Index by author
September 01, 2005; Volume 33,Issue 9
A
Alterman, Michail A.
- You have accessQUANTITATIVE ANALYSIS OF CYTOCHROME P450 ISOZYMES BY MEANS OF UNIQUE ISOZYME-SPECIFIC TRYPTIC PEPTIDES: A PROTEOMIC APPROACHMichail A. Alterman, Boris Kornilayev, Tatyana Duzhak and Dmitry YakovlevDrug Metabolism and Disposition September 2005, 33 (9) 1399-1407; DOI: https://doi.org/10.1124/dmd.105.004812
Austin, R. P.
- You have accessA UNIFIED MODEL FOR PREDICTING HUMAN HEPATIC, METABOLIC CLEARANCE FROM IN VITRO INTRINSIC CLEARANCE DATA IN HEPATOCYTES AND MICROSOMESRobert J. Riley, D. F. McGinnity and R. P. AustinDrug Metabolism and Disposition September 2005, 33 (9) 1304-1311; DOI: https://doi.org/10.1124/dmd.105.004259
B
Barendregt, Arjan
- You have accessTHE USE OF SANDWICH-CULTURED RAT HEPATOCYTES TO DETERMINE THE INTRINSIC CLEARANCE OF COMPOUNDS WITH DIFFERENT EXTRACTION RATIOS: 7-ETHOXYCOUMARIN AND WARFARINNicoline Treijtel, Hanneke van Helvoort, Arjan Barendregt, Bas J. Blaauboer and Jan C. H. van EijkerenDrug Metabolism and Disposition September 2005, 33 (9) 1325-1332; DOI: https://doi.org/10.1124/dmd.105.004390
Bauman, Jonathan N.
- You have accessUDP-GLUCURONOSYLTRANSFERASE 2B7 IS THE MAJOR ENZYME RESPONSIBLE FOR GEMCABENE GLUCURONIDATION IN HUMAN LIVER MICROSOMESJonathan N. Bauman, Theunis C. Goosen, Meera Tugnait, Vincent Peterkin, Susan I. Hurst, Lee C. Menning, Mark Milad, Michael H. Court and J. Andrew WilliamsDrug Metabolism and Disposition September 2005, 33 (9) 1349-1354; DOI: https://doi.org/10.1124/dmd.105.005108
Blaauboer, Bas J.
- You have accessTHE USE OF SANDWICH-CULTURED RAT HEPATOCYTES TO DETERMINE THE INTRINSIC CLEARANCE OF COMPOUNDS WITH DIFFERENT EXTRACTION RATIOS: 7-ETHOXYCOUMARIN AND WARFARINNicoline Treijtel, Hanneke van Helvoort, Arjan Barendregt, Bas J. Blaauboer and Jan C. H. van EijkerenDrug Metabolism and Disposition September 2005, 33 (9) 1325-1332; DOI: https://doi.org/10.1124/dmd.105.004390
Brunner, Janice
- You have accessMETABOLISM AND DISPOSITION OF A POTENT GROUP II METABOTROPIC GLUTAMATE RECEPTOR AGONIST, IN RATS, DOGS, AND MONKEYSJoyce K. James, Masato Nakamura, Atsuro Nakazato, Kanyin E. Zhang, Merryl Cramer, Janice Brunner, Jacquelynn Cook and Weichao G. ChenDrug Metabolism and Disposition September 2005, 33 (9) 1373-1381; DOI: https://doi.org/10.1124/dmd.105.004978
C
Chen, Chong-Sheng
- You have accessENANTIOSELECTIVE METABOLISM AND CYTOTOXICITY OF R-IFOSFAMIDE AND S-IFOSFAMIDE BY TUMOR CELL-EXPRESSED CYTOCHROMES P450Chong-Sheng Chen, Youssef Jounaidi and David J. WaxmanDrug Metabolism and Disposition September 2005, 33 (9) 1261-1267; DOI: https://doi.org/10.1124/dmd.105.004788
Chen, Weichao G.
- You have accessMETABOLISM AND DISPOSITION OF A POTENT GROUP II METABOTROPIC GLUTAMATE RECEPTOR AGONIST, IN RATS, DOGS, AND MONKEYSJoyce K. James, Masato Nakamura, Atsuro Nakazato, Kanyin E. Zhang, Merryl Cramer, Janice Brunner, Jacquelynn Cook and Weichao G. ChenDrug Metabolism and Disposition September 2005, 33 (9) 1373-1381; DOI: https://doi.org/10.1124/dmd.105.004978
Cheng, Xingguo
- You have accessREGULATION OF MOUSE ORGANIC ANION-TRANSPORTING POLYPEPTIDES (OATPS) IN LIVER BY PROTOTYPICAL MICROSOMAL ENZYME INDUCERS THAT ACTIVATE DISTINCT TRANSCRIPTION FACTOR PATHWAYSXingguo Cheng, Jonathan Maher, Matthew Z. Dieter and Curtis D. KlaassenDrug Metabolism and Disposition September 2005, 33 (9) 1276-1282; DOI: https://doi.org/10.1124/dmd.105.003988
Chow, Moses S. S.
- You have accessEFFECT OF CYP2D6*10 ALLELE ON THE PHARMACOKINETICS OF LORATADINE IN CHINESE SUBJECTSOphelia Q. P. Yin, X. J. Shi, B. Tomlinson and Moses S. S. ChowDrug Metabolism and Disposition September 2005, 33 (9) 1283-1287; DOI: https://doi.org/10.1124/dmd.105.005025
Cook, Jacquelynn
- You have accessMETABOLISM AND DISPOSITION OF A POTENT GROUP II METABOTROPIC GLUTAMATE RECEPTOR AGONIST, IN RATS, DOGS, AND MONKEYSJoyce K. James, Masato Nakamura, Atsuro Nakazato, Kanyin E. Zhang, Merryl Cramer, Janice Brunner, Jacquelynn Cook and Weichao G. ChenDrug Metabolism and Disposition September 2005, 33 (9) 1373-1381; DOI: https://doi.org/10.1124/dmd.105.004978
Court, Michael H.
