Index by author
January 01, 2009; Volume 37,Issue 1
A
Alvarez, Ana I.
- You have accessNatural Allelic Variants of Bovine ATP-Binding Cassette Transporter ABCG2: Increased Activity of the Ser581 Variant and Development of Tools for the Discovery of New ABCG2 InhibitorsGracia Merino, Rebeca Real, Marta F. Baro, Lucia Gonzalez-Lobato, Julio G. Prieto, Ana I. Alvarez and Margarita M. MarquesDrug Metabolism and Disposition January 2009, 37 (1) 5-9; DOI: https://doi.org/10.1124/dmd.108.022715
Andersson, Tommy B.
- You have accessThe Multiple Depletion Curves Method Provides Accurate Estimates of Intrinsic Clearance (CLint), Maximum Velocity of the Metabolic Reaction (Vmax), and Michaelis Constant (Km): Accuracy and Robustness Evaluated through Experimental Data and Monte Carlo SimulationsErik Sjögren, Hans Lennernäs, Tommy B. Andersson, Johan Gråsjö and Ulf BredbergDrug Metabolism and Disposition January 2009, 37 (1) 47-58; DOI: https://doi.org/10.1124/dmd.108.021477
Argikar, Upendra A.
- You have accessEffect of Aging on Glucuronidation of Valproic Acid in Human Liver Microsomes and the Role of UDP-Glucuronosyltransferase UGT1A4, UGT1A8, and UGT1A10Upendra A. Argikar and Rory P. RemmelDrug Metabolism and Disposition January 2009, 37 (1) 229-236; DOI: https://doi.org/10.1124/dmd.108.022426
Ashgodom, Rezene T.
- You have accessStructural Modulation of Oxidative Metabolism in Design of Improved Benzothiophene Selective Estrogen Receptor ModulatorsZhihui Qin, Irida Kastrati, Rezene T. Ashgodom, Daniel D. Lantvit, Cassia R. Overk, Yongsoo Choi, Richard B. van Breemen, Judy L. Bolton and Gregory R. J. ThatcherDrug Metabolism and Disposition January 2009, 37 (1) 161-169; DOI: https://doi.org/10.1124/dmd.108.023408
B
Balogh, Larissa M.
- You have accessMechanism-Based Inactivation of Cytochrome P450 2C9 by Tienilic Acid and (±)-Suprofen: A Comparison of Kinetics and Probe Substrate SelectionJ. Matthew Hutzler, Larissa M. Balogh, Michael Zientek, Vikas Kumar and Timothy S. TracyDrug Metabolism and Disposition January 2009, 37 (1) 59-65; DOI: https://doi.org/10.1124/dmd.108.023358
Baro, Marta F.
- You have accessNatural Allelic Variants of Bovine ATP-Binding Cassette Transporter ABCG2: Increased Activity of the Ser581 Variant and Development of Tools for the Discovery of New ABCG2 InhibitorsGracia Merino, Rebeca Real, Marta F. Baro, Lucia Gonzalez-Lobato, Julio G. Prieto, Ana I. Alvarez and Margarita M. MarquesDrug Metabolism and Disposition January 2009, 37 (1) 5-9; DOI: https://doi.org/10.1124/dmd.108.022715
Beijnen, Jos H.
- You have accessTransport of Diclofenac by Breast Cancer Resistance Protein (ABCG2) and Stimulation of Multidrug Resistance Protein 2 (ABCC2)-Mediated Drug Transport by Diclofenac and BenzbromaroneJurjen S. Lagas, Cornelia M. M. van der Kruijssen, Koen van de Wetering, Jos H. Beijnen and Alfred H. SchinkelDrug Metabolism and Disposition January 2009, 37 (1) 129-136; DOI: https://doi.org/10.1124/dmd.108.023200
Bolton, Judy L.
- You have accessStructural Modulation of Oxidative Metabolism in Design of Improved Benzothiophene Selective Estrogen Receptor ModulatorsZhihui Qin, Irida Kastrati, Rezene T. Ashgodom, Daniel D. Lantvit, Cassia R. Overk, Yongsoo Choi, Richard B. van Breemen, Judy L. Bolton and Gregory R. J. ThatcherDrug Metabolism and Disposition January 2009, 37 (1) 161-169; DOI: https://doi.org/10.1124/dmd.108.023408
Bonacorsi, Samuel
- You have accessApixaban Metabolism and Pharmacokinetics after Oral Administration to HumansNirmala Raghavan, Charles E. Frost, Zhigang Yu, Kan He, Haiying Zhang, W. Griffith Humphreys, Donald Pinto, Shiangyuan Chen, Samuel Bonacorsi, Pancras C. Wong and Donglu ZhangDrug Metabolism and Disposition January 2009, 37 (1) 74-81; DOI: https://doi.org/10.1124/dmd.108.023143
Brandsch, Matthias
- You have accessHigh-Affinity Interaction of Sartans with H+/Peptide TransportersIlka Knütter, Gabor Kottra, Wiebke Fischer, Hannelore Daniel and Matthias BrandschDrug Metabolism and Disposition January 2009, 37 (1) 143-149; DOI: https://doi.org/10.1124/dmd.108.022418
Bredberg, Ulf
- You have accessThe Multiple Depletion Curves Method Provides Accurate Estimates of Intrinsic Clearance (CLint), Maximum Velocity of the Metabolic Reaction (Vmax), and Michaelis Constant (Km): Accuracy and Robustness Evaluated through Experimental Data and Monte Carlo SimulationsErik Sjögren, Hans Lennernäs, Tommy B. Andersson, Johan Gråsjö and Ulf BredbergDrug Metabolism and Disposition January 2009, 37 (1) 47-58; DOI: https://doi.org/10.1124/dmd.108.021477
C
Cao, Jin
- You have accessQuantitation of Human Cytochrome P450 2D6 Protein with Immunoblot and Mass Spectrometry AnalysisAi-Ming Yu, Jun Qu, Melanie A. Felmlee, Jin Cao and Xi-Ling JiangDrug Metabolism and Disposition January 2009, 37 (1) 170-177; DOI: https://doi.org/10.1124/dmd.108.024166
Chang, Huai-Chia
- You have accessCytoskeleton Interruption in Human Hepatoma HepG2 Cells Induced by Ketamine Occurs Possibly through Suppression of Calcium Mobilization and Mitochondrial FunctionHuai-Chia Chang, Ta-Liang Chen and Ruei-Ming ChenDrug Metabolism and Disposition January 2009, 37 (1) 24-31; DOI: https://doi.org/10.1124/dmd.108.023325
Chen, Ruei-Ming
- You have accessCytoskeleton Interruption in Human Hepatoma HepG2 Cells Induced by Ketamine Occurs Possibly through Suppression of Calcium Mobilization and Mitochondrial FunctionHuai-Chia Chang, Ta-Liang Chen and Ruei-Ming ChenDrug Metabolism and Disposition January 2009, 37 (1) 24-31; DOI: https://doi.org/10.1124/dmd.108.023325
Chen, Shiangyuan
- You have accessApixaban Metabolism and Pharmacokinetics after Oral Administration to HumansNirmala Raghavan, Charles E. Frost, Zhigang Yu, Kan He, Haiying Zhang, W. Griffith Humphreys, Donald Pinto, Shiangyuan Chen, Samuel Bonacorsi, Pancras C. Wong and Donglu ZhangDrug Metabolism and Disposition January 2009, 37 (1) 74-81; DOI: https://doi.org/10.1124/dmd.108.023143
Chen, Ta-Liang
- You have accessCytoskeleton Interruption in Human Hepatoma HepG2 Cells Induced by Ketamine Occurs Possibly through Suppression of Calcium Mobilization and Mitochondrial FunctionHuai-Chia Chang, Ta-Liang Chen and Ruei-Ming ChenDrug Metabolism and Disposition January 2009, 37 (1) 24-31; DOI: https://doi.org/10.1124/dmd.108.023325
Cheng, Xingguo
- You have accessTissue Distribution, Gender-Divergent Expression, Ontogeny, and Chemical Induction of Multidrug Resistance Transporter Genes (Mdr1a, Mdr1b, Mdr2) in MiceYue Julia Cui, Xingguo Cheng, Yi Miao Weaver and Curtis D. KlaassenDrug Metabolism and Disposition January 2009, 37 (1) 203-210; DOI: https://doi.org/10.1124/dmd.108.023721
Choi, Yongsoo
- You have accessStructural Modulation of Oxidative Metabolism in Design of Improved Benzothiophene Selective Estrogen Receptor ModulatorsZhihui Qin, Irida Kastrati, Rezene T. Ashgodom, Daniel D. Lantvit, Cassia R. Overk, Yongsoo Choi, Richard B. van Breemen, Judy L. Bolton and Gregory R. J. ThatcherDrug Metabolism and Disposition January 2009, 37 (1) 161-169; DOI: https://doi.org/10.1124/dmd.108.023408
Court, Michael H.
