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Validation of uPA/SCID Mouse with Humanized Liver as a Human Liver Model: Protein Quantification of Transporters, Cytochromes P450, and UDP-Glucuronosyltransferases by LC-MS/MS
Sumio Ohtsuki, Hirotaka Kawakami, Tae Inoue, Kenji Nakamura, Chise Tateno, Yuki Katsukura, Wataru Obuchi, Yasuo Uchida, Junichi Kamiie, Toru Horie and Tetsuya Terasaki
Drug Metabolism and Disposition June 2014, 42 (6) 1039-1043; DOI: https://doi.org/10.1124/dmd.114.057646
Sumio Ohtsuki
Department of Pharmaceutical Microbiology, Faculty of Life Sciences, Kumamoto University, Kumamoto, Japan (S.O., K.N.); Laboratory of Veterinary Pathology, School of Veterinary Medicine, Azabu University, Kanagawa, Japan (H.K., J.K.); Division of Membrane Transport and Drug Targeting, Graduate School of Pharmaceutical Sciences, Tohoku University, Sendai, Japan (T.I, Y.K., W.O., Y.U., T.T.); PhoenixBio, Co., Ltd., Hiroshima, Japan (C.T.); DeThree Research Laboratory Inc., Ibaraki, Japan (T.H.)
Hirotaka Kawakami
Department of Pharmaceutical Microbiology, Faculty of Life Sciences, Kumamoto University, Kumamoto, Japan (S.O., K.N.); Laboratory of Veterinary Pathology, School of Veterinary Medicine, Azabu University, Kanagawa, Japan (H.K., J.K.); Division of Membrane Transport and Drug Targeting, Graduate School of Pharmaceutical Sciences, Tohoku University, Sendai, Japan (T.I, Y.K., W.O., Y.U., T.T.); PhoenixBio, Co., Ltd., Hiroshima, Japan (C.T.); DeThree Research Laboratory Inc., Ibaraki, Japan (T.H.)
Tae Inoue
Department of Pharmaceutical Microbiology, Faculty of Life Sciences, Kumamoto University, Kumamoto, Japan (S.O., K.N.); Laboratory of Veterinary Pathology, School of Veterinary Medicine, Azabu University, Kanagawa, Japan (H.K., J.K.); Division of Membrane Transport and Drug Targeting, Graduate School of Pharmaceutical Sciences, Tohoku University, Sendai, Japan (T.I, Y.K., W.O., Y.U., T.T.); PhoenixBio, Co., Ltd., Hiroshima, Japan (C.T.); DeThree Research Laboratory Inc., Ibaraki, Japan (T.H.)
Kenji Nakamura
Department of Pharmaceutical Microbiology, Faculty of Life Sciences, Kumamoto University, Kumamoto, Japan (S.O., K.N.); Laboratory of Veterinary Pathology, School of Veterinary Medicine, Azabu University, Kanagawa, Japan (H.K., J.K.); Division of Membrane Transport and Drug Targeting, Graduate School of Pharmaceutical Sciences, Tohoku University, Sendai, Japan (T.I, Y.K., W.O., Y.U., T.T.); PhoenixBio, Co., Ltd., Hiroshima, Japan (C.T.); DeThree Research Laboratory Inc., Ibaraki, Japan (T.H.)
Chise Tateno
Department of Pharmaceutical Microbiology, Faculty of Life Sciences, Kumamoto University, Kumamoto, Japan (S.O., K.N.); Laboratory of Veterinary Pathology, School of Veterinary Medicine, Azabu University, Kanagawa, Japan (H.K., J.K.); Division of Membrane Transport and Drug Targeting, Graduate School of Pharmaceutical Sciences, Tohoku University, Sendai, Japan (T.I, Y.K., W.O., Y.U., T.T.); PhoenixBio, Co., Ltd., Hiroshima, Japan (C.T.); DeThree Research Laboratory Inc., Ibaraki, Japan (T.H.)
Yuki Katsukura
Department of Pharmaceutical Microbiology, Faculty of Life Sciences, Kumamoto University, Kumamoto, Japan (S.O., K.N.); Laboratory of Veterinary Pathology, School of Veterinary Medicine, Azabu University, Kanagawa, Japan (H.K., J.K.); Division of Membrane Transport and Drug Targeting, Graduate School of Pharmaceutical Sciences, Tohoku University, Sendai, Japan (T.I, Y.K., W.O., Y.U., T.T.); PhoenixBio, Co., Ltd., Hiroshima, Japan (C.T.); DeThree Research Laboratory Inc., Ibaraki, Japan (T.H.)