- You have accessUDP-GLUCURONOSYLTRANSFERASE 2B7 IS THE MAJOR ENZYME RESPONSIBLE FOR GEMCABENE GLUCURONIDATION IN HUMAN LIVER MICROSOMESJonathan N. Bauman, Theunis C. Goosen, Meera Tugnait, Vincent Peterkin, Susan I. Hurst, Lee C. Menning, Mark Milad, Michael H. Court and J. Andrew WilliamsDrug Metabolism and Disposition September 2005, 33 (9) 1349-1354; DOI: https://doi.org/10.1124/dmd.105.005108
Cramer, Merryl
- You have accessMETABOLISM AND DISPOSITION OF A POTENT GROUP II METABOTROPIC GLUTAMATE RECEPTOR AGONIST, IN RATS, DOGS, AND MONKEYSJoyce K. James, Masato Nakamura, Atsuro Nakazato, Kanyin E. Zhang, Merryl Cramer, Janice Brunner, Jacquelynn Cook and Weichao G. ChenDrug Metabolism and Disposition September 2005, 33 (9) 1373-1381; DOI: https://doi.org/10.1124/dmd.105.004978
Cui, Fu-De
- You have accessPOPULATION PHARMACOKINETICS OF CYCLOSPORINE IN CLINICAL RENAL TRANSPLANT PATIENTSKe-Hua Wu, Yi-Min Cui, Jin-Feng Guo, Ying Zhou, Suo-Di Zhai, Fu-De Cui and Wei LuDrug Metabolism and Disposition September 2005, 33 (9) 1268-1275; DOI: https://doi.org/10.1124/dmd.105.004358
Cui, Yi-Min
- You have accessPOPULATION PHARMACOKINETICS OF CYCLOSPORINE IN CLINICAL RENAL TRANSPLANT PATIENTSKe-Hua Wu, Yi-Min Cui, Jin-Feng Guo, Ying Zhou, Suo-Di Zhai, Fu-De Cui and Wei LuDrug Metabolism and Disposition September 2005, 33 (9) 1268-1275; DOI: https://doi.org/10.1124/dmd.105.004358
D
Dieter, Matthew Z.
- You have accessREGULATION OF MOUSE ORGANIC ANION-TRANSPORTING POLYPEPTIDES (OATPS) IN LIVER BY PROTOTYPICAL MICROSOMAL ENZYME INDUCERS THAT ACTIVATE DISTINCT TRANSCRIPTION FACTOR PATHWAYSXingguo Cheng, Jonathan Maher, Matthew Z. Dieter and Curtis D. KlaassenDrug Metabolism and Disposition September 2005, 33 (9) 1276-1282; DOI: https://doi.org/10.1124/dmd.105.003988
Duzhak, Tatyana
- You have accessQUANTITATIVE ANALYSIS OF CYTOCHROME P450 ISOZYMES BY MEANS OF UNIQUE ISOZYME-SPECIFIC TRYPTIC PEPTIDES: A PROTEOMIC APPROACHMichail A. Alterman, Boris Kornilayev, Tatyana Duzhak and Dmitry YakovlevDrug Metabolism and Disposition September 2005, 33 (9) 1399-1407; DOI: https://doi.org/10.1124/dmd.105.004812
F
Fujieda, Masaki
- You have accessCYP2A6 IS A PRINCIPAL ENZYME INVOLVED IN HYDROXYLATION OF 1,7-DIMETHYLXANTHINE, A MAIN CAFFEINE METABOLITE, IN HUMANSMiyuki Kimura, Hiroshi Yamazaki, Masaki Fujieda, Kazuma Kiyotani, Goro Honda, Junji Saruwatari, Kazuko Nakagawa, Takashi Ishizaki and Tetsuya KamatakiDrug Metabolism and Disposition September 2005, 33 (9) 1361-1366; DOI: https://doi.org/10.1124/dmd.105.004796
G
Ganaha, Sawako
- You have accessISOFORM-SPECIFIC EXPRESSION AND INDUCTION OF UDP-GLUCURONOSYLTRANSFERASE IN IMMUNOACTIVATED PERITONEAL MACROPHAGES OF THE RATYuki Tochigi, Naoko Yamashiki, Satoru Ohgiya, Sawako Ganaha and Hiroshi YokotaDrug Metabolism and Disposition September 2005, 33 (9) 1391-1398; DOI: https://doi.org/10.1124/dmd.105.004879
Giuliano, Claudio
- You have accessDIRECT DETERMINATION OF UNBOUND INTRINSIC DRUG CLEARANCE IN THE MICROSOMAL STABILITY ASSAYClaudio Giuliano, Mark Jairaj, Christian M. Zafiu and Ralph LauferDrug Metabolism and Disposition September 2005, 33 (9) 1319-1324; DOI: https://doi.org/10.1124/dmd.105.005033
Goosen, Theunis C.
- You have accessUDP-GLUCURONOSYLTRANSFERASE 2B7 IS THE MAJOR ENZYME RESPONSIBLE FOR GEMCABENE GLUCURONIDATION IN HUMAN LIVER MICROSOMESJonathan N. Bauman, Theunis C. Goosen, Meera Tugnait, Vincent Peterkin, Susan I. Hurst, Lee C. Menning, Mark Milad, Michael H. Court and J. Andrew WilliamsDrug Metabolism and Disposition September 2005, 33 (9) 1349-1354; DOI: https://doi.org/10.1124/dmd.105.005108
Guo, Jin-Feng
- You have accessPOPULATION PHARMACOKINETICS OF CYCLOSPORINE IN CLINICAL RENAL TRANSPLANT PATIENTSKe-Hua Wu, Yi-Min Cui, Jin-Feng Guo, Ying Zhou, Suo-Di Zhai, Fu-De Cui and Wei LuDrug Metabolism and Disposition September 2005, 33 (9) 1268-1275; DOI: https://doi.org/10.1124/dmd.105.004358
H
Hasinoff, Brian B.
- You have accessMETABOLISM OF THE ONE-RING OPEN METABOLITES OF THE CARDIOPROTECTIVE DRUG DEXRAZOXANE TO ITS ACTIVE METAL-CHELATING FORM IN THE RATPatricia E. Schroeder and Brian B. HasinoffDrug Metabolism and Disposition September 2005, 33 (9) 1367-1372; DOI: https://doi.org/10.1124/dmd.105.005546
Honda, Goro
- You have accessCYP2A6 IS A PRINCIPAL ENZYME INVOLVED IN HYDROXYLATION OF 1,7-DIMETHYLXANTHINE, A MAIN CAFFEINE METABOLITE, IN HUMANSMiyuki Kimura, Hiroshi Yamazaki, Masaki Fujieda, Kazuma Kiyotani, Goro Honda, Junji Saruwatari, Kazuko Nakagawa, Takashi Ishizaki and Tetsuya KamatakiDrug Metabolism and Disposition September 2005, 33 (9) 1361-1366; DOI: https://doi.org/10.1124/dmd.105.004796
Hurst, Susan I.