- You have accessRole of NADPH-Cytochrome P450 Reductase and Cytochrome-b5/NADH-b5 Reductase in Variability of CYP3A Activity in Human Liver MicrosomesLu Gan, Lisa L. von Moltke, Lauren A. Trepanier, Jerold S. Harmatz, David J. Greenblatt and Michael H. CourtDrug Metabolism and Disposition January 2009, 37 (1) 90-96; DOI: https://doi.org/10.1124/dmd.108.023424
Cui, Yue
- You have accessThree Patterns of Cytochrome P450 Gene Expression during Liver Maturation in MiceSteven N. Hart, Yue Cui, Curtis D. Klaassen and Xiao-bo ZhongDrug Metabolism and Disposition January 2009, 37 (1) 116-121; DOI: https://doi.org/10.1124/dmd.108.023812
Cui, Yue Julia
- You have accessTissue Distribution, Gender-Divergent Expression, Ontogeny, and Chemical Induction of Multidrug Resistance Transporter Genes (Mdr1a, Mdr1b, Mdr2) in MiceYue Julia Cui, Xingguo Cheng, Yi Miao Weaver and Curtis D. KlaassenDrug Metabolism and Disposition January 2009, 37 (1) 203-210; DOI: https://doi.org/10.1124/dmd.108.023721
D
Daniel, Hannelore
- You have accessHigh-Affinity Interaction of Sartans with H+/Peptide TransportersIlka Knütter, Gabor Kottra, Wiebke Fischer, Hannelore Daniel and Matthias BrandschDrug Metabolism and Disposition January 2009, 37 (1) 143-149; DOI: https://doi.org/10.1124/dmd.108.022418
de Montellano, Paul R. Ortiz
- You have accessHuman Flavin-Containing Monooxygenase 2.1 Catalyzes Oxygenation of the Antitubercular Drugs Thiacetazone and EthionamideAsvi A. Francois, Clinton R. Nishida, Paul R. Ortiz de Montellano, Ian R. Phillips and Elizabeth A. ShephardDrug Metabolism and Disposition January 2009, 37 (1) 178-186; DOI: https://doi.org/10.1124/dmd.108.024158
DeVito, Michael J.
- You have accessIn Vitro Metabolism of Pyrethroid Pesticides by Rat and Human Hepatic Microsomes and Cytochrome P450 IsoformsEdward J. Scollon, James M. Starr, Stephen J. Godin, Michael J. DeVito and Michael F. HughesDrug Metabolism and Disposition January 2009, 37 (1) 221-228; DOI: https://doi.org/10.1124/dmd.108.022343
E
Eriksson, André H.
- You have accessTransepithelial Transport of the Group II Metabotropic Glutamate 2/3 Receptor Agonist (1S,2S,5R,6S)-2-Aminobicyclo[3.1.0]hexane-2,6-dicarboxylate (LY354740) and Its Prodrug (1S,2S,5R,6S)-2-[(2′S)-(2′-Amino)propionyl]aminobicyclo[3.1.0]hexane-2,6-dicarboxylate (LY544344)Manthena V. S. Varma, André H. Eriksson, Geri Sawada, Youngeen A. Pak, Everett J. Perkins and Cheryl L. ZimmermanDrug Metabolism and Disposition January 2009, 37 (1) 211-220; DOI: https://doi.org/10.1124/dmd.108.022012
F
Felmlee, Melanie A.
- You have accessQuantitation of Human Cytochrome P450 2D6 Protein with Immunoblot and Mass Spectrometry AnalysisAi-Ming Yu, Jun Qu, Melanie A. Felmlee, Jin Cao and Xi-Ling JiangDrug Metabolism and Disposition January 2009, 37 (1) 170-177; DOI: https://doi.org/10.1124/dmd.108.024166
Fischer, Wiebke
- You have accessHigh-Affinity Interaction of Sartans with H+/Peptide TransportersIlka Knütter, Gabor Kottra, Wiebke Fischer, Hannelore Daniel and Matthias BrandschDrug Metabolism and Disposition January 2009, 37 (1) 143-149; DOI: https://doi.org/10.1124/dmd.108.022418
Francois, Asvi A.
- You have accessHuman Flavin-Containing Monooxygenase 2.1 Catalyzes Oxygenation of the Antitubercular Drugs Thiacetazone and EthionamideAsvi A. Francois, Clinton R. Nishida, Paul R. Ortiz de Montellano, Ian R. Phillips and Elizabeth A. ShephardDrug Metabolism and Disposition January 2009, 37 (1) 178-186; DOI: https://doi.org/10.1124/dmd.108.024158
Frost, Charles E.
- You have accessApixaban Metabolism and Pharmacokinetics after Oral Administration to HumansNirmala Raghavan, Charles E. Frost, Zhigang Yu, Kan He, Haiying Zhang, W. Griffith Humphreys, Donald Pinto, Shiangyuan Chen, Samuel Bonacorsi, Pancras C. Wong and Donglu ZhangDrug Metabolism and Disposition January 2009, 37 (1) 74-81; DOI: https://doi.org/10.1124/dmd.108.023143
Fujiwara, Ryoichi
- You have accessKey Amino Acid Residues Responsible for the Differences in Substrate Specificity of Human UDP-Glucuronosyltransferase (UGT)1A9 and UGT1A8Ryoichi Fujiwara, Miki Nakajima, Hiroyuki Yamanaka and Tsuyoshi YokoiDrug Metabolism and Disposition January 2009, 37 (1) 41-46; DOI: https://doi.org/10.1124/dmd.108.022913
Fukuzaki, Koichiro
- You have accessEffect of Oral Ketoconazole on Oral and Intravenous Pharmacokinetics of Simvastatin and Its Acid in Cynomolgus MonkeysAkihito Ogasawara, Masahiro Utoh, Kazuo Nii, Ayumi Ueda, Takahiro Yoshikawa, Toshiyuki Kume and Koichiro FukuzakiDrug Metabolism and Disposition January 2009, 37 (1) 122-128; DOI: https://doi.org/10.1124/dmd.108.022574
G
Galetin, Aleksandra
- You have accessPrediction of Drug Clearance by Glucuronidation from in Vitro Data: Use of Combined Cytochrome P450 and UDP-Glucuronosyltransferase Cofactors in Alamethicin-Activated Human Liver MicrosomesPeter J. Kilford, Rowan Stringer, Bindi Sohal, J. Brian Houston and Aleksandra GaletinDrug Metabolism and Disposition January 2009, 37 (1) 82-89; DOI: https://doi.org/10.1124/dmd.108.023853
Gan, Lu
- You have accessRole of NADPH-Cytochrome P450 Reductase and Cytochrome-b5/NADH-b5 Reductase in Variability of CYP3A Activity in Human Liver MicrosomesLu Gan, Lisa L. von Moltke, Lauren A. Trepanier, Jerold S. Harmatz, David J. Greenblatt and Michael H. CourtDrug Metabolism and Disposition January 2009, 37 (1) 90-96; DOI: https://doi.org/10.1124/dmd.108.023424
Godin, Stephen J.
- You have accessIn Vitro Metabolism of Pyrethroid Pesticides by Rat and Human Hepatic Microsomes and Cytochrome P450 IsoformsEdward J. Scollon, James M. Starr, Stephen J. Godin, Michael J. DeVito and Michael F. HughesDrug Metabolism and Disposition January 2009, 37 (1) 221-228; DOI: https://doi.org/10.1124/dmd.108.022343
Gonzalez-Lobato, Lucia
- You have accessNatural Allelic Variants of Bovine ATP-Binding Cassette Transporter ABCG2: Increased Activity of the Ser581 Variant and Development of Tools for the Discovery of New ABCG2 InhibitorsGracia Merino, Rebeca Real, Marta F. Baro, Lucia Gonzalez-Lobato, Julio G. Prieto, Ana I. Alvarez and Margarita M. MarquesDrug Metabolism and Disposition January 2009, 37 (1) 5-9; DOI: https://doi.org/10.1124/dmd.108.022715
Gråsjö, Johan
- You have accessThe Multiple Depletion Curves Method Provides Accurate Estimates of Intrinsic Clearance (CLint), Maximum Velocity of the Metabolic Reaction (Vmax), and Michaelis Constant (Km): Accuracy and Robustness Evaluated through Experimental Data and Monte Carlo SimulationsErik Sjögren, Hans Lennernäs, Tommy B. Andersson, Johan Gråsjö and Ulf BredbergDrug Metabolism and Disposition January 2009, 37 (1) 47-58; DOI: https://doi.org/10.1124/dmd.108.021477
Greenblatt, David J.
