, Takashi Isobe, Yumi Tsuneto, Ryosuke Nakamura, Akiko Soyama, Shogo Ozawa, Toshiko Tanaka-Kagawa, Hideto Jinno, Shizuo Narimatsu and Jun-ichi SawadaDrug Metabolism and Disposition December 2005, 33 (12) 1905-1910; DOI: https://doi.org/10.1124/dmd.105.005819
Sawada, Yasufumi
- You have accessFUNCTIONAL CHARACTERIZATION OF HUMAN MONOCARBOXYLATE TRANSPORTER 6 (SLC16A5)Yuichi Murakami, Noriko Kohyama, Yasuna Kobayashi, Masayuki Ohbayashi, Hisakazu Ohtani, Yasufumi Sawada and Toshinori YamamotoDrug Metabolism and Disposition December 2005, 33 (12) 1845-1851; DOI: https://doi.org/10.1124/dmd.105.005264
Schuetz, Erin G.
- You have accessROLE OF THE NUCLEAR RECEPTOR PREGNANE X RECEPTOR IN ACETAMINOPHEN HEPATOTOXICITYKristina K. Wolf, Sheryl G. Wood, Jane A. Hunt, Brooke W. Walton-Strong, Kazuto Yasuda, Lubin Lan, Su X. Duan, Qin Hao, Steven A. Wrighton, Elizabeth H. Jeffery, Ronald M. Evans, Juliana G. Szakacs, Lisa L. von Moltke, David J. Greenblatt, Michael H. Court, Erin G. Schuetz, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition December 2005, 33 (12) 1827-1836; DOI: https://doi.org/10.1124/dmd.105.005256
Shankar, Kartik
- You have accessSATURATION TOXICOKINETICS OF THIOACETAMIDE: ROLE IN INITIATION OF LIVER INJURYJaya Chilakapati, Kartik Shankar, Midhun C. Korrapati, Ronald A. Hill and Harihara M. MehendaleDrug Metabolism and Disposition December 2005, 33 (12) 1877-1885; DOI: https://doi.org/10.1124/dmd.105.005520
Sinclair, Jacqueline F.
- You have accessROLE OF THE NUCLEAR RECEPTOR PREGNANE X RECEPTOR IN ACETAMINOPHEN HEPATOTOXICITYKristina K. Wolf, Sheryl G. Wood, Jane A. Hunt, Brooke W. Walton-Strong, Kazuto Yasuda, Lubin Lan, Su X. Duan, Qin Hao, Steven A. Wrighton, Elizabeth H. Jeffery, Ronald M. Evans, Juliana G. Szakacs, Lisa L. von Moltke, David J. Greenblatt, Michael H. Court, Erin G. Schuetz, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition December 2005, 33 (12) 1827-1836; DOI: https://doi.org/10.1124/dmd.105.005256
Sinclair, Peter R.
- You have accessROLE OF THE NUCLEAR RECEPTOR PREGNANE X RECEPTOR IN ACETAMINOPHEN HEPATOTOXICITYKristina K. Wolf, Sheryl G. Wood, Jane A. Hunt, Brooke W. Walton-Strong, Kazuto Yasuda, Lubin Lan, Su X. Duan, Qin Hao, Steven A. Wrighton, Elizabeth H. Jeffery, Ronald M. Evans, Juliana G. Szakacs, Lisa L. von Moltke, David J. Greenblatt, Michael H. Court, Erin G. Schuetz, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition December 2005, 33 (12) 1827-1836; DOI: https://doi.org/10.1124/dmd.105.005256
Skott, A.
- You have accessEFFECT OF PROPIVERINE ON CYTOCHROME P450 ENZYMES: A COCKTAIL INTERACTION STUDY IN HEALTHY VOLUNTEERSD. Tomalik-Scharte, A. Jetter, M. Kinzig-Schippers, A. Skott, F. Sörgel, T. Klaassen, D. Kasel, S. Harlfinger, O. Doroshyenko, D. Frank, J. Kirchheiner, M. Bräter, K. Richter, T. Gramatté and U. FuhrDrug Metabolism and Disposition December 2005, 33 (12) 1859-1866; DOI: https://doi.org/10.1124/dmd.105.005272
Skrlin, Sara M.