- You have accessUDP-GLUCURONOSYLTRANSFERASE 2B7 IS THE MAJOR ENZYME RESPONSIBLE FOR GEMCABENE GLUCURONIDATION IN HUMAN LIVER MICROSOMESJonathan N. Bauman, Theunis C. Goosen, Meera Tugnait, Vincent Peterkin, Susan I. Hurst, Lee C. Menning, Mark Milad, Michael H. Court and J. Andrew WilliamsDrug Metabolism and Disposition September 2005, 33 (9) 1349-1354; DOI: https://doi.org/10.1124/dmd.105.005108
I
Ishizaki, Takashi
- You have accessCYP2A6 IS A PRINCIPAL ENZYME INVOLVED IN HYDROXYLATION OF 1,7-DIMETHYLXANTHINE, A MAIN CAFFEINE METABOLITE, IN HUMANSMiyuki Kimura, Hiroshi Yamazaki, Masaki Fujieda, Kazuma Kiyotani, Goro Honda, Junji Saruwatari, Kazuko Nakagawa, Takashi Ishizaki and Tetsuya KamatakiDrug Metabolism and Disposition September 2005, 33 (9) 1361-1366; DOI: https://doi.org/10.1124/dmd.105.004796
J
Jairaj, Mark
- You have accessDIRECT DETERMINATION OF UNBOUND INTRINSIC DRUG CLEARANCE IN THE MICROSOMAL STABILITY ASSAYClaudio Giuliano, Mark Jairaj, Christian M. Zafiu and Ralph LauferDrug Metabolism and Disposition September 2005, 33 (9) 1319-1324; DOI: https://doi.org/10.1124/dmd.105.005033
James, Joyce K.
- You have accessMETABOLISM AND DISPOSITION OF A POTENT GROUP II METABOTROPIC GLUTAMATE RECEPTOR AGONIST, IN RATS, DOGS, AND MONKEYSJoyce K. James, Masato Nakamura, Atsuro Nakazato, Kanyin E. Zhang, Merryl Cramer, Janice Brunner, Jacquelynn Cook and Weichao G. ChenDrug Metabolism and Disposition September 2005, 33 (9) 1373-1381; DOI: https://doi.org/10.1124/dmd.105.004978
James, Margaret O.
- You have accessSULFONATION OF ENVIRONMENTAL CHEMICALS AND THEIR METABOLITES IN THE POLAR BEAR (Ursus maritimus)James C. Sacco and Margaret O. JamesDrug Metabolism and Disposition September 2005, 33 (9) 1341-1348; DOI: https://doi.org/10.1124/dmd.105.004648
Jemnitz, Katalin
- You have accessCANALICULAR AND SINUSOIDAL DISPOSITION OF BILIRUBIN MONO- AND DIGLUCURONIDES IN SANDWICH-CULTURED HUMAN AND RAT PRIMARY HEPATOCYTESGyörgy Lengyel, Zsuzsa Veres, Pál Szabó, László Vereczkey and Katalin JemnitzDrug Metabolism and Disposition September 2005, 33 (9) 1355-1360; DOI: https://doi.org/10.1124/dmd.105.004481
Jounaidi, Youssef
- You have accessENANTIOSELECTIVE METABOLISM AND CYTOTOXICITY OF R-IFOSFAMIDE AND S-IFOSFAMIDE BY TUMOR CELL-EXPRESSED CYTOCHROMES P450Chong-Sheng Chen, Youssef Jounaidi and David J. WaxmanDrug Metabolism and Disposition September 2005, 33 (9) 1261-1267; DOI: https://doi.org/10.1124/dmd.105.004788
K
Kamataki, Tetsuya
- You have accessCYP2A6 IS A PRINCIPAL ENZYME INVOLVED IN HYDROXYLATION OF 1,7-DIMETHYLXANTHINE, A MAIN CAFFEINE METABOLITE, IN HUMANSMiyuki Kimura, Hiroshi Yamazaki, Masaki Fujieda, Kazuma Kiyotani, Goro Honda, Junji Saruwatari, Kazuko Nakagawa, Takashi Ishizaki and Tetsuya KamatakiDrug Metabolism and Disposition September 2005, 33 (9) 1361-1366; DOI: https://doi.org/10.1124/dmd.105.004796
Katoh, Miki
- You have accessEXPRESSION OF HUMAN PHASE II ENZYMES IN CHIMERIC MICE WITH HUMANIZED LIVERMiki Katoh, Tomohito Matsui, Hirotoshi Okumura, Miki Nakajima, Masuhiro Nishimura, Shinsaku Naito, Chise Tateno, Katsutoshi Yoshizato and Tsuyoshi YokoiDrug Metabolism and Disposition September 2005, 33 (9) 1333-1340; DOI: https://doi.org/10.1124/dmd.105.005157
Kemper, Byron
- You have accessBIMOLECULAR FLUORESCENCE COMPLEMENTATION ANALYSIS OF CYTOCHROME P450 2C2, 2E1, AND NADPH-CYTOCHROME P450 REDUCTASE MOLECULAR INTERACTIONS IN LIVING CELLSCengiz Ozalp, Elzbieta Szczesna-Skorupa and Byron KemperDrug Metabolism and Disposition September 2005, 33 (9) 1382-1390; DOI: https://doi.org/10.1124/dmd.105.005538
Kimura, Miyuki
- You have accessCYP2A6 IS A PRINCIPAL ENZYME INVOLVED IN HYDROXYLATION OF 1,7-DIMETHYLXANTHINE, A MAIN CAFFEINE METABOLITE, IN HUMANSMiyuki Kimura, Hiroshi Yamazaki, Masaki Fujieda, Kazuma Kiyotani, Goro Honda, Junji Saruwatari, Kazuko Nakagawa, Takashi Ishizaki and Tetsuya KamatakiDrug Metabolism and Disposition September 2005, 33 (9) 1361-1366; DOI: https://doi.org/10.1124/dmd.105.004796
Kitamura, Shigeyuki
- You have accessINVOLVEMENT OF MOLYBDENUM HYDROXYLASES IN REDUCTIVE METABOLISM OF NITRO POLYCYCLIC AROMATIC HYDROCARBONS IN MAMMALIAN SKINOsamu Ueda, Kazumi Sugihara, Shigeru Ohta and Shigeyuki KitamuraDrug Metabolism and Disposition September 2005, 33 (9) 1312-1318; DOI: https://doi.org/10.1124/dmd.105.005306
Kiyotani, Kazuma
- You have accessCYP2A6 IS A PRINCIPAL ENZYME INVOLVED IN HYDROXYLATION OF 1,7-DIMETHYLXANTHINE, A MAIN CAFFEINE METABOLITE, IN HUMANSMiyuki Kimura, Hiroshi Yamazaki, Masaki Fujieda, Kazuma Kiyotani, Goro Honda, Junji Saruwatari, Kazuko Nakagawa, Takashi Ishizaki and Tetsuya KamatakiDrug Metabolism and Disposition September 2005, 33 (9) 1361-1366; DOI: https://doi.org/10.1124/dmd.105.004796
Klaassen, Curtis D.