- You have accessRole of NADPH-Cytochrome P450 Reductase and Cytochrome-b5/NADH-b5 Reductase in Variability of CYP3A Activity in Human Liver MicrosomesLu Gan, Lisa L. von Moltke, Lauren A. Trepanier, Jerold S. Harmatz, David J. Greenblatt and Michael H. CourtDrug Metabolism and Disposition January 2009, 37 (1) 90-96; DOI: https://doi.org/10.1124/dmd.108.023424
Guengerich, F. Peter
- You have accessDrug Interactions of Thalidomide with Midazolam and Cyclosporine A: Heterotropic Cooperativity of Human Cytochrome P450 3A5Yusuke Okada, Norie Murayama, Chihiro Yanagida, Makiko Shimizu, F. Peter Guengerich and Hiroshi YamazakiDrug Metabolism and Disposition January 2009, 37 (1) 18-23; DOI: https://doi.org/10.1124/dmd.108.024679
H
Haining, Robert L.
- You have accessExpression and Functional Analysis of CYP2D6.24, CYP2D6.26, CYP2D6.27, and CYP2D7 IsozymesWei-Yan Zhang, You-Bin Tu, Robert L. Haining and Ai-Ming YuDrug Metabolism and Disposition January 2009, 37 (1) 1-4; DOI: https://doi.org/10.1124/dmd.108.023663
Hall, Stephen D.
- You have accessPrediction of the Effect of Erythromycin, Diltiazem, and Their Metabolites, Alone and in Combination, on CYP3A4 InhibitionXin Zhang, David R. Jones and Stephen D. HallDrug Metabolism and Disposition January 2009, 37 (1) 150-160; DOI: https://doi.org/10.1124/dmd.108.022178
Harmatz, Jerold S.
- You have accessRole of NADPH-Cytochrome P450 Reductase and Cytochrome-b5/NADH-b5 Reductase in Variability of CYP3A Activity in Human Liver MicrosomesLu Gan, Lisa L. von Moltke, Lauren A. Trepanier, Jerold S. Harmatz, David J. Greenblatt and Michael H. CourtDrug Metabolism and Disposition January 2009, 37 (1) 90-96; DOI: https://doi.org/10.1124/dmd.108.023424
Hart, Steven N.
- You have accessThree Patterns of Cytochrome P450 Gene Expression during Liver Maturation in MiceSteven N. Hart, Yue Cui, Curtis D. Klaassen and Xiao-bo ZhongDrug Metabolism and Disposition January 2009, 37 (1) 116-121; DOI: https://doi.org/10.1124/dmd.108.023812
He, Kan
- You have accessApixaban Metabolism and Pharmacokinetics after Oral Administration to HumansNirmala Raghavan, Charles E. Frost, Zhigang Yu, Kan He, Haiying Zhang, W. Griffith Humphreys, Donald Pinto, Shiangyuan Chen, Samuel Bonacorsi, Pancras C. Wong and Donglu ZhangDrug Metabolism and Disposition January 2009, 37 (1) 74-81; DOI: https://doi.org/10.1124/dmd.108.023143
Houston, J. Brian
- You have accessPrediction of Drug Clearance by Glucuronidation from in Vitro Data: Use of Combined Cytochrome P450 and UDP-Glucuronosyltransferase Cofactors in Alamethicin-Activated Human Liver MicrosomesPeter J. Kilford, Rowan Stringer, Bindi Sohal, J. Brian Houston and Aleksandra GaletinDrug Metabolism and Disposition January 2009, 37 (1) 82-89; DOI: https://doi.org/10.1124/dmd.108.023853
Hua, Fengmei
- You have accessAbsolute Difference of Hepatobiliary Transporter Multidrug Resistance-Associated Protein (MRP2/Mrp2) in Liver Tissues and Isolated Hepatocytes from Rat, Dog, Monkey, and HumanNa Li, Yiqun Zhang, Fengmei Hua and Yurong LaiDrug Metabolism and Disposition January 2009, 37 (1) 66-73; DOI: https://doi.org/10.1124/dmd.108.023234
Hughes, Michael F.
- You have accessIn Vitro Metabolism of Pyrethroid Pesticides by Rat and Human Hepatic Microsomes and Cytochrome P450 IsoformsEdward J. Scollon, James M. Starr, Stephen J. Godin, Michael J. DeVito and Michael F. HughesDrug Metabolism and Disposition January 2009, 37 (1) 221-228; DOI: https://doi.org/10.1124/dmd.108.022343
Humphreys, W. Griffith
- You have accessApixaban Metabolism and Pharmacokinetics after Oral Administration to HumansNirmala Raghavan, Charles E. Frost, Zhigang Yu, Kan He, Haiying Zhang, W. Griffith Humphreys, Donald Pinto, Shiangyuan Chen, Samuel Bonacorsi, Pancras C. Wong and Donglu ZhangDrug Metabolism and Disposition January 2009, 37 (1) 74-81; DOI: https://doi.org/10.1124/dmd.108.023143
Hunt, C. Anthony
- You have accessDiscovering Plausible Mechanistic Details of Hepatic Drug InteractionsTai Ning Lam and C. Anthony HuntDrug Metabolism and Disposition January 2009, 37 (1) 237-246; DOI: https://doi.org/10.1124/dmd.108.023820
Hutzler, J. Matthew
- You have accessIs 1-Aminobenzotriazole an Appropriate in Vitro Tool as a Nonspecific Cytochrome P450 Inactivator?Collette D. Linder, Nicole A. Renaud and J. Matthew HutzlerDrug Metabolism and Disposition January 2009, 37 (1) 10-13; DOI: https://doi.org/10.1124/dmd.108.024075
- You have accessMechanism-Based Inactivation of Cytochrome P450 2C9 by Tienilic Acid and (±)-Suprofen: A Comparison of Kinetics and Probe Substrate SelectionJ. Matthew Hutzler, Larissa M. Balogh, Michael Zientek, Vikas Kumar and Timothy S. TracyDrug Metabolism and Disposition January 2009, 37 (1) 59-65; DOI: https://doi.org/10.1124/dmd.108.023358
J
Jiang, Xi-Ling
- You have accessQuantitation of Human Cytochrome P450 2D6 Protein with Immunoblot and Mass Spectrometry AnalysisAi-Ming Yu, Jun Qu, Melanie A. Felmlee, Jin Cao and Xi-Ling JiangDrug Metabolism and Disposition January 2009, 37 (1) 170-177; DOI: https://doi.org/10.1124/dmd.108.024166
Jones, David R.
- You have accessPrediction of the Effect of Erythromycin, Diltiazem, and Their Metabolites, Alone and in Combination, on CYP3A4 InhibitionXin Zhang, David R. Jones and Stephen D. HallDrug Metabolism and Disposition January 2009, 37 (1) 150-160; DOI: https://doi.org/10.1124/dmd.108.022178
K
Kalvass, J. Cory
- You have accessMicrodialysis Evaluation of Atomoxetine Brain Penetration and Central Nervous System Pharmacokinetics in RatsWilliam Kielbasa, J. Cory Kalvass and Robert StratfordDrug Metabolism and Disposition January 2009, 37 (1) 137-142; DOI: https://doi.org/10.1124/dmd.108.023119
Kamataki, Tetsuya
- You have accessA Null Allele Impairs Function of CYP2C76 Gene in Cynomolgus Monkeys: A Possible Genetic Tool for Generation of a Better Animal Model in Drug MetabolismYasuhiro Uno, Hiroko Sakuraba, Shotaro Uehara, Takayuki Kumano, Kiyomi Matsuno, Chika Nakamura, Go Kito, Tetsuya Kamataki and Ryoichi NagataDrug Metabolism and Disposition January 2009, 37 (1) 14-17; DOI: https://doi.org/10.1124/dmd.108.023622
Kastrati, Irida
- You have accessStructural Modulation of Oxidative Metabolism in Design of Improved Benzothiophene Selective Estrogen Receptor ModulatorsZhihui Qin, Irida Kastrati, Rezene T. Ashgodom, Daniel D. Lantvit, Cassia R. Overk, Yongsoo Choi, Richard B. van Breemen, Judy L. Bolton and Gregory R. J. ThatcherDrug Metabolism and Disposition January 2009, 37 (1) 161-169; DOI: https://doi.org/10.1124/dmd.108.023408
Kielbasa, William
- You have accessMicrodialysis Evaluation of Atomoxetine Brain Penetration and Central Nervous System Pharmacokinetics in RatsWilliam Kielbasa, J. Cory Kalvass and Robert StratfordDrug Metabolism and Disposition January 2009, 37 (1) 137-142; DOI: https://doi.org/10.1124/dmd.108.023119
Kilford, Peter J.
- You have accessPrediction of Drug Clearance by Glucuronidation from in Vitro Data: Use of Combined Cytochrome P450 and UDP-Glucuronosyltransferase Cofactors in Alamethicin-Activated Human Liver MicrosomesPeter J. Kilford, Rowan Stringer, Bindi Sohal, J. Brian Houston and Aleksandra GaletinDrug Metabolism and Disposition January 2009, 37 (1) 82-89; DOI: https://doi.org/10.1124/dmd.108.023853
Kito, Go
- You have accessA Null Allele Impairs Function of CYP2C76 Gene in Cynomolgus Monkeys: A Possible Genetic Tool for Generation of a Better Animal Model in Drug MetabolismYasuhiro Uno, Hiroko Sakuraba, Shotaro Uehara, Takayuki Kumano, Kiyomi Matsuno, Chika Nakamura, Go Kito, Tetsuya Kamataki and Ryoichi NagataDrug Metabolism and Disposition January 2009, 37 (1) 14-17; DOI: https://doi.org/10.1124/dmd.108.023622
Klaassen, Curtis D.
