Research ArticleSpecial Section on Prediction of Human Pharmacokinetic Parameters from In Vitro Systems
In Vitro P-glycoprotein Efflux Ratio Can Predict the In Vivo Brain Penetration Regardless of Biopharmaceutics Drug Disposition Classification System Class
Ryota Kikuchi, Sonia M. de Morais and J. Cory Kalvass
Drug Metabolism and Disposition December 2013, 41 (12) 2012-2017; DOI: https://doi.org/10.1124/dmd.113.053868