- You have accessREGULATION OF MOUSE ORGANIC ANION-TRANSPORTING POLYPEPTIDES (OATPS) IN LIVER BY PROTOTYPICAL MICROSOMAL ENZYME INDUCERS THAT ACTIVATE DISTINCT TRANSCRIPTION FACTOR PATHWAYSXingguo Cheng, Jonathan Maher, Matthew Z. Dieter and Curtis D. KlaassenDrug Metabolism and Disposition September 2005, 33 (9) 1276-1282; DOI: https://doi.org/10.1124/dmd.105.003988
Kornilayev, Boris
- You have accessQUANTITATIVE ANALYSIS OF CYTOCHROME P450 ISOZYMES BY MEANS OF UNIQUE ISOZYME-SPECIFIC TRYPTIC PEPTIDES: A PROTEOMIC APPROACHMichail A. Alterman, Boris Kornilayev, Tatyana Duzhak and Dmitry YakovlevDrug Metabolism and Disposition September 2005, 33 (9) 1399-1407; DOI: https://doi.org/10.1124/dmd.105.004812
L
Laufer, Ralph
- You have accessDIRECT DETERMINATION OF UNBOUND INTRINSIC DRUG CLEARANCE IN THE MICROSOMAL STABILITY ASSAYClaudio Giuliano, Mark Jairaj, Christian M. Zafiu and Ralph LauferDrug Metabolism and Disposition September 2005, 33 (9) 1319-1324; DOI: https://doi.org/10.1124/dmd.105.005033
Lengyel, György
- You have accessCANALICULAR AND SINUSOIDAL DISPOSITION OF BILIRUBIN MONO- AND DIGLUCURONIDES IN SANDWICH-CULTURED HUMAN AND RAT PRIMARY HEPATOCYTESGyörgy Lengyel, Zsuzsa Veres, Pál Szabó, László Vereczkey and Katalin JemnitzDrug Metabolism and Disposition September 2005, 33 (9) 1355-1360; DOI: https://doi.org/10.1124/dmd.105.004481
Lu, Wei
- You have accessPOPULATION PHARMACOKINETICS OF CYCLOSPORINE IN CLINICAL RENAL TRANSPLANT PATIENTSKe-Hua Wu, Yi-Min Cui, Jin-Feng Guo, Ying Zhou, Suo-Di Zhai, Fu-De Cui and Wei LuDrug Metabolism and Disposition September 2005, 33 (9) 1268-1275; DOI: https://doi.org/10.1124/dmd.105.004358
M
Maher, Jonathan
- You have accessREGULATION OF MOUSE ORGANIC ANION-TRANSPORTING POLYPEPTIDES (OATPS) IN LIVER BY PROTOTYPICAL MICROSOMAL ENZYME INDUCERS THAT ACTIVATE DISTINCT TRANSCRIPTION FACTOR PATHWAYSXingguo Cheng, Jonathan Maher, Matthew Z. Dieter and Curtis D. KlaassenDrug Metabolism and Disposition September 2005, 33 (9) 1276-1282; DOI: https://doi.org/10.1124/dmd.105.003988
Matsui, Tomohito
- You have accessEXPRESSION OF HUMAN PHASE II ENZYMES IN CHIMERIC MICE WITH HUMANIZED LIVERMiki Katoh, Tomohito Matsui, Hirotoshi Okumura, Miki Nakajima, Masuhiro Nishimura, Shinsaku Naito, Chise Tateno, Katsutoshi Yoshizato and Tsuyoshi YokoiDrug Metabolism and Disposition September 2005, 33 (9) 1333-1340; DOI: https://doi.org/10.1124/dmd.105.005157
Mayersohn, Michael
- You have accessACCURACY OF ALLOMETRICALLY PREDICTED PHARMACOKINETIC PARAMETERS IN HUMANS: ROLE OF SPECIES SELECTIONHuadong Tang and Michael MayersohnDrug Metabolism and Disposition September 2005, 33 (9) 1288-1293; DOI: https://doi.org/10.1124/dmd.105.004127
- You have accessA MATHEMATICAL DESCRIPTION OF THE FUNCTIONALITY OF CORRECTION FACTORS USED IN ALLOMETRY FOR PREDICTING HUMAN DRUG CLEARANCEHuadong Tang and Michael MayersohnDrug Metabolism and Disposition September 2005, 33 (9) 1294-1296; DOI: https://doi.org/10.1124/dmd.105.004135
- You have accessA NOVEL MODEL FOR PREDICTION OF HUMAN DRUG CLEARANCE BY ALLOMETRIC SCALINGHuadong Tang and Michael MayersohnDrug Metabolism and Disposition September 2005, 33 (9) 1297-1303; DOI: https://doi.org/10.1124/dmd.105.004143
McGinnity, D. F.
- You have accessA UNIFIED MODEL FOR PREDICTING HUMAN HEPATIC, METABOLIC CLEARANCE FROM IN VITRO INTRINSIC CLEARANCE DATA IN HEPATOCYTES AND MICROSOMESRobert J. Riley, D. F. McGinnity and R. P. AustinDrug Metabolism and Disposition September 2005, 33 (9) 1304-1311; DOI: https://doi.org/10.1124/dmd.105.004259
Menning, Lee C.