- You have accessCircadian Expression Profiles of Drug-Processing Genes and Transcription Factors in Mouse LiverYu-Kun Jennifer Zhang, Ronnie L. Yeager and Curtis D. KlaassenDrug Metabolism and Disposition January 2009, 37 (1) 106-115; DOI: https://doi.org/10.1124/dmd.108.024174
- You have accessThree Patterns of Cytochrome P450 Gene Expression during Liver Maturation in MiceSteven N. Hart, Yue Cui, Curtis D. Klaassen and Xiao-bo ZhongDrug Metabolism and Disposition January 2009, 37 (1) 116-121; DOI: https://doi.org/10.1124/dmd.108.023812
- You have accessTissue Distribution, Gender-Divergent Expression, Ontogeny, and Chemical Induction of Multidrug Resistance Transporter Genes (Mdr1a, Mdr1b, Mdr2) in MiceYue Julia Cui, Xingguo Cheng, Yi Miao Weaver and Curtis D. KlaassenDrug Metabolism and Disposition January 2009, 37 (1) 203-210; DOI: https://doi.org/10.1124/dmd.108.023721
Knütter, Ilka
- You have accessHigh-Affinity Interaction of Sartans with H+/Peptide TransportersIlka Knütter, Gabor Kottra, Wiebke Fischer, Hannelore Daniel and Matthias BrandschDrug Metabolism and Disposition January 2009, 37 (1) 143-149; DOI: https://doi.org/10.1124/dmd.108.022418
Kottra, Gabor
- You have accessHigh-Affinity Interaction of Sartans with H+/Peptide TransportersIlka Knütter, Gabor Kottra, Wiebke Fischer, Hannelore Daniel and Matthias BrandschDrug Metabolism and Disposition January 2009, 37 (1) 143-149; DOI: https://doi.org/10.1124/dmd.108.022418
Kumano, Takayuki
- You have accessA Null Allele Impairs Function of CYP2C76 Gene in Cynomolgus Monkeys: A Possible Genetic Tool for Generation of a Better Animal Model in Drug MetabolismYasuhiro Uno, Hiroko Sakuraba, Shotaro Uehara, Takayuki Kumano, Kiyomi Matsuno, Chika Nakamura, Go Kito, Tetsuya Kamataki and Ryoichi NagataDrug Metabolism and Disposition January 2009, 37 (1) 14-17; DOI: https://doi.org/10.1124/dmd.108.023622
Kumar, Vikas
- You have accessMechanism-Based Inactivation of Cytochrome P450 2C9 by Tienilic Acid and (±)-Suprofen: A Comparison of Kinetics and Probe Substrate SelectionJ. Matthew Hutzler, Larissa M. Balogh, Michael Zientek, Vikas Kumar and Timothy S. TracyDrug Metabolism and Disposition January 2009, 37 (1) 59-65; DOI: https://doi.org/10.1124/dmd.108.023358
Kume, Toshiyuki
- You have accessEffect of Oral Ketoconazole on Oral and Intravenous Pharmacokinetics of Simvastatin and Its Acid in Cynomolgus MonkeysAkihito Ogasawara, Masahiro Utoh, Kazuo Nii, Ayumi Ueda, Takahiro Yoshikawa, Toshiyuki Kume and Koichiro FukuzakiDrug Metabolism and Disposition January 2009, 37 (1) 122-128; DOI: https://doi.org/10.1124/dmd.108.022574
L
Lagas, Jurjen S.
- You have accessTransport of Diclofenac by Breast Cancer Resistance Protein (ABCG2) and Stimulation of Multidrug Resistance Protein 2 (ABCC2)-Mediated Drug Transport by Diclofenac and BenzbromaroneJurjen S. Lagas, Cornelia M. M. van der Kruijssen, Koen van de Wetering, Jos H. Beijnen and Alfred H. SchinkelDrug Metabolism and Disposition January 2009, 37 (1) 129-136; DOI: https://doi.org/10.1124/dmd.108.023200
Lai, Yurong
- You have accessAbsolute Difference of Hepatobiliary Transporter Multidrug Resistance-Associated Protein (MRP2/Mrp2) in Liver Tissues and Isolated Hepatocytes from Rat, Dog, Monkey, and HumanNa Li, Yiqun Zhang, Fengmei Hua and Yurong LaiDrug Metabolism and Disposition January 2009, 37 (1) 66-73; DOI: https://doi.org/10.1124/dmd.108.023234
Lam, Tai Ning
- You have accessDiscovering Plausible Mechanistic Details of Hepatic Drug InteractionsTai Ning Lam and C. Anthony HuntDrug Metabolism and Disposition January 2009, 37 (1) 237-246; DOI: https://doi.org/10.1124/dmd.108.023820
Lantvit, Daniel D.
- You have accessStructural Modulation of Oxidative Metabolism in Design of Improved Benzothiophene Selective Estrogen Receptor ModulatorsZhihui Qin, Irida Kastrati, Rezene T. Ashgodom, Daniel D. Lantvit, Cassia R. Overk, Yongsoo Choi, Richard B. van Breemen, Judy L. Bolton and Gregory R. J. ThatcherDrug Metabolism and Disposition January 2009, 37 (1) 161-169; DOI: https://doi.org/10.1124/dmd.108.023408
Lennernäs, Hans
- You have accessThe Multiple Depletion Curves Method Provides Accurate Estimates of Intrinsic Clearance (CLint), Maximum Velocity of the Metabolic Reaction (Vmax), and Michaelis Constant (Km): Accuracy and Robustness Evaluated through Experimental Data and Monte Carlo SimulationsErik Sjögren, Hans Lennernäs, Tommy B. Andersson, Johan Gråsjö and Ulf BredbergDrug Metabolism and Disposition January 2009, 37 (1) 47-58; DOI: https://doi.org/10.1124/dmd.108.021477
Li, Na
- You have accessAbsolute Difference of Hepatobiliary Transporter Multidrug Resistance-Associated Protein (MRP2/Mrp2) in Liver Tissues and Isolated Hepatocytes from Rat, Dog, Monkey, and HumanNa Li, Yiqun Zhang, Fengmei Hua and Yurong LaiDrug Metabolism and Disposition January 2009, 37 (1) 66-73; DOI: https://doi.org/10.1124/dmd.108.023234
Linder, Collette D.
- You have accessIs 1-Aminobenzotriazole an Appropriate in Vitro Tool as a Nonspecific Cytochrome P450 Inactivator?Collette D. Linder, Nicole A. Renaud and J. Matthew HutzlerDrug Metabolism and Disposition January 2009, 37 (1) 10-13; DOI: https://doi.org/10.1124/dmd.108.024075
M
Marques, Margarita M.