- You have accessNICOTINE AND 4-(METHYLNITROSAMINO)-1-(3-PYRIDYL)-BUTANONE METABOLISM BY CYTOCHROME P450 2B6Kari E. Dicke, Sara M. Skrlin and Sharon E. MurphyDrug Metabolism and Disposition December 2005, 33 (12) 1760-1764; DOI: https://doi.org/10.1124/dmd.105.006718
Sörgel, F.
- You have accessEFFECT OF PROPIVERINE ON CYTOCHROME P450 ENZYMES: A COCKTAIL INTERACTION STUDY IN HEALTHY VOLUNTEERSD. Tomalik-Scharte, A. Jetter, M. Kinzig-Schippers, A. Skott, F. Sörgel, T. Klaassen, D. Kasel, S. Harlfinger, O. Doroshyenko, D. Frank, J. Kirchheiner, M. Bräter, K. Richter, T. Gramatté and U. FuhrDrug Metabolism and Disposition December 2005, 33 (12) 1859-1866; DOI: https://doi.org/10.1124/dmd.105.005272
Soyama, Akiko
- You have accessFUNCTIONAL ANALYSIS OF THREE CYP1A2 VARIANTS FOUND IN A JAPANESE POPULATIONYoshiro Saito, Nobumitsu Hanioka, Keiko Maekawa, Takashi Isobe, Yumi Tsuneto, Ryosuke Nakamura, Akiko Soyama, Shogo Ozawa, Toshiko Tanaka-Kagawa, Hideto Jinno, Shizuo Narimatsu and Jun-ichi SawadaDrug Metabolism and Disposition December 2005, 33 (12) 1905-1910; DOI: https://doi.org/10.1124/dmd.105.005819
Stephens, Chad E.
- You have accessUNUSUAL DEHYDROXYLATION OF ANTIMICROBIAL AMIDOXIME PRODRUGS BY CYTOCHROME b5 AND NADH CYTOCHROME b5 REDUCTASEJanelle Y. Saulter, Joseph R. Kurian, Lauren A. Trepanier, Richard R. Tidwell, Arlene S. Bridges, David W. Boykin, Chad E. Stephens, Mariappan Anbazhagan and James Edwin HallDrug Metabolism and Disposition December 2005, 33 (12) 1886-1893; DOI: https://doi.org/10.1124/dmd.105.005017
Szakacs, Juliana G.
- You have accessROLE OF THE NUCLEAR RECEPTOR PREGNANE X RECEPTOR IN ACETAMINOPHEN HEPATOTOXICITYKristina K. Wolf, Sheryl G. Wood, Jane A. Hunt, Brooke W. Walton-Strong, Kazuto Yasuda, Lubin Lan, Su X. Duan, Qin Hao, Steven A. Wrighton, Elizabeth H. Jeffery, Ronald M. Evans, Juliana G. Szakacs, Lisa L. von Moltke, David J. Greenblatt, Michael H. Court, Erin G. Schuetz, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition December 2005, 33 (12) 1827-1836; DOI: https://doi.org/10.1124/dmd.105.005256
T
Takamiya, Masataka
- You have accessCYP2A6 AND CYP2B6 ARE INVOLVED IN NORNICOTINE FORMATION FROM NICOTINE IN HUMANS: INTERINDIVIDUAL DIFFERENCES IN THESE CONTRIBUTIONSHiroyuki Yamanaka, Miki Nakajima, Tatsuki Fukami, Haruko Sakai, Akiko Nakamura, Miki Katoh, Masataka Takamiya, Yasuhiro Aoki and Tsuyoshi YokoiDrug Metabolism and Disposition December 2005, 33 (12) 1811-1818; DOI: https://doi.org/10.1124/dmd.105.006254
Tam, Vincent H.
