Research ArticleArticle
Metabolism-Dependent Inhibition of CYP3A4 by Lapatinib: Evidence for Formation of a Metabolic Intermediate Complex with a Nitroso/Oxime Metabolite Formed via a Nitrone Intermediate
Joanna E. Barbara, Faraz Kazmi, Andrew Parkinson and David B. Buckley
Drug Metabolism and Disposition May 2013, 41 (5) 1012-1022; DOI: https://doi.org/10.1124/dmd.113.051151