- You have accessNatural Allelic Variants of Bovine ATP-Binding Cassette Transporter ABCG2: Increased Activity of the Ser581 Variant and Development of Tools for the Discovery of New ABCG2 InhibitorsGracia Merino, Rebeca Real, Marta F. Baro, Lucia Gonzalez-Lobato, Julio G. Prieto, Ana I. Alvarez and Margarita M. MarquesDrug Metabolism and Disposition January 2009, 37 (1) 5-9; DOI: https://doi.org/10.1124/dmd.108.022715
Matsuno, Kiyomi
- You have accessA Null Allele Impairs Function of CYP2C76 Gene in Cynomolgus Monkeys: A Possible Genetic Tool for Generation of a Better Animal Model in Drug MetabolismYasuhiro Uno, Hiroko Sakuraba, Shotaro Uehara, Takayuki Kumano, Kiyomi Matsuno, Chika Nakamura, Go Kito, Tetsuya Kamataki and Ryoichi NagataDrug Metabolism and Disposition January 2009, 37 (1) 14-17; DOI: https://doi.org/10.1124/dmd.108.023622
Merino, Gracia
- You have accessNatural Allelic Variants of Bovine ATP-Binding Cassette Transporter ABCG2: Increased Activity of the Ser581 Variant and Development of Tools for the Discovery of New ABCG2 InhibitorsGracia Merino, Rebeca Real, Marta F. Baro, Lucia Gonzalez-Lobato, Julio G. Prieto, Ana I. Alvarez and Margarita M. MarquesDrug Metabolism and Disposition January 2009, 37 (1) 5-9; DOI: https://doi.org/10.1124/dmd.108.022715
Miyata, Masaaki
- You have accessRole of Enzymatic N-Hydroxylation and Reduction in Flutamide Metabolite-Induced Liver ToxicityMasato Ohbuchi, Masaaki Miyata, Daichi Nagai, Miki Shimada, Kouichi Yoshinari and Yasushi YamazoeDrug Metabolism and Disposition January 2009, 37 (1) 97-105; DOI: https://doi.org/10.1124/dmd.108.021964
Murayama, Norie
- You have accessDrug Interactions of Thalidomide with Midazolam and Cyclosporine A: Heterotropic Cooperativity of Human Cytochrome P450 3A5Yusuke Okada, Norie Murayama, Chihiro Yanagida, Makiko Shimizu, F. Peter Guengerich and Hiroshi YamazakiDrug Metabolism and Disposition January 2009, 37 (1) 18-23; DOI: https://doi.org/10.1124/dmd.108.024679
N
Nagai, Daichi
- You have accessRole of Enzymatic N-Hydroxylation and Reduction in Flutamide Metabolite-Induced Liver ToxicityMasato Ohbuchi, Masaaki Miyata, Daichi Nagai, Miki Shimada, Kouichi Yoshinari and Yasushi YamazoeDrug Metabolism and Disposition January 2009, 37 (1) 97-105; DOI: https://doi.org/10.1124/dmd.108.021964
Nagata, Ryoichi
- You have accessA Null Allele Impairs Function of CYP2C76 Gene in Cynomolgus Monkeys: A Possible Genetic Tool for Generation of a Better Animal Model in Drug MetabolismYasuhiro Uno, Hiroko Sakuraba, Shotaro Uehara, Takayuki Kumano, Kiyomi Matsuno, Chika Nakamura, Go Kito, Tetsuya Kamataki and Ryoichi NagataDrug Metabolism and Disposition January 2009, 37 (1) 14-17; DOI: https://doi.org/10.1124/dmd.108.023622
Nakajima, Miki
- You have accessKey Amino Acid Residues Responsible for the Differences in Substrate Specificity of Human UDP-Glucuronosyltransferase (UGT)1A9 and UGT1A8Ryoichi Fujiwara, Miki Nakajima, Hiroyuki Yamanaka and Tsuyoshi YokoiDrug Metabolism and Disposition January 2009, 37 (1) 41-46; DOI: https://doi.org/10.1124/dmd.108.022913
Nakajin, Shizuo
- You have accessDetermination of mRNA Expression of Human UDP-Glucuronosyltransferases and Application for Localization in Various Human Tissues by Real-Time Reverse Transcriptase-Polymerase Chain ReactionShuji Ohno and Shizuo NakajinDrug Metabolism and Disposition January 2009, 37 (1) 32-40; DOI: https://doi.org/10.1124/dmd.108.023598
Nakamura, Chika
- You have accessA Null Allele Impairs Function of CYP2C76 Gene in Cynomolgus Monkeys: A Possible Genetic Tool for Generation of a Better Animal Model in Drug MetabolismYasuhiro Uno, Hiroko Sakuraba, Shotaro Uehara, Takayuki Kumano, Kiyomi Matsuno, Chika Nakamura, Go Kito, Tetsuya Kamataki and Ryoichi NagataDrug Metabolism and Disposition January 2009, 37 (1) 14-17; DOI: https://doi.org/10.1124/dmd.108.023622
Nii, Kazuo
- You have accessEffect of Oral Ketoconazole on Oral and Intravenous Pharmacokinetics of Simvastatin and Its Acid in Cynomolgus MonkeysAkihito Ogasawara, Masahiro Utoh, Kazuo Nii, Ayumi Ueda, Takahiro Yoshikawa, Toshiyuki Kume and Koichiro FukuzakiDrug Metabolism and Disposition January 2009, 37 (1) 122-128; DOI: https://doi.org/10.1124/dmd.108.022574
Nishida, Clinton R.
- You have accessHuman Flavin-Containing Monooxygenase 2.1 Catalyzes Oxygenation of the Antitubercular Drugs Thiacetazone and EthionamideAsvi A. Francois, Clinton R. Nishida, Paul R. Ortiz de Montellano, Ian R. Phillips and Elizabeth A. ShephardDrug Metabolism and Disposition January 2009, 37 (1) 178-186; DOI: https://doi.org/10.1124/dmd.108.024158
O
Ogasawara, Akihito
- You have accessEffect of Oral Ketoconazole on Oral and Intravenous Pharmacokinetics of Simvastatin and Its Acid in Cynomolgus MonkeysAkihito Ogasawara, Masahiro Utoh, Kazuo Nii, Ayumi Ueda, Takahiro Yoshikawa, Toshiyuki Kume and Koichiro FukuzakiDrug Metabolism and Disposition January 2009, 37 (1) 122-128; DOI: https://doi.org/10.1124/dmd.108.022574
Ohbuchi, Masato
- You have accessRole of Enzymatic N-Hydroxylation and Reduction in Flutamide Metabolite-Induced Liver ToxicityMasato Ohbuchi, Masaaki Miyata, Daichi Nagai, Miki Shimada, Kouichi Yoshinari and Yasushi YamazoeDrug Metabolism and Disposition January 2009, 37 (1) 97-105; DOI: https://doi.org/10.1124/dmd.108.021964
Ohno, Shuji
- You have accessDetermination of mRNA Expression of Human UDP-Glucuronosyltransferases and Application for Localization in Various Human Tissues by Real-Time Reverse Transcriptase-Polymerase Chain ReactionShuji Ohno and Shizuo NakajinDrug Metabolism and Disposition January 2009, 37 (1) 32-40; DOI: https://doi.org/10.1124/dmd.108.023598
Okada, Yusuke
- You have accessDrug Interactions of Thalidomide with Midazolam and Cyclosporine A: Heterotropic Cooperativity of Human Cytochrome P450 3A5Yusuke Okada, Norie Murayama, Chihiro Yanagida, Makiko Shimizu, F. Peter Guengerich and Hiroshi YamazakiDrug Metabolism and Disposition January 2009, 37 (1) 18-23; DOI: https://doi.org/10.1124/dmd.108.024679
Overk, Cassia R.
- You have accessStructural Modulation of Oxidative Metabolism in Design of Improved Benzothiophene Selective Estrogen Receptor ModulatorsZhihui Qin, Irida Kastrati, Rezene T. Ashgodom, Daniel D. Lantvit, Cassia R. Overk, Yongsoo Choi, Richard B. van Breemen, Judy L. Bolton and Gregory R. J. ThatcherDrug Metabolism and Disposition January 2009, 37 (1) 161-169; DOI: https://doi.org/10.1124/dmd.108.023408
P
Pak, Youngeen A.
- You have accessTransepithelial Transport of the Group II Metabotropic Glutamate 2/3 Receptor Agonist (1S,2S,5R,6S)-2-Aminobicyclo[3.1.0]hexane-2,6-dicarboxylate (LY354740) and Its Prodrug (1S,2S,5R,6S)-2-[(2′S)-(2′-Amino)propionyl]aminobicyclo[3.1.0]hexane-2,6-dicarboxylate (LY544344)Manthena V. S. Varma, André H. Eriksson, Geri Sawada, Youngeen A. Pak, Everett J. Perkins and Cheryl L. ZimmermanDrug Metabolism and Disposition January 2009, 37 (1) 211-220; DOI: https://doi.org/10.1124/dmd.108.022012
Pang, K. Sandy
- You have accessDisparity in Intestine Disposition between Formed and Preformed Metabolites and Implications: A Theoretical StudyHuadong Sun and K. Sandy PangDrug Metabolism and Disposition January 2009, 37 (1) 187-202; DOI: https://doi.org/10.1124/dmd.108.022483
Perkins, Everett J.
- You have accessTransepithelial Transport of the Group II Metabotropic Glutamate 2/3 Receptor Agonist (1S,2S,5R,6S)-2-Aminobicyclo[3.1.0]hexane-2,6-dicarboxylate (LY354740) and Its Prodrug (1S,2S,5R,6S)-2-[(2′S)-(2′-Amino)propionyl]aminobicyclo[3.1.0]hexane-2,6-dicarboxylate (LY544344)Manthena V. S. Varma, André H. Eriksson, Geri Sawada, Youngeen A. Pak, Everett J. Perkins and Cheryl L. ZimmermanDrug Metabolism and Disposition January 2009, 37 (1) 211-220; DOI: https://doi.org/10.1124/dmd.108.022012
Phillips, Ian R.
- You have accessHuman Flavin-Containing Monooxygenase 2.1 Catalyzes Oxygenation of the Antitubercular Drugs Thiacetazone and EthionamideAsvi A. Francois, Clinton R. Nishida, Paul R. Ortiz de Montellano, Ian R. Phillips and Elizabeth A. ShephardDrug Metabolism and Disposition January 2009, 37 (1) 178-186; DOI: https://doi.org/10.1124/dmd.108.024158
Pinto, Donald
- You have accessApixaban Metabolism and Pharmacokinetics after Oral Administration to HumansNirmala Raghavan, Charles E. Frost, Zhigang Yu, Kan He, Haiying Zhang, W. Griffith Humphreys, Donald Pinto, Shiangyuan Chen, Samuel Bonacorsi, Pancras C. Wong and Donglu ZhangDrug Metabolism and Disposition January 2009, 37 (1) 74-81; DOI: https://doi.org/10.1124/dmd.108.023143
Prieto, Julio G.