- You have accessDISPOSITION OF FLAVONOIDS VIA RECYCLING: COMPARISON OF INTESTINAL VERSUS HEPATIC DISPOSITIONJun Chen, Stephen Wang, Xiaobin Jia, Susan Bajimaya, Huimin Lin, Vincent H. Tam and Ming HuDrug Metabolism and Disposition December 2005, 33 (12) 1777-1784; DOI: https://doi.org/10.1124/dmd.105.003673
Tamai, Ikumi
- You have accessINVOLVEMENT OF URIC ACID TRANSPORTER IN INCREASED RENAL CLEARANCE OF THE XANTHINE OXIDASE INHIBITOR OXYPURINOL INDUCED BY A URICOSURIC AGENT, BENZBROMARONETakashi Iwanaga, Daisuke Kobayashi, Masamichi Hirayama, Tomoji Maeda and Ikumi TamaiDrug Metabolism and Disposition December 2005, 33 (12) 1791-1795; DOI: https://doi.org/10.1124/dmd.105.006056
Tanaka-Kagawa, Toshiko
- You have accessFUNCTIONAL ANALYSIS OF THREE CYP1A2 VARIANTS FOUND IN A JAPANESE POPULATIONYoshiro Saito, Nobumitsu Hanioka, Keiko Maekawa, Takashi Isobe, Yumi Tsuneto, Ryosuke Nakamura, Akiko Soyama, Shogo Ozawa, Toshiko Tanaka-Kagawa, Hideto Jinno, Shizuo Narimatsu and Jun-ichi SawadaDrug Metabolism and Disposition December 2005, 33 (12) 1905-1910; DOI: https://doi.org/10.1124/dmd.105.005819
Tang, Cuyue
- You have accessGLYCOSIDATION OF AN ENDOTHELIN ETA RECEPTOR ANTAGONIST AND DICLOFENAC IN HUMAN LIVER MICROSOMES: AGLYCONE-DEPENDENT UDP-SUGAR SELECTIVITYCuyue Tang and Bennett MaDrug Metabolism and Disposition December 2005, 33 (12) 1796-1802; DOI: https://doi.org/10.1124/dmd.105.005801
Tidwell, Richard R.
- You have accessUNUSUAL DEHYDROXYLATION OF ANTIMICROBIAL AMIDOXIME PRODRUGS BY CYTOCHROME b5 AND NADH CYTOCHROME b5 REDUCTASEJanelle Y. Saulter, Joseph R. Kurian, Lauren A. Trepanier, Richard R. Tidwell, Arlene S. Bridges, David W. Boykin, Chad E. Stephens, Mariappan Anbazhagan and James Edwin HallDrug Metabolism and Disposition December 2005, 33 (12) 1886-1893; DOI: https://doi.org/10.1124/dmd.105.005017
Tomalik-Scharte, D.
- You have accessEFFECT OF PROPIVERINE ON CYTOCHROME P450 ENZYMES: A COCKTAIL INTERACTION STUDY IN HEALTHY VOLUNTEERSD. Tomalik-Scharte, A. Jetter, M. Kinzig-Schippers, A. Skott, F. Sörgel, T. Klaassen, D. Kasel, S. Harlfinger, O. Doroshyenko, D. Frank, J. Kirchheiner, M. Bräter, K. Richter, T. Gramatté and U. FuhrDrug Metabolism and Disposition December 2005, 33 (12) 1859-1866; DOI: https://doi.org/10.1124/dmd.105.005272
Torres, Rhoda
- You have accessBIOACTIVATION OF 4-METHYLPHENOL (p-CRESOL) VIA CYTOCHROME P450-MEDIATED AROMATIC OXIDATION IN HUMAN LIVER MICROSOMESZhengyin Yan, H. Marlon Zhong, Noureddine Maher, Rhoda Torres, Gregory C. Leo, Gary W. Caldwell and Norman HuebertDrug Metabolism and Disposition December 2005, 33 (12) 1867-1876; DOI: https://doi.org/10.1124/dmd.105.006387
Trepanier, Lauren A.