Wataru Obuchi
Department of Pharmaceutical Microbiology, Faculty of Life Sciences, Kumamoto University, Kumamoto, Japan (S.O., K.N.); Laboratory of Veterinary Pathology, School of Veterinary Medicine, Azabu University, Kanagawa, Japan (H.K., J.K.); Division of Membrane Transport and Drug Targeting, Graduate School of Pharmaceutical Sciences, Tohoku University, Sendai, Japan (T.I, Y.K., W.O., Y.U., T.T.); PhoenixBio, Co., Ltd., Hiroshima, Japan (C.T.); DeThree Research Laboratory Inc., Ibaraki, Japan (T.H.)
Yasuo Uchida
Department of Pharmaceutical Microbiology, Faculty of Life Sciences, Kumamoto University, Kumamoto, Japan (S.O., K.N.); Laboratory of Veterinary Pathology, School of Veterinary Medicine, Azabu University, Kanagawa, Japan (H.K., J.K.); Division of Membrane Transport and Drug Targeting, Graduate School of Pharmaceutical Sciences, Tohoku University, Sendai, Japan (T.I, Y.K., W.O., Y.U., T.T.); PhoenixBio, Co., Ltd., Hiroshima, Japan (C.T.); DeThree Research Laboratory Inc., Ibaraki, Japan (T.H.)
Junichi Kamiie
Department of Pharmaceutical Microbiology, Faculty of Life Sciences, Kumamoto University, Kumamoto, Japan (S.O., K.N.); Laboratory of Veterinary Pathology, School of Veterinary Medicine, Azabu University, Kanagawa, Japan (H.K., J.K.); Division of Membrane Transport and Drug Targeting, Graduate School of Pharmaceutical Sciences, Tohoku University, Sendai, Japan (T.I, Y.K., W.O., Y.U., T.T.); PhoenixBio, Co., Ltd., Hiroshima, Japan (C.T.); DeThree Research Laboratory Inc., Ibaraki, Japan (T.H.)
Toru Horie
Department of Pharmaceutical Microbiology, Faculty of Life Sciences, Kumamoto University, Kumamoto, Japan (S.O., K.N.); Laboratory of Veterinary Pathology, School of Veterinary Medicine, Azabu University, Kanagawa, Japan (H.K., J.K.); Division of Membrane Transport and Drug Targeting, Graduate School of Pharmaceutical Sciences, Tohoku University, Sendai, Japan (T.I, Y.K., W.O., Y.U., T.T.); PhoenixBio, Co., Ltd., Hiroshima, Japan (C.T.); DeThree Research Laboratory Inc., Ibaraki, Japan (T.H.)
Tetsuya Terasaki
Department of Pharmaceutical Microbiology, Faculty of Life Sciences, Kumamoto University, Kumamoto, Japan (S.O., K.N.); Laboratory of Veterinary Pathology, School of Veterinary Medicine, Azabu University, Kanagawa, Japan (H.K., J.K.); Division of Membrane Transport and Drug Targeting, Graduate School of Pharmaceutical Sciences, Tohoku University, Sendai, Japan (T.I, Y.K., W.O., Y.U., T.T.); PhoenixBio, Co., Ltd., Hiroshima, Japan (C.T.); DeThree Research Laboratory Inc., Ibaraki, Japan (T.H.)
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Protein Levels of P450s, UGTs, and Transporters in PXB Mice
Sumio Ohtsuki, Hirotaka Kawakami, Tae Inoue, Kenji Nakamura, Chise Tateno, Yuki Katsukura, Wataru Obuchi, Yasuo Uchida, Junichi Kamiie, Toru Horie and Tetsuya Terasaki
Drug Metabolism and Disposition June 1, 2014, 42 (6) 1039-1043; DOI: https://doi.org/10.1124/dmd.114.057646
Rapid CommunicationShort Communication
Protein Levels of P450s, UGTs, and Transporters in PXB Mice
Sumio Ohtsuki, Hirotaka Kawakami, Tae Inoue, Kenji Nakamura, Chise Tateno, Yuki Katsukura, Wataru Obuchi, Yasuo Uchida, Junichi Kamiie, Toru Horie and Tetsuya Terasaki
Drug Metabolism and Disposition June 1, 2014, 42 (6) 1039-1043; DOI: https://doi.org/10.1124/dmd.114.057646
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