- You have accessNatural Allelic Variants of Bovine ATP-Binding Cassette Transporter ABCG2: Increased Activity of the Ser581 Variant and Development of Tools for the Discovery of New ABCG2 InhibitorsGracia Merino, Rebeca Real, Marta F. Baro, Lucia Gonzalez-Lobato, Julio G. Prieto, Ana I. Alvarez and Margarita M. MarquesDrug Metabolism and Disposition January 2009, 37 (1) 5-9; DOI: https://doi.org/10.1124/dmd.108.022715
Q
Qin, Zhihui
- You have accessStructural Modulation of Oxidative Metabolism in Design of Improved Benzothiophene Selective Estrogen Receptor ModulatorsZhihui Qin, Irida Kastrati, Rezene T. Ashgodom, Daniel D. Lantvit, Cassia R. Overk, Yongsoo Choi, Richard B. van Breemen, Judy L. Bolton and Gregory R. J. ThatcherDrug Metabolism and Disposition January 2009, 37 (1) 161-169; DOI: https://doi.org/10.1124/dmd.108.023408
Qu, Jun
- You have accessQuantitation of Human Cytochrome P450 2D6 Protein with Immunoblot and Mass Spectrometry AnalysisAi-Ming Yu, Jun Qu, Melanie A. Felmlee, Jin Cao and Xi-Ling JiangDrug Metabolism and Disposition January 2009, 37 (1) 170-177; DOI: https://doi.org/10.1124/dmd.108.024166
R
Raghavan, Nirmala
- You have accessApixaban Metabolism and Pharmacokinetics after Oral Administration to HumansNirmala Raghavan, Charles E. Frost, Zhigang Yu, Kan He, Haiying Zhang, W. Griffith Humphreys, Donald Pinto, Shiangyuan Chen, Samuel Bonacorsi, Pancras C. Wong and Donglu ZhangDrug Metabolism and Disposition January 2009, 37 (1) 74-81; DOI: https://doi.org/10.1124/dmd.108.023143
Real, Rebeca
- You have accessNatural Allelic Variants of Bovine ATP-Binding Cassette Transporter ABCG2: Increased Activity of the Ser581 Variant and Development of Tools for the Discovery of New ABCG2 InhibitorsGracia Merino, Rebeca Real, Marta F. Baro, Lucia Gonzalez-Lobato, Julio G. Prieto, Ana I. Alvarez and Margarita M. MarquesDrug Metabolism and Disposition January 2009, 37 (1) 5-9; DOI: https://doi.org/10.1124/dmd.108.022715
Remmel, Rory P.
- You have accessEffect of Aging on Glucuronidation of Valproic Acid in Human Liver Microsomes and the Role of UDP-Glucuronosyltransferase UGT1A4, UGT1A8, and UGT1A10Upendra A. Argikar and Rory P. RemmelDrug Metabolism and Disposition January 2009, 37 (1) 229-236; DOI: https://doi.org/10.1124/dmd.108.022426
Renaud, Nicole A.
- You have accessIs 1-Aminobenzotriazole an Appropriate in Vitro Tool as a Nonspecific Cytochrome P450 Inactivator?Collette D. Linder, Nicole A. Renaud and J. Matthew HutzlerDrug Metabolism and Disposition January 2009, 37 (1) 10-13; DOI: https://doi.org/10.1124/dmd.108.024075
S
Sakuraba, Hiroko
- You have accessA Null Allele Impairs Function of CYP2C76 Gene in Cynomolgus Monkeys: A Possible Genetic Tool for Generation of a Better Animal Model in Drug MetabolismYasuhiro Uno, Hiroko Sakuraba, Shotaro Uehara, Takayuki Kumano, Kiyomi Matsuno, Chika Nakamura, Go Kito, Tetsuya Kamataki and Ryoichi NagataDrug Metabolism and Disposition January 2009, 37 (1) 14-17; DOI: https://doi.org/10.1124/dmd.108.023622
Sawada, Geri
- You have accessTransepithelial Transport of the Group II Metabotropic Glutamate 2/3 Receptor Agonist (1S,2S,5R,6S)-2-Aminobicyclo[3.1.0]hexane-2,6-dicarboxylate (LY354740) and Its Prodrug (1S,2S,5R,6S)-2-[(2′S)-(2′-Amino)propionyl]aminobicyclo[3.1.0]hexane-2,6-dicarboxylate (LY544344)Manthena V. S. Varma, André H. Eriksson, Geri Sawada, Youngeen A. Pak, Everett J. Perkins and Cheryl L. ZimmermanDrug Metabolism and Disposition January 2009, 37 (1) 211-220; DOI: https://doi.org/10.1124/dmd.108.022012
Schinkel, Alfred H.
- You have accessTransport of Diclofenac by Breast Cancer Resistance Protein (ABCG2) and Stimulation of Multidrug Resistance Protein 2 (ABCC2)-Mediated Drug Transport by Diclofenac and BenzbromaroneJurjen S. Lagas, Cornelia M. M. van der Kruijssen, Koen van de Wetering, Jos H. Beijnen and Alfred H. SchinkelDrug Metabolism and Disposition January 2009, 37 (1) 129-136; DOI: https://doi.org/10.1124/dmd.108.023200
Scollon, Edward J.
- You have accessIn Vitro Metabolism of Pyrethroid Pesticides by Rat and Human Hepatic Microsomes and Cytochrome P450 IsoformsEdward J. Scollon, James M. Starr, Stephen J. Godin, Michael J. DeVito and Michael F. HughesDrug Metabolism and Disposition January 2009, 37 (1) 221-228; DOI: https://doi.org/10.1124/dmd.108.022343
Shephard, Elizabeth A.
- You have accessHuman Flavin-Containing Monooxygenase 2.1 Catalyzes Oxygenation of the Antitubercular Drugs Thiacetazone and EthionamideAsvi A. Francois, Clinton R. Nishida, Paul R. Ortiz de Montellano, Ian R. Phillips and Elizabeth A. ShephardDrug Metabolism and Disposition January 2009, 37 (1) 178-186; DOI: https://doi.org/10.1124/dmd.108.024158
Shimada, Miki
- You have accessRole of Enzymatic N-Hydroxylation and Reduction in Flutamide Metabolite-Induced Liver ToxicityMasato Ohbuchi, Masaaki Miyata, Daichi Nagai, Miki Shimada, Kouichi Yoshinari and Yasushi YamazoeDrug Metabolism and Disposition January 2009, 37 (1) 97-105; DOI: https://doi.org/10.1124/dmd.108.021964
Shimizu, Makiko
- You have accessDrug Interactions of Thalidomide with Midazolam and Cyclosporine A: Heterotropic Cooperativity of Human Cytochrome P450 3A5Yusuke Okada, Norie Murayama, Chihiro Yanagida, Makiko Shimizu, F. Peter Guengerich and Hiroshi YamazakiDrug Metabolism and Disposition January 2009, 37 (1) 18-23; DOI: https://doi.org/10.1124/dmd.108.024679
Sjögren, Erik
- You have accessThe Multiple Depletion Curves Method Provides Accurate Estimates of Intrinsic Clearance (CLint), Maximum Velocity of the Metabolic Reaction (Vmax), and Michaelis Constant (Km): Accuracy and Robustness Evaluated through Experimental Data and Monte Carlo SimulationsErik Sjögren, Hans Lennernäs, Tommy B. Andersson, Johan Gråsjö and Ulf BredbergDrug Metabolism and Disposition January 2009, 37 (1) 47-58; DOI: https://doi.org/10.1124/dmd.108.021477
Sohal, Bindi
- You have accessPrediction of Drug Clearance by Glucuronidation from in Vitro Data: Use of Combined Cytochrome P450 and UDP-Glucuronosyltransferase Cofactors in Alamethicin-Activated Human Liver MicrosomesPeter J. Kilford, Rowan Stringer, Bindi Sohal, J. Brian Houston and Aleksandra GaletinDrug Metabolism and Disposition January 2009, 37 (1) 82-89; DOI: https://doi.org/10.1124/dmd.108.023853
Starr, James M.