- You have accessUNUSUAL DEHYDROXYLATION OF ANTIMICROBIAL AMIDOXIME PRODRUGS BY CYTOCHROME b5 AND NADH CYTOCHROME b5 REDUCTASEJanelle Y. Saulter, Joseph R. Kurian, Lauren A. Trepanier, Richard R. Tidwell, Arlene S. Bridges, David W. Boykin, Chad E. Stephens, Mariappan Anbazhagan and James Edwin HallDrug Metabolism and Disposition December 2005, 33 (12) 1886-1893; DOI: https://doi.org/10.1124/dmd.105.005017
Tsuneto, Yumi
- You have accessFUNCTIONAL ANALYSIS OF THREE CYP1A2 VARIANTS FOUND IN A JAPANESE POPULATIONYoshiro Saito, Nobumitsu Hanioka, Keiko Maekawa, Takashi Isobe, Yumi Tsuneto, Ryosuke Nakamura, Akiko Soyama, Shogo Ozawa, Toshiko Tanaka-Kagawa, Hideto Jinno, Shizuo Narimatsu and Jun-ichi SawadaDrug Metabolism and Disposition December 2005, 33 (12) 1905-1910; DOI: https://doi.org/10.1124/dmd.105.005819
U
Uetrecht, Jack P.
- You have accessPATHWAYS OF CARBAMAZEPINE BIOACTIVATION IN VITRO: II. THE ROLE OF HUMAN CYTOCHROME P450 ENZYMES IN THE FORMATION OF 2-HYDROXYIMINOSTILBENERobin E. Pearce, Jack P. Uetrecht and J. Steven LeederDrug Metabolism and Disposition December 2005, 33 (12) 1819-1826; DOI: https://doi.org/10.1124/dmd.105.004861
V
Vincent, Stella H.
- You have accessSPECIES DIFFERENCES IN THE ELIMINATION OF A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR AGONIST HIGHLIGHTED BY OXIDATIVE METABOLISM OF ITS ACYL GLUCURONIDEChristopher J. Kochansky, Yuan-Qing Xia, Sui Wang, Brian Cato, Mellissa Creighton, Stella H. Vincent, Ronald B. Franklin and James R. ReedDrug Metabolism and Disposition December 2005, 33 (12) 1894-1904; DOI: https://doi.org/10.1124/dmd.105.004010
von Moltke, Lisa L.
- You have accessROLE OF THE NUCLEAR RECEPTOR PREGNANE X RECEPTOR IN ACETAMINOPHEN HEPATOTOXICITYKristina K. Wolf, Sheryl G. Wood, Jane A. Hunt, Brooke W. Walton-Strong, Kazuto Yasuda, Lubin Lan, Su X. Duan, Qin Hao, Steven A. Wrighton, Elizabeth H. Jeffery, Ronald M. Evans, Juliana G. Szakacs, Lisa L. von Moltke, David J. Greenblatt, Michael H. Court, Erin G. Schuetz, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition December 2005, 33 (12) 1827-1836; DOI: https://doi.org/10.1124/dmd.105.005256
W
Walton-Strong, Brooke W.
- You have accessROLE OF THE NUCLEAR RECEPTOR PREGNANE X RECEPTOR IN ACETAMINOPHEN HEPATOTOXICITYKristina K. Wolf, Sheryl G. Wood, Jane A. Hunt, Brooke W. Walton-Strong, Kazuto Yasuda, Lubin Lan, Su X. Duan, Qin Hao, Steven A. Wrighton, Elizabeth H. Jeffery, Ronald M. Evans, Juliana G. Szakacs, Lisa L. von Moltke, David J. Greenblatt, Michael H. Court, Erin G. Schuetz, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition December 2005, 33 (12) 1827-1836; DOI: https://doi.org/10.1124/dmd.105.005256
Wang, Stephen
- You have accessDISPOSITION OF FLAVONOIDS VIA RECYCLING: COMPARISON OF INTESTINAL VERSUS HEPATIC DISPOSITIONJun Chen, Stephen Wang, Xiaobin Jia, Susan Bajimaya, Huimin Lin, Vincent H. Tam and Ming HuDrug Metabolism and Disposition December 2005, 33 (12) 1777-1784; DOI: https://doi.org/10.1124/dmd.105.003673
Wang, Sui
- You have accessSPECIES DIFFERENCES IN THE ELIMINATION OF A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR AGONIST HIGHLIGHTED BY OXIDATIVE METABOLISM OF ITS ACYL GLUCURONIDEChristopher J. Kochansky, Yuan-Qing Xia, Sui Wang, Brian Cato, Mellissa Creighton, Stella H. Vincent, Ronald B. Franklin and James R. ReedDrug Metabolism and Disposition December 2005, 33 (12) 1894-1904; DOI: https://doi.org/10.1124/dmd.105.004010
Wolf, Kristina K.