- You have accessUDP-GLUCURONOSYLTRANSFERASE 2B7 IS THE MAJOR ENZYME RESPONSIBLE FOR GEMCABENE GLUCURONIDATION IN HUMAN LIVER MICROSOMESJonathan N. Bauman, Theunis C. Goosen, Meera Tugnait, Vincent Peterkin, Susan I. Hurst, Lee C. Menning, Mark Milad, Michael H. Court and J. Andrew WilliamsDrug Metabolism and Disposition September 2005, 33 (9) 1349-1354; DOI: https://doi.org/10.1124/dmd.105.005108
Milad, Mark
- You have accessUDP-GLUCURONOSYLTRANSFERASE 2B7 IS THE MAJOR ENZYME RESPONSIBLE FOR GEMCABENE GLUCURONIDATION IN HUMAN LIVER MICROSOMESJonathan N. Bauman, Theunis C. Goosen, Meera Tugnait, Vincent Peterkin, Susan I. Hurst, Lee C. Menning, Mark Milad, Michael H. Court and J. Andrew WilliamsDrug Metabolism and Disposition September 2005, 33 (9) 1349-1354; DOI: https://doi.org/10.1124/dmd.105.005108
N
Naito, Shinsaku
- You have accessEXPRESSION OF HUMAN PHASE II ENZYMES IN CHIMERIC MICE WITH HUMANIZED LIVERMiki Katoh, Tomohito Matsui, Hirotoshi Okumura, Miki Nakajima, Masuhiro Nishimura, Shinsaku Naito, Chise Tateno, Katsutoshi Yoshizato and Tsuyoshi YokoiDrug Metabolism and Disposition September 2005, 33 (9) 1333-1340; DOI: https://doi.org/10.1124/dmd.105.005157
Nakagawa, Kazuko
- You have accessCYP2A6 IS A PRINCIPAL ENZYME INVOLVED IN HYDROXYLATION OF 1,7-DIMETHYLXANTHINE, A MAIN CAFFEINE METABOLITE, IN HUMANSMiyuki Kimura, Hiroshi Yamazaki, Masaki Fujieda, Kazuma Kiyotani, Goro Honda, Junji Saruwatari, Kazuko Nakagawa, Takashi Ishizaki and Tetsuya KamatakiDrug Metabolism and Disposition September 2005, 33 (9) 1361-1366; DOI: https://doi.org/10.1124/dmd.105.004796
Nakajima, Miki
- You have accessEXPRESSION OF HUMAN PHASE II ENZYMES IN CHIMERIC MICE WITH HUMANIZED LIVERMiki Katoh, Tomohito Matsui, Hirotoshi Okumura, Miki Nakajima, Masuhiro Nishimura, Shinsaku Naito, Chise Tateno, Katsutoshi Yoshizato and Tsuyoshi YokoiDrug Metabolism and Disposition September 2005, 33 (9) 1333-1340; DOI: https://doi.org/10.1124/dmd.105.005157
Nakamura, Masato
- You have accessMETABOLISM AND DISPOSITION OF A POTENT GROUP II METABOTROPIC GLUTAMATE RECEPTOR AGONIST, IN RATS, DOGS, AND MONKEYSJoyce K. James, Masato Nakamura, Atsuro Nakazato, Kanyin E. Zhang, Merryl Cramer, Janice Brunner, Jacquelynn Cook and Weichao G. ChenDrug Metabolism and Disposition September 2005, 33 (9) 1373-1381; DOI: https://doi.org/10.1124/dmd.105.004978
Nakazato, Atsuro
- You have accessMETABOLISM AND DISPOSITION OF A POTENT GROUP II METABOTROPIC GLUTAMATE RECEPTOR AGONIST, IN RATS, DOGS, AND MONKEYSJoyce K. James, Masato Nakamura, Atsuro Nakazato, Kanyin E. Zhang, Merryl Cramer, Janice Brunner, Jacquelynn Cook and Weichao G. ChenDrug Metabolism and Disposition September 2005, 33 (9) 1373-1381; DOI: https://doi.org/10.1124/dmd.105.004978
Nishimura, Masuhiro
- You have accessEXPRESSION OF HUMAN PHASE II ENZYMES IN CHIMERIC MICE WITH HUMANIZED LIVERMiki Katoh, Tomohito Matsui, Hirotoshi Okumura, Miki Nakajima, Masuhiro Nishimura, Shinsaku Naito, Chise Tateno, Katsutoshi Yoshizato and Tsuyoshi YokoiDrug Metabolism and Disposition September 2005, 33 (9) 1333-1340; DOI: https://doi.org/10.1124/dmd.105.005157
O
Ohgiya, Satoru
- You have accessISOFORM-SPECIFIC EXPRESSION AND INDUCTION OF UDP-GLUCURONOSYLTRANSFERASE IN IMMUNOACTIVATED PERITONEAL MACROPHAGES OF THE RATYuki Tochigi, Naoko Yamashiki, Satoru Ohgiya, Sawako Ganaha and Hiroshi YokotaDrug Metabolism and Disposition September 2005, 33 (9) 1391-1398; DOI: https://doi.org/10.1124/dmd.105.004879
Ohta, Shigeru
- You have accessINVOLVEMENT OF MOLYBDENUM HYDROXYLASES IN REDUCTIVE METABOLISM OF NITRO POLYCYCLIC AROMATIC HYDROCARBONS IN MAMMALIAN SKINOsamu Ueda, Kazumi Sugihara, Shigeru Ohta and Shigeyuki KitamuraDrug Metabolism and Disposition September 2005, 33 (9) 1312-1318; DOI: https://doi.org/10.1124/dmd.105.005306
Okumura, Hirotoshi
- You have accessEXPRESSION OF HUMAN PHASE II ENZYMES IN CHIMERIC MICE WITH HUMANIZED LIVERMiki Katoh, Tomohito Matsui, Hirotoshi Okumura, Miki Nakajima, Masuhiro Nishimura, Shinsaku Naito, Chise Tateno, Katsutoshi Yoshizato and Tsuyoshi YokoiDrug Metabolism and Disposition September 2005, 33 (9) 1333-1340; DOI: https://doi.org/10.1124/dmd.105.005157
Ozalp, Cengiz
- You have accessBIMOLECULAR FLUORESCENCE COMPLEMENTATION ANALYSIS OF CYTOCHROME P450 2C2, 2E1, AND NADPH-CYTOCHROME P450 REDUCTASE MOLECULAR INTERACTIONS IN LIVING CELLSCengiz Ozalp, Elzbieta Szczesna-Skorupa and Byron KemperDrug Metabolism and Disposition September 2005, 33 (9) 1382-1390; DOI: https://doi.org/10.1124/dmd.105.005538
P
Peterkin, Vincent
- You have accessUDP-GLUCURONOSYLTRANSFERASE 2B7 IS THE MAJOR ENZYME RESPONSIBLE FOR GEMCABENE GLUCURONIDATION IN HUMAN LIVER MICROSOMESJonathan N. Bauman, Theunis C. Goosen, Meera Tugnait, Vincent Peterkin, Susan I. Hurst, Lee C. Menning, Mark Milad, Michael H. Court and J. Andrew WilliamsDrug Metabolism and Disposition September 2005, 33 (9) 1349-1354; DOI: https://doi.org/10.1124/dmd.105.005108
R
Riley, Robert J.