- You have accessIn Vitro Metabolism of Pyrethroid Pesticides by Rat and Human Hepatic Microsomes and Cytochrome P450 IsoformsEdward J. Scollon, James M. Starr, Stephen J. Godin, Michael J. DeVito and Michael F. HughesDrug Metabolism and Disposition January 2009, 37 (1) 221-228; DOI: https://doi.org/10.1124/dmd.108.022343
Stratford, Robert
- You have accessMicrodialysis Evaluation of Atomoxetine Brain Penetration and Central Nervous System Pharmacokinetics in RatsWilliam Kielbasa, J. Cory Kalvass and Robert StratfordDrug Metabolism and Disposition January 2009, 37 (1) 137-142; DOI: https://doi.org/10.1124/dmd.108.023119
Stringer, Rowan
- You have accessPrediction of Drug Clearance by Glucuronidation from in Vitro Data: Use of Combined Cytochrome P450 and UDP-Glucuronosyltransferase Cofactors in Alamethicin-Activated Human Liver MicrosomesPeter J. Kilford, Rowan Stringer, Bindi Sohal, J. Brian Houston and Aleksandra GaletinDrug Metabolism and Disposition January 2009, 37 (1) 82-89; DOI: https://doi.org/10.1124/dmd.108.023853
Sun, Huadong
- You have accessDisparity in Intestine Disposition between Formed and Preformed Metabolites and Implications: A Theoretical StudyHuadong Sun and K. Sandy PangDrug Metabolism and Disposition January 2009, 37 (1) 187-202; DOI: https://doi.org/10.1124/dmd.108.022483
T
Thatcher, Gregory R. J.
- You have accessStructural Modulation of Oxidative Metabolism in Design of Improved Benzothiophene Selective Estrogen Receptor ModulatorsZhihui Qin, Irida Kastrati, Rezene T. Ashgodom, Daniel D. Lantvit, Cassia R. Overk, Yongsoo Choi, Richard B. van Breemen, Judy L. Bolton and Gregory R. J. ThatcherDrug Metabolism and Disposition January 2009, 37 (1) 161-169; DOI: https://doi.org/10.1124/dmd.108.023408
Tracy, Timothy S.
- You have accessMechanism-Based Inactivation of Cytochrome P450 2C9 by Tienilic Acid and (±)-Suprofen: A Comparison of Kinetics and Probe Substrate SelectionJ. Matthew Hutzler, Larissa M. Balogh, Michael Zientek, Vikas Kumar and Timothy S. TracyDrug Metabolism and Disposition January 2009, 37 (1) 59-65; DOI: https://doi.org/10.1124/dmd.108.023358
Trepanier, Lauren A.
- You have accessRole of NADPH-Cytochrome P450 Reductase and Cytochrome-b5/NADH-b5 Reductase in Variability of CYP3A Activity in Human Liver MicrosomesLu Gan, Lisa L. von Moltke, Lauren A. Trepanier, Jerold S. Harmatz, David J. Greenblatt and Michael H. CourtDrug Metabolism and Disposition January 2009, 37 (1) 90-96; DOI: https://doi.org/10.1124/dmd.108.023424
Tu, You-Bin
- You have accessExpression and Functional Analysis of CYP2D6.24, CYP2D6.26, CYP2D6.27, and CYP2D7 IsozymesWei-Yan Zhang, You-Bin Tu, Robert L. Haining and Ai-Ming YuDrug Metabolism and Disposition January 2009, 37 (1) 1-4; DOI: https://doi.org/10.1124/dmd.108.023663
U
Ueda, Ayumi
- You have accessEffect of Oral Ketoconazole on Oral and Intravenous Pharmacokinetics of Simvastatin and Its Acid in Cynomolgus MonkeysAkihito Ogasawara, Masahiro Utoh, Kazuo Nii, Ayumi Ueda, Takahiro Yoshikawa, Toshiyuki Kume and Koichiro FukuzakiDrug Metabolism and Disposition January 2009, 37 (1) 122-128; DOI: https://doi.org/10.1124/dmd.108.022574
Uehara, Shotaro
- You have accessA Null Allele Impairs Function of CYP2C76 Gene in Cynomolgus Monkeys: A Possible Genetic Tool for Generation of a Better Animal Model in Drug MetabolismYasuhiro Uno, Hiroko Sakuraba, Shotaro Uehara, Takayuki Kumano, Kiyomi Matsuno, Chika Nakamura, Go Kito, Tetsuya Kamataki and Ryoichi NagataDrug Metabolism and Disposition January 2009, 37 (1) 14-17; DOI: https://doi.org/10.1124/dmd.108.023622
Uno, Yasuhiro
- You have accessA Null Allele Impairs Function of CYP2C76 Gene in Cynomolgus Monkeys: A Possible Genetic Tool for Generation of a Better Animal Model in Drug MetabolismYasuhiro Uno, Hiroko Sakuraba, Shotaro Uehara, Takayuki Kumano, Kiyomi Matsuno, Chika Nakamura, Go Kito, Tetsuya Kamataki and Ryoichi NagataDrug Metabolism and Disposition January 2009, 37 (1) 14-17; DOI: https://doi.org/10.1124/dmd.108.023622
Utoh, Masahiro
- You have accessEffect of Oral Ketoconazole on Oral and Intravenous Pharmacokinetics of Simvastatin and Its Acid in Cynomolgus MonkeysAkihito Ogasawara, Masahiro Utoh, Kazuo Nii, Ayumi Ueda, Takahiro Yoshikawa, Toshiyuki Kume and Koichiro FukuzakiDrug Metabolism and Disposition January 2009, 37 (1) 122-128; DOI: https://doi.org/10.1124/dmd.108.022574
V
van Breemen, Richard B.
- You have accessStructural Modulation of Oxidative Metabolism in Design of Improved Benzothiophene Selective Estrogen Receptor ModulatorsZhihui Qin, Irida Kastrati, Rezene T. Ashgodom, Daniel D. Lantvit, Cassia R. Overk, Yongsoo Choi, Richard B. van Breemen, Judy L. Bolton and Gregory R. J. ThatcherDrug Metabolism and Disposition January 2009, 37 (1) 161-169; DOI: https://doi.org/10.1124/dmd.108.023408
van der Kruijssen, Cornelia M. M.
- You have accessTransport of Diclofenac by Breast Cancer Resistance Protein (ABCG2) and Stimulation of Multidrug Resistance Protein 2 (ABCC2)-Mediated Drug Transport by Diclofenac and BenzbromaroneJurjen S. Lagas, Cornelia M. M. van der Kruijssen, Koen van de Wetering, Jos H. Beijnen and Alfred H. SchinkelDrug Metabolism and Disposition January 2009, 37 (1) 129-136; DOI: https://doi.org/10.1124/dmd.108.023200
van de Wetering, Koen
- You have accessTransport of Diclofenac by Breast Cancer Resistance Protein (ABCG2) and Stimulation of Multidrug Resistance Protein 2 (ABCC2)-Mediated Drug Transport by Diclofenac and BenzbromaroneJurjen S. Lagas, Cornelia M. M. van der Kruijssen, Koen van de Wetering, Jos H. Beijnen and Alfred H. SchinkelDrug Metabolism and Disposition January 2009, 37 (1) 129-136; DOI: https://doi.org/10.1124/dmd.108.023200
Varma, Manthena V. S.
- You have accessTransepithelial Transport of the Group II Metabotropic Glutamate 2/3 Receptor Agonist (1S,2S,5R,6S)-2-Aminobicyclo[3.1.0]hexane-2,6-dicarboxylate (LY354740) and Its Prodrug (1S,2S,5R,6S)-2-[(2′S)-(2′-Amino)propionyl]aminobicyclo[3.1.0]hexane-2,6-dicarboxylate (LY544344)Manthena V. S. Varma, André H. Eriksson, Geri Sawada, Youngeen A. Pak, Everett J. Perkins and Cheryl L. ZimmermanDrug Metabolism and Disposition January 2009, 37 (1) 211-220; DOI: https://doi.org/10.1124/dmd.108.022012
von Moltke, Lisa L.
- You have accessRole of NADPH-Cytochrome P450 Reductase and Cytochrome-b5/NADH-b5 Reductase in Variability of CYP3A Activity in Human Liver MicrosomesLu Gan, Lisa L. von Moltke, Lauren A. Trepanier, Jerold S. Harmatz, David J. Greenblatt and Michael H. CourtDrug Metabolism and Disposition January 2009, 37 (1) 90-96; DOI: https://doi.org/10.1124/dmd.108.023424
W
Weaver, Yi Miao
- You have accessTissue Distribution, Gender-Divergent Expression, Ontogeny, and Chemical Induction of Multidrug Resistance Transporter Genes (Mdr1a, Mdr1b, Mdr2) in MiceYue Julia Cui, Xingguo Cheng, Yi Miao Weaver and Curtis D. KlaassenDrug Metabolism and Disposition January 2009, 37 (1) 203-210; DOI: https://doi.org/10.1124/dmd.108.023721
Wong, Pancras C.