- You have accessROLE OF THE NUCLEAR RECEPTOR PREGNANE X RECEPTOR IN ACETAMINOPHEN HEPATOTOXICITYKristina K. Wolf, Sheryl G. Wood, Jane A. Hunt, Brooke W. Walton-Strong, Kazuto Yasuda, Lubin Lan, Su X. Duan, Qin Hao, Steven A. Wrighton, Elizabeth H. Jeffery, Ronald M. Evans, Juliana G. Szakacs, Lisa L. von Moltke, David J. Greenblatt, Michael H. Court, Erin G. Schuetz, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition December 2005, 33 (12) 1827-1836; DOI: https://doi.org/10.1124/dmd.105.005256
Wood, Sheryl G.
- You have accessROLE OF THE NUCLEAR RECEPTOR PREGNANE X RECEPTOR IN ACETAMINOPHEN HEPATOTOXICITYKristina K. Wolf, Sheryl G. Wood, Jane A. Hunt, Brooke W. Walton-Strong, Kazuto Yasuda, Lubin Lan, Su X. Duan, Qin Hao, Steven A. Wrighton, Elizabeth H. Jeffery, Ronald M. Evans, Juliana G. Szakacs, Lisa L. von Moltke, David J. Greenblatt, Michael H. Court, Erin G. Schuetz, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition December 2005, 33 (12) 1827-1836; DOI: https://doi.org/10.1124/dmd.105.005256
Wrighton, Steven A.
- You have accessROLE OF THE NUCLEAR RECEPTOR PREGNANE X RECEPTOR IN ACETAMINOPHEN HEPATOTOXICITYKristina K. Wolf, Sheryl G. Wood, Jane A. Hunt, Brooke W. Walton-Strong, Kazuto Yasuda, Lubin Lan, Su X. Duan, Qin Hao, Steven A. Wrighton, Elizabeth H. Jeffery, Ronald M. Evans, Juliana G. Szakacs, Lisa L. von Moltke, David J. Greenblatt, Michael H. Court, Erin G. Schuetz, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition December 2005, 33 (12) 1827-1836; DOI: https://doi.org/10.1124/dmd.105.005256
X
Xia, Yuan-Qing
- You have accessSPECIES DIFFERENCES IN THE ELIMINATION OF A PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR AGONIST HIGHLIGHTED BY OXIDATIVE METABOLISM OF ITS ACYL GLUCURONIDEChristopher J. Kochansky, Yuan-Qing Xia, Sui Wang, Brian Cato, Mellissa Creighton, Stella H. Vincent, Ronald B. Franklin and James R. ReedDrug Metabolism and Disposition December 2005, 33 (12) 1894-1904; DOI: https://doi.org/10.1124/dmd.105.004010
Y
Yamamoto, Toshinori
- You have accessFUNCTIONAL CHARACTERIZATION OF HUMAN MONOCARBOXYLATE TRANSPORTER 6 (SLC16A5)Yuichi Murakami, Noriko Kohyama, Yasuna Kobayashi, Masayuki Ohbayashi, Hisakazu Ohtani, Yasufumi Sawada and Toshinori YamamotoDrug Metabolism and Disposition December 2005, 33 (12) 1845-1851; DOI: https://doi.org/10.1124/dmd.105.005264
Yamamoto, Wataru
- You have accessGEFITINIB (IRESSA) INHIBITS THE CYP3A4-MEDIATED FORMATION OF 7-ETHYL-10-(4-AMINO-1-PIPERIDINO)CARBONYLOXYCAMPTOTHECIN BUT ACTIVATES THAT OF 7-ETHYL-10-[4-N-(5-AMINOPENTANOIC ACID)-1-PIPERIDINO]CARBONYLOXYCAMPTOTHECIN FROM IRINOTECANKen-ichi Fujita, Yuichi Ando, Masaru Narabayashi, Toshimichi Miya, Fumio Nagashima, Wataru Yamamoto, Keiji Kodama, Kazuhiro Araki, Hisashi Endo and Yasutsuna SasakiDrug Metabolism and Disposition December 2005, 33 (12) 1785-1790; DOI: https://doi.org/10.1124/dmd.105.006205