- You have accessA UNIFIED MODEL FOR PREDICTING HUMAN HEPATIC, METABOLIC CLEARANCE FROM IN VITRO INTRINSIC CLEARANCE DATA IN HEPATOCYTES AND MICROSOMESRobert J. Riley, D. F. McGinnity and R. P. AustinDrug Metabolism and Disposition September 2005, 33 (9) 1304-1311; DOI: https://doi.org/10.1124/dmd.105.004259
S
Sacco, James C.
- You have accessSULFONATION OF ENVIRONMENTAL CHEMICALS AND THEIR METABOLITES IN THE POLAR BEAR (Ursus maritimus)James C. Sacco and Margaret O. JamesDrug Metabolism and Disposition September 2005, 33 (9) 1341-1348; DOI: https://doi.org/10.1124/dmd.105.004648
Saruwatari, Junji
- You have accessCYP2A6 IS A PRINCIPAL ENZYME INVOLVED IN HYDROXYLATION OF 1,7-DIMETHYLXANTHINE, A MAIN CAFFEINE METABOLITE, IN HUMANSMiyuki Kimura, Hiroshi Yamazaki, Masaki Fujieda, Kazuma Kiyotani, Goro Honda, Junji Saruwatari, Kazuko Nakagawa, Takashi Ishizaki and Tetsuya KamatakiDrug Metabolism and Disposition September 2005, 33 (9) 1361-1366; DOI: https://doi.org/10.1124/dmd.105.004796
Schroeder, Patricia E.
- You have accessMETABOLISM OF THE ONE-RING OPEN METABOLITES OF THE CARDIOPROTECTIVE DRUG DEXRAZOXANE TO ITS ACTIVE METAL-CHELATING FORM IN THE RATPatricia E. Schroeder and Brian B. HasinoffDrug Metabolism and Disposition September 2005, 33 (9) 1367-1372; DOI: https://doi.org/10.1124/dmd.105.005546
Shi, X. J.
- You have accessEFFECT OF CYP2D6*10 ALLELE ON THE PHARMACOKINETICS OF LORATADINE IN CHINESE SUBJECTSOphelia Q. P. Yin, X. J. Shi, B. Tomlinson and Moses S. S. ChowDrug Metabolism and Disposition September 2005, 33 (9) 1283-1287; DOI: https://doi.org/10.1124/dmd.105.005025
Sugihara, Kazumi
- You have accessINVOLVEMENT OF MOLYBDENUM HYDROXYLASES IN REDUCTIVE METABOLISM OF NITRO POLYCYCLIC AROMATIC HYDROCARBONS IN MAMMALIAN SKINOsamu Ueda, Kazumi Sugihara, Shigeru Ohta and Shigeyuki KitamuraDrug Metabolism and Disposition September 2005, 33 (9) 1312-1318; DOI: https://doi.org/10.1124/dmd.105.005306
Szabó, Pál
- You have accessCANALICULAR AND SINUSOIDAL DISPOSITION OF BILIRUBIN MONO- AND DIGLUCURONIDES IN SANDWICH-CULTURED HUMAN AND RAT PRIMARY HEPATOCYTESGyörgy Lengyel, Zsuzsa Veres, Pál Szabó, László Vereczkey and Katalin JemnitzDrug Metabolism and Disposition September 2005, 33 (9) 1355-1360; DOI: https://doi.org/10.1124/dmd.105.004481
Szczesna-Skorupa, Elzbieta
- You have accessBIMOLECULAR FLUORESCENCE COMPLEMENTATION ANALYSIS OF CYTOCHROME P450 2C2, 2E1, AND NADPH-CYTOCHROME P450 REDUCTASE MOLECULAR INTERACTIONS IN LIVING CELLSCengiz Ozalp, Elzbieta Szczesna-Skorupa and Byron KemperDrug Metabolism and Disposition September 2005, 33 (9) 1382-1390; DOI: https://doi.org/10.1124/dmd.105.005538
T
Tang, Huadong
- You have accessACCURACY OF ALLOMETRICALLY PREDICTED PHARMACOKINETIC PARAMETERS IN HUMANS: ROLE OF SPECIES SELECTIONHuadong Tang and Michael MayersohnDrug Metabolism and Disposition September 2005, 33 (9) 1288-1293; DOI: https://doi.org/10.1124/dmd.105.004127
- You have accessA MATHEMATICAL DESCRIPTION OF THE FUNCTIONALITY OF CORRECTION FACTORS USED IN ALLOMETRY FOR PREDICTING HUMAN DRUG CLEARANCEHuadong Tang and Michael MayersohnDrug Metabolism and Disposition September 2005, 33 (9) 1294-1296; DOI: https://doi.org/10.1124/dmd.105.004135
- You have accessA NOVEL MODEL FOR PREDICTION OF HUMAN DRUG CLEARANCE BY ALLOMETRIC SCALINGHuadong Tang and Michael MayersohnDrug Metabolism and Disposition September 2005, 33 (9) 1297-1303; DOI: https://doi.org/10.1124/dmd.105.004143
Tateno, Chise
- You have accessEXPRESSION OF HUMAN PHASE II ENZYMES IN CHIMERIC MICE WITH HUMANIZED LIVERMiki Katoh, Tomohito Matsui, Hirotoshi Okumura, Miki Nakajima, Masuhiro Nishimura, Shinsaku Naito, Chise Tateno, Katsutoshi Yoshizato and Tsuyoshi YokoiDrug Metabolism and Disposition September 2005, 33 (9) 1333-1340; DOI: https://doi.org/10.1124/dmd.105.005157
Tochigi, Yuki
- You have accessISOFORM-SPECIFIC EXPRESSION AND INDUCTION OF UDP-GLUCURONOSYLTRANSFERASE IN IMMUNOACTIVATED PERITONEAL MACROPHAGES OF THE RATYuki Tochigi, Naoko Yamashiki, Satoru Ohgiya, Sawako Ganaha and Hiroshi YokotaDrug Metabolism and Disposition September 2005, 33 (9) 1391-1398; DOI: https://doi.org/10.1124/dmd.105.004879
Tomlinson, B.