- You have accessApixaban Metabolism and Pharmacokinetics after Oral Administration to HumansNirmala Raghavan, Charles E. Frost, Zhigang Yu, Kan He, Haiying Zhang, W. Griffith Humphreys, Donald Pinto, Shiangyuan Chen, Samuel Bonacorsi, Pancras C. Wong and Donglu ZhangDrug Metabolism and Disposition January 2009, 37 (1) 74-81; DOI: https://doi.org/10.1124/dmd.108.023143
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Yamanaka, Hiroyuki
- You have accessKey Amino Acid Residues Responsible for the Differences in Substrate Specificity of Human UDP-Glucuronosyltransferase (UGT)1A9 and UGT1A8Ryoichi Fujiwara, Miki Nakajima, Hiroyuki Yamanaka and Tsuyoshi YokoiDrug Metabolism and Disposition January 2009, 37 (1) 41-46; DOI: https://doi.org/10.1124/dmd.108.022913
Yamazaki, Hiroshi
- You have accessDrug Interactions of Thalidomide with Midazolam and Cyclosporine A: Heterotropic Cooperativity of Human Cytochrome P450 3A5Yusuke Okada, Norie Murayama, Chihiro Yanagida, Makiko Shimizu, F. Peter Guengerich and Hiroshi YamazakiDrug Metabolism and Disposition January 2009, 37 (1) 18-23; DOI: https://doi.org/10.1124/dmd.108.024679
Yamazoe, Yasushi
- You have accessRole of Enzymatic N-Hydroxylation and Reduction in Flutamide Metabolite-Induced Liver ToxicityMasato Ohbuchi, Masaaki Miyata, Daichi Nagai, Miki Shimada, Kouichi Yoshinari and Yasushi YamazoeDrug Metabolism and Disposition January 2009, 37 (1) 97-105; DOI: https://doi.org/10.1124/dmd.108.021964
Yanagida, Chihiro
- You have accessDrug Interactions of Thalidomide with Midazolam and Cyclosporine A: Heterotropic Cooperativity of Human Cytochrome P450 3A5Yusuke Okada, Norie Murayama, Chihiro Yanagida, Makiko Shimizu, F. Peter Guengerich and Hiroshi YamazakiDrug Metabolism and Disposition January 2009, 37 (1) 18-23; DOI: https://doi.org/10.1124/dmd.108.024679
Yeager, Ronnie L.
- You have accessCircadian Expression Profiles of Drug-Processing Genes and Transcription Factors in Mouse LiverYu-Kun Jennifer Zhang, Ronnie L. Yeager and Curtis D. KlaassenDrug Metabolism and Disposition January 2009, 37 (1) 106-115; DOI: https://doi.org/10.1124/dmd.108.024174
Yokoi, Tsuyoshi
- You have accessKey Amino Acid Residues Responsible for the Differences in Substrate Specificity of Human UDP-Glucuronosyltransferase (UGT)1A9 and UGT1A8Ryoichi Fujiwara, Miki Nakajima, Hiroyuki Yamanaka and Tsuyoshi YokoiDrug Metabolism and Disposition January 2009, 37 (1) 41-46; DOI: https://doi.org/10.1124/dmd.108.022913
Yoshikawa, Takahiro
- You have accessEffect of Oral Ketoconazole on Oral and Intravenous Pharmacokinetics of Simvastatin and Its Acid in Cynomolgus MonkeysAkihito Ogasawara, Masahiro Utoh, Kazuo Nii, Ayumi Ueda, Takahiro Yoshikawa, Toshiyuki Kume and Koichiro FukuzakiDrug Metabolism and Disposition January 2009, 37 (1) 122-128; DOI: https://doi.org/10.1124/dmd.108.022574
Yoshinari, Kouichi
- You have accessRole of Enzymatic N-Hydroxylation and Reduction in Flutamide Metabolite-Induced Liver ToxicityMasato Ohbuchi, Masaaki Miyata, Daichi Nagai, Miki Shimada, Kouichi Yoshinari and Yasushi YamazoeDrug Metabolism and Disposition January 2009, 37 (1) 97-105; DOI: https://doi.org/10.1124/dmd.108.021964
Yu, Ai-Ming
- You have accessQuantitation of Human Cytochrome P450 2D6 Protein with Immunoblot and Mass Spectrometry AnalysisAi-Ming Yu, Jun Qu, Melanie A. Felmlee, Jin Cao and Xi-Ling JiangDrug Metabolism and Disposition January 2009, 37 (1) 170-177; DOI: https://doi.org/10.1124/dmd.108.024166
- You have accessExpression and Functional Analysis of CYP2D6.24, CYP2D6.26, CYP2D6.27, and CYP2D7 IsozymesWei-Yan Zhang, You-Bin Tu, Robert L. Haining and Ai-Ming YuDrug Metabolism and Disposition January 2009, 37 (1) 1-4; DOI: https://doi.org/10.1124/dmd.108.023663
Yu, Zhigang
- You have accessApixaban Metabolism and Pharmacokinetics after Oral Administration to HumansNirmala Raghavan, Charles E. Frost, Zhigang Yu, Kan He, Haiying Zhang, W. Griffith Humphreys, Donald Pinto, Shiangyuan Chen, Samuel Bonacorsi, Pancras C. Wong and Donglu ZhangDrug Metabolism and Disposition January 2009, 37 (1) 74-81; DOI: https://doi.org/10.1124/dmd.108.023143
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Zhang, Donglu
- You have accessApixaban Metabolism and Pharmacokinetics after Oral Administration to HumansNirmala Raghavan, Charles E. Frost, Zhigang Yu, Kan He, Haiying Zhang, W. Griffith Humphreys, Donald Pinto, Shiangyuan Chen, Samuel Bonacorsi, Pancras C. Wong and Donglu ZhangDrug Metabolism and Disposition January 2009, 37 (1) 74-81; DOI: https://doi.org/10.1124/dmd.108.023143
Zhang, Haiying
- You have accessApixaban Metabolism and Pharmacokinetics after Oral Administration to HumansNirmala Raghavan, Charles E. Frost, Zhigang Yu, Kan He, Haiying Zhang, W. Griffith Humphreys, Donald Pinto, Shiangyuan Chen, Samuel Bonacorsi, Pancras C. Wong and Donglu ZhangDrug Metabolism and Disposition January 2009, 37 (1) 74-81; DOI: https://doi.org/10.1124/dmd.108.023143
Zhang, Wei-Yan
- You have accessExpression and Functional Analysis of CYP2D6.24, CYP2D6.26, CYP2D6.27, and CYP2D7 IsozymesWei-Yan Zhang, You-Bin Tu, Robert L. Haining and Ai-Ming YuDrug Metabolism and Disposition January 2009, 37 (1) 1-4; DOI: https://doi.org/10.1124/dmd.108.023663
Zhang, Xin
- You have accessPrediction of the Effect of Erythromycin, Diltiazem, and Their Metabolites, Alone and in Combination, on CYP3A4 InhibitionXin Zhang, David R. Jones and Stephen D. HallDrug Metabolism and Disposition January 2009, 37 (1) 150-160; DOI: https://doi.org/10.1124/dmd.108.022178
Zhang, Yiqun
- You have accessAbsolute Difference of Hepatobiliary Transporter Multidrug Resistance-Associated Protein (MRP2/Mrp2) in Liver Tissues and Isolated Hepatocytes from Rat, Dog, Monkey, and HumanNa Li, Yiqun Zhang, Fengmei Hua and Yurong LaiDrug Metabolism and Disposition January 2009, 37 (1) 66-73; DOI: https://doi.org/10.1124/dmd.108.023234
Zhang, Yu-Kun Jennifer
- You have accessCircadian Expression Profiles of Drug-Processing Genes and Transcription Factors in Mouse LiverYu-Kun Jennifer Zhang, Ronnie L. Yeager and Curtis D. KlaassenDrug Metabolism and Disposition January 2009, 37 (1) 106-115; DOI: https://doi.org/10.1124/dmd.108.024174
Zhong, Xiao-bo
- You have accessThree Patterns of Cytochrome P450 Gene Expression during Liver Maturation in MiceSteven N. Hart, Yue Cui, Curtis D. Klaassen and Xiao-bo ZhongDrug Metabolism and Disposition January 2009, 37 (1) 116-121; DOI: https://doi.org/10.1124/dmd.108.023812
Zientek, Michael
- You have accessMechanism-Based Inactivation of Cytochrome P450 2C9 by Tienilic Acid and (±)-Suprofen: A Comparison of Kinetics and Probe Substrate SelectionJ. Matthew Hutzler, Larissa M. Balogh, Michael Zientek, Vikas Kumar and Timothy S. TracyDrug Metabolism and Disposition January 2009, 37 (1) 59-65; DOI: https://doi.org/10.1124/dmd.108.023358
Zimmerman, Cheryl L.
- You have accessTransepithelial Transport of the Group II Metabotropic Glutamate 2/3 Receptor Agonist (1S,2S,5R,6S)-2-Aminobicyclo[3.1.0]hexane-2,6-dicarboxylate (LY354740) and Its Prodrug (1S,2S,5R,6S)-2-[(2′S)-(2′-Amino)propionyl]aminobicyclo[3.1.0]hexane-2,6-dicarboxylate (LY544344)Manthena V. S. Varma, André H. Eriksson, Geri Sawada, Youngeen A. Pak, Everett J. Perkins and Cheryl L. ZimmermanDrug Metabolism and Disposition January 2009, 37 (1) 211-220; DOI: https://doi.org/10.1124/dmd.108.022012
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