Yamanaka, Hiroyuki
- You have accessCYP2A6 AND CYP2B6 ARE INVOLVED IN NORNICOTINE FORMATION FROM NICOTINE IN HUMANS: INTERINDIVIDUAL DIFFERENCES IN THESE CONTRIBUTIONSHiroyuki Yamanaka, Miki Nakajima, Tatsuki Fukami, Haruko Sakai, Akiko Nakamura, Miki Katoh, Masataka Takamiya, Yasuhiro Aoki and Tsuyoshi YokoiDrug Metabolism and Disposition December 2005, 33 (12) 1811-1818; DOI: https://doi.org/10.1124/dmd.105.006254
Yamaotsu, Noriyuki
- You have accessHYDROLYSIS OF ANGIOTENSIN II RECEPTOR BLOCKER PRODRUG OLMESARTAN MEDOXOMIL BY HUMAN SERUM ALBUMIN AND IDENTIFICATION OF ITS CATALYTIC ACTIVE SITESShen-Feng Ma, Makoto Anraku, Yasunori Iwao, Keishi Yamasaki, Ulrich Kragh-Hansen, Noriyuki Yamaotsu, Shuichi Hirono, Toshihiko Ikeda and Masaki OtagiriDrug Metabolism and Disposition December 2005, 33 (12) 1911-1919; DOI: https://doi.org/10.1124/dmd.105.006163
Yamasaki, Keishi
- You have accessHYDROLYSIS OF ANGIOTENSIN II RECEPTOR BLOCKER PRODRUG OLMESARTAN MEDOXOMIL BY HUMAN SERUM ALBUMIN AND IDENTIFICATION OF ITS CATALYTIC ACTIVE SITESShen-Feng Ma, Makoto Anraku, Yasunori Iwao, Keishi Yamasaki, Ulrich Kragh-Hansen, Noriyuki Yamaotsu, Shuichi Hirono, Toshihiko Ikeda and Masaki OtagiriDrug Metabolism and Disposition December 2005, 33 (12) 1911-1919; DOI: https://doi.org/10.1124/dmd.105.006163
Yan, Zhengyin
- You have accessBIOACTIVATION OF 4-METHYLPHENOL (p-CRESOL) VIA CYTOCHROME P450-MEDIATED AROMATIC OXIDATION IN HUMAN LIVER MICROSOMESZhengyin Yan, H. Marlon Zhong, Noureddine Maher, Rhoda Torres, Gregory C. Leo, Gary W. Caldwell and Norman HuebertDrug Metabolism and Disposition December 2005, 33 (12) 1867-1876; DOI: https://doi.org/10.1124/dmd.105.006387
Yasuda, Kazuto
- You have accessROLE OF THE NUCLEAR RECEPTOR PREGNANE X RECEPTOR IN ACETAMINOPHEN HEPATOTOXICITYKristina K. Wolf, Sheryl G. Wood, Jane A. Hunt, Brooke W. Walton-Strong, Kazuto Yasuda, Lubin Lan, Su X. Duan, Qin Hao, Steven A. Wrighton, Elizabeth H. Jeffery, Ronald M. Evans, Juliana G. Szakacs, Lisa L. von Moltke, David J. Greenblatt, Michael H. Court, Erin G. Schuetz, Peter R. Sinclair and Jacqueline F. SinclairDrug Metabolism and Disposition December 2005, 33 (12) 1827-1836; DOI: https://doi.org/10.1124/dmd.105.005256
Yokoi, Tsuyoshi
- You have accessCYP2A6 AND CYP2B6 ARE INVOLVED IN NORNICOTINE FORMATION FROM NICOTINE IN HUMANS: INTERINDIVIDUAL DIFFERENCES IN THESE CONTRIBUTIONSHiroyuki Yamanaka, Miki Nakajima, Tatsuki Fukami, Haruko Sakai, Akiko Nakamura, Miki Katoh, Masataka Takamiya, Yasuhiro Aoki and Tsuyoshi YokoiDrug Metabolism and Disposition December 2005, 33 (12) 1811-1818; DOI: https://doi.org/10.1124/dmd.105.006254
Z
Zhao, Ping
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Zhong, H. Marlon
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