- You have accessEFFECT OF CYP2D6*10 ALLELE ON THE PHARMACOKINETICS OF LORATADINE IN CHINESE SUBJECTSOphelia Q. P. Yin, X. J. Shi, B. Tomlinson and Moses S. S. ChowDrug Metabolism and Disposition September 2005, 33 (9) 1283-1287; DOI: https://doi.org/10.1124/dmd.105.005025
Treijtel, Nicoline
- You have accessTHE USE OF SANDWICH-CULTURED RAT HEPATOCYTES TO DETERMINE THE INTRINSIC CLEARANCE OF COMPOUNDS WITH DIFFERENT EXTRACTION RATIOS: 7-ETHOXYCOUMARIN AND WARFARINNicoline Treijtel, Hanneke van Helvoort, Arjan Barendregt, Bas J. Blaauboer and Jan C. H. van EijkerenDrug Metabolism and Disposition September 2005, 33 (9) 1325-1332; DOI: https://doi.org/10.1124/dmd.105.004390
Tugnait, Meera
- You have accessUDP-GLUCURONOSYLTRANSFERASE 2B7 IS THE MAJOR ENZYME RESPONSIBLE FOR GEMCABENE GLUCURONIDATION IN HUMAN LIVER MICROSOMESJonathan N. Bauman, Theunis C. Goosen, Meera Tugnait, Vincent Peterkin, Susan I. Hurst, Lee C. Menning, Mark Milad, Michael H. Court and J. Andrew WilliamsDrug Metabolism and Disposition September 2005, 33 (9) 1349-1354; DOI: https://doi.org/10.1124/dmd.105.005108
U
Ueda, Osamu
- You have accessINVOLVEMENT OF MOLYBDENUM HYDROXYLASES IN REDUCTIVE METABOLISM OF NITRO POLYCYCLIC AROMATIC HYDROCARBONS IN MAMMALIAN SKINOsamu Ueda, Kazumi Sugihara, Shigeru Ohta and Shigeyuki KitamuraDrug Metabolism and Disposition September 2005, 33 (9) 1312-1318; DOI: https://doi.org/10.1124/dmd.105.005306
V
van Eijkeren, Jan C. H.
- You have accessTHE USE OF SANDWICH-CULTURED RAT HEPATOCYTES TO DETERMINE THE INTRINSIC CLEARANCE OF COMPOUNDS WITH DIFFERENT EXTRACTION RATIOS: 7-ETHOXYCOUMARIN AND WARFARINNicoline Treijtel, Hanneke van Helvoort, Arjan Barendregt, Bas J. Blaauboer and Jan C. H. van EijkerenDrug Metabolism and Disposition September 2005, 33 (9) 1325-1332; DOI: https://doi.org/10.1124/dmd.105.004390
van Helvoort, Hanneke
- You have accessTHE USE OF SANDWICH-CULTURED RAT HEPATOCYTES TO DETERMINE THE INTRINSIC CLEARANCE OF COMPOUNDS WITH DIFFERENT EXTRACTION RATIOS: 7-ETHOXYCOUMARIN AND WARFARINNicoline Treijtel, Hanneke van Helvoort, Arjan Barendregt, Bas J. Blaauboer and Jan C. H. van EijkerenDrug Metabolism and Disposition September 2005, 33 (9) 1325-1332; DOI: https://doi.org/10.1124/dmd.105.004390
Vereczkey, László
- You have accessCANALICULAR AND SINUSOIDAL DISPOSITION OF BILIRUBIN MONO- AND DIGLUCURONIDES IN SANDWICH-CULTURED HUMAN AND RAT PRIMARY HEPATOCYTESGyörgy Lengyel, Zsuzsa Veres, Pál Szabó, László Vereczkey and Katalin JemnitzDrug Metabolism and Disposition September 2005, 33 (9) 1355-1360; DOI: https://doi.org/10.1124/dmd.105.004481
Veres, Zsuzsa
- You have accessCANALICULAR AND SINUSOIDAL DISPOSITION OF BILIRUBIN MONO- AND DIGLUCURONIDES IN SANDWICH-CULTURED HUMAN AND RAT PRIMARY HEPATOCYTESGyörgy Lengyel, Zsuzsa Veres, Pál Szabó, László Vereczkey and Katalin JemnitzDrug Metabolism and Disposition September 2005, 33 (9) 1355-1360; DOI: https://doi.org/10.1124/dmd.105.004481
W
Waxman, David J.
- You have accessENANTIOSELECTIVE METABOLISM AND CYTOTOXICITY OF R-IFOSFAMIDE AND S-IFOSFAMIDE BY TUMOR CELL-EXPRESSED CYTOCHROMES P450Chong-Sheng Chen, Youssef Jounaidi and David J. WaxmanDrug Metabolism and Disposition September 2005, 33 (9) 1261-1267; DOI: https://doi.org/10.1124/dmd.105.004788
Williams, J. Andrew
- You have accessUDP-GLUCURONOSYLTRANSFERASE 2B7 IS THE MAJOR ENZYME RESPONSIBLE FOR GEMCABENE GLUCURONIDATION IN HUMAN LIVER MICROSOMESJonathan N. Bauman, Theunis C. Goosen, Meera Tugnait, Vincent Peterkin, Susan I. Hurst, Lee C. Menning, Mark Milad, Michael H. Court and J. Andrew WilliamsDrug Metabolism and Disposition September 2005, 33 (9) 1349-1354; DOI: https://doi.org/10.1124/dmd.105.005108
Wu, Ke-Hua
- You have accessPOPULATION PHARMACOKINETICS OF CYCLOSPORINE IN CLINICAL RENAL TRANSPLANT PATIENTSKe-Hua Wu, Yi-Min Cui, Jin-Feng Guo, Ying Zhou, Suo-Di Zhai, Fu-De Cui and Wei LuDrug Metabolism and Disposition September 2005, 33 (9) 1268-1275; DOI: https://doi.org/10.1124/dmd.105.004358
Y
Yakovlev, Dmitry
- You have accessQUANTITATIVE ANALYSIS OF CYTOCHROME P450 ISOZYMES BY MEANS OF UNIQUE ISOZYME-SPECIFIC TRYPTIC PEPTIDES: A PROTEOMIC APPROACHMichail A. Alterman, Boris Kornilayev, Tatyana Duzhak and Dmitry YakovlevDrug Metabolism and Disposition September 2005, 33 (9) 1399-1407; DOI: https://doi.org/10.1124/dmd.105.004812
Yamashiki, Naoko
- You have accessISOFORM-SPECIFIC EXPRESSION AND INDUCTION OF UDP-GLUCURONOSYLTRANSFERASE IN IMMUNOACTIVATED PERITONEAL MACROPHAGES OF THE RATYuki Tochigi, Naoko Yamashiki, Satoru Ohgiya, Sawako Ganaha and Hiroshi YokotaDrug Metabolism and Disposition September 2005, 33 (9) 1391-1398; DOI: https://doi.org/10.1124/dmd.105.004879
Yamazaki, Hiroshi
- You have accessCYP2A6 IS A PRINCIPAL ENZYME INVOLVED IN HYDROXYLATION OF 1,7-DIMETHYLXANTHINE, A MAIN CAFFEINE METABOLITE, IN HUMANSMiyuki Kimura, Hiroshi Yamazaki, Masaki Fujieda, Kazuma Kiyotani, Goro Honda, Junji Saruwatari, Kazuko Nakagawa, Takashi Ishizaki and Tetsuya KamatakiDrug Metabolism and Disposition September 2005, 33 (9) 1361-1366; DOI: https://doi.org/10.1124/dmd.105.004796
Yin, Ophelia Q. P.
- You have accessEFFECT OF CYP2D6*10 ALLELE ON THE PHARMACOKINETICS OF LORATADINE IN CHINESE SUBJECTSOphelia Q. P. Yin, X. J. Shi, B. Tomlinson and Moses S. S. ChowDrug Metabolism and Disposition September 2005, 33 (9) 1283-1287; DOI: https://doi.org/10.1124/dmd.105.005025
Yokoi, Tsuyoshi
- You have accessEXPRESSION OF HUMAN PHASE II ENZYMES IN CHIMERIC MICE WITH HUMANIZED LIVERMiki Katoh, Tomohito Matsui, Hirotoshi Okumura, Miki Nakajima, Masuhiro Nishimura, Shinsaku Naito, Chise Tateno, Katsutoshi Yoshizato and Tsuyoshi YokoiDrug Metabolism and Disposition September 2005, 33 (9) 1333-1340; DOI: https://doi.org/10.1124/dmd.105.005157
Yokota, Hiroshi
- You have accessISOFORM-SPECIFIC EXPRESSION AND INDUCTION OF UDP-GLUCURONOSYLTRANSFERASE IN IMMUNOACTIVATED PERITONEAL MACROPHAGES OF THE RATYuki Tochigi, Naoko Yamashiki, Satoru Ohgiya, Sawako Ganaha and Hiroshi YokotaDrug Metabolism and Disposition September 2005, 33 (9) 1391-1398; DOI: https://doi.org/10.1124/dmd.105.004879
Yoshizato, Katsutoshi
- You have accessEXPRESSION OF HUMAN PHASE II ENZYMES IN CHIMERIC MICE WITH HUMANIZED LIVERMiki Katoh, Tomohito Matsui, Hirotoshi Okumura, Miki Nakajima, Masuhiro Nishimura, Shinsaku Naito, Chise Tateno, Katsutoshi Yoshizato and Tsuyoshi YokoiDrug Metabolism and Disposition September 2005, 33 (9) 1333-1340; DOI: https://doi.org/10.1124/dmd.105.005157
Z
Zafiu, Christian M.
- You have accessDIRECT DETERMINATION OF UNBOUND INTRINSIC DRUG CLEARANCE IN THE MICROSOMAL STABILITY ASSAYClaudio Giuliano, Mark Jairaj, Christian M. Zafiu and Ralph LauferDrug Metabolism and Disposition September 2005, 33 (9) 1319-1324; DOI: https://doi.org/10.1124/dmd.105.005033
Zhai, Suo-Di
- You have accessPOPULATION PHARMACOKINETICS OF CYCLOSPORINE IN CLINICAL RENAL TRANSPLANT PATIENTSKe-Hua Wu, Yi-Min Cui, Jin-Feng Guo, Ying Zhou, Suo-Di Zhai, Fu-De Cui and Wei LuDrug Metabolism and Disposition September 2005, 33 (9) 1268-1275; DOI: https://doi.org/10.1124/dmd.105.004358
Zhang, Kanyin E.
- You have accessMETABOLISM AND DISPOSITION OF A POTENT GROUP II METABOTROPIC GLUTAMATE RECEPTOR AGONIST, IN RATS, DOGS, AND MONKEYSJoyce K. James, Masato Nakamura, Atsuro Nakazato, Kanyin E. Zhang, Merryl Cramer, Janice Brunner, Jacquelynn Cook and Weichao G. ChenDrug Metabolism and Disposition September 2005, 33 (9) 1373-1381; DOI: https://doi.org/10.1124/dmd.105.004978
Zhou, Ying
- You have accessPOPULATION PHARMACOKINETICS OF CYCLOSPORINE IN CLINICAL RENAL TRANSPLANT PATIENTSKe-Hua Wu, Yi-Min Cui, Jin-Feng Guo, Ying Zhou, Suo-Di Zhai, Fu-De Cui and Wei LuDrug Metabolism and Disposition September 2005, 33 (9) 1268-1275; DOI: https://doi.org/10.1124/dmd.105.004358