Index by author
May 01, 2018; Volume 46,Issue 5
A
Abe, Koji
- You have accessCurcumin as an In Vivo Selective Intestinal Breast Cancer Resistance Protein Inhibitor in Cynomolgus MonkeysTsuyoshi Karibe, Tomoki Imaoka, Koji Abe and Osamu AndoDrug Metabolism and Disposition May 2018, 46 (5) 667-679; DOI: https://doi.org/10.1124/dmd.117.078931
Ahituv, Nadav
- You have accessRare Variants in the ABCG2 Promoter Modulate In Vivo ActivityRachel J. Eclov, Mee J. Kim, Robin Smith, Nadav Ahituv and Deanna L. KroetzDrug Metabolism and Disposition May 2018, 46 (5) 636-642; DOI: https://doi.org/10.1124/dmd.117.079541
Al-Judaibi, Bandar
- You have accessApixaban and Rosuvastatin Pharmacokinetics in Nonalcoholic Fatty Liver DiseaseRommel G. Tirona, Zahra Kassam, Ruth Strapp, Mala Ramu, Catherine Zhu, Melissa Liu, Ute I. Schwarz, Richard B. Kim, Bandar Al-Judaibi and Melanie D. BeatonDrug Metabolism and Disposition May 2018, 46 (5) 485-492; DOI: https://doi.org/10.1124/dmd.117.079624
Aleksunes, Lauren M.
- You have accessInterindividual Regulation of the Breast Cancer Resistance Protein/ABCG2 Transporter in Term Human PlacentasKristin M. Bircsak, Jamie E. Moscovitz, Xia Wen, Faith Archer, Poi Yu Sofia Yuen, Moiz Mohammed, Naureen Memon, Barry I. Weinberger, Laura M. Saba, Anna M. Vetrano and Lauren M. AleksunesDrug Metabolism and Disposition May 2018, 46 (5) 619-627; DOI: https://doi.org/10.1124/dmd.117.079228
Allain, Eric P.
- You have accessPost-transcriptional Regulation of UGT2B10 Hepatic Expression and Activity by Alternative SplicingAdrien Labriet, Eric P. Allain, Michèle Rouleau, Yannick Audet-Delage, Lyne Villeneuve and Chantal GuillemetteDrug Metabolism and Disposition May 2018, 46 (5) 514-524; DOI: https://doi.org/10.1124/dmd.117.079921
Ando, Osamu
- You have accessCurcumin as an In Vivo Selective Intestinal Breast Cancer Resistance Protein Inhibitor in Cynomolgus MonkeysTsuyoshi Karibe, Tomoki Imaoka, Koji Abe and Osamu AndoDrug Metabolism and Disposition May 2018, 46 (5) 667-679; DOI: https://doi.org/10.1124/dmd.117.078931
Annaert, Pieter
- You have accessMRP2 Inhibition by HIV Protease Inhibitors in Rat and Human Hepatocytes: A Quantitative Confocal Microscopy StudyNico Holmstock, Marlies Oorts, Jan Snoeys and Pieter AnnaertDrug Metabolism and Disposition May 2018, 46 (5) 697-703; DOI: https://doi.org/10.1124/dmd.117.079467
Archer, Faith
- You have accessInterindividual Regulation of the Breast Cancer Resistance Protein/ABCG2 Transporter in Term Human PlacentasKristin M. Bircsak, Jamie E. Moscovitz, Xia Wen, Faith Archer, Poi Yu Sofia Yuen, Moiz Mohammed, Naureen Memon, Barry I. Weinberger, Laura M. Saba, Anna M. Vetrano and Lauren M. AleksunesDrug Metabolism and Disposition May 2018, 46 (5) 619-627; DOI: https://doi.org/10.1124/dmd.117.079228
Audet-Delage, Yannick
- You have accessPost-transcriptional Regulation of UGT2B10 Hepatic Expression and Activity by Alternative SplicingAdrien Labriet, Eric P. Allain, Michèle Rouleau, Yannick Audet-Delage, Lyne Villeneuve and Chantal GuillemetteDrug Metabolism and Disposition May 2018, 46 (5) 514-524; DOI: https://doi.org/10.1124/dmd.117.079921
B
Beaton, Melanie D.
- You have accessApixaban and Rosuvastatin Pharmacokinetics in Nonalcoholic Fatty Liver DiseaseRommel G. Tirona, Zahra Kassam, Ruth Strapp, Mala Ramu, Catherine Zhu, Melissa Liu, Ute I. Schwarz, Richard B. Kim, Bandar Al-Judaibi and Melanie D. BeatonDrug Metabolism and Disposition May 2018, 46 (5) 485-492; DOI: https://doi.org/10.1124/dmd.117.079624
Bircsak, Kristin M.
- You have accessInterindividual Regulation of the Breast Cancer Resistance Protein/ABCG2 Transporter in Term Human PlacentasKristin M. Bircsak, Jamie E. Moscovitz, Xia Wen, Faith Archer, Poi Yu Sofia Yuen, Moiz Mohammed, Naureen Memon, Barry I. Weinberger, Laura M. Saba, Anna M. Vetrano and Lauren M. AleksunesDrug Metabolism and Disposition May 2018, 46 (5) 619-627; DOI: https://doi.org/10.1124/dmd.117.079228
Bourbonais, Francis
- You have accessComparison of Proteomic Quantification Approaches for Hepatic Drug Transporters: Multiplexed Global Quantitation Correlates with Targeted Proteomic QuantitationAnna Vildhede, Chuong Nguyen, Brian K. Erickson, Ryan C. Kunz, Richard Jones, Emi Kimoto, Francis Bourbonais, A. David Rodrigues and Manthena V.S. VarmaDrug Metabolism and Disposition May 2018, 46 (5) 692-696; DOI: https://doi.org/10.1124/dmd.117.079285
C
Cai, Qingyun
- You have accessA Promising Microtubule Inhibitor Deoxypodophyllotoxin Exhibits Better Efficacy to Multidrug-Resistant Breast Cancer than Paclitaxel via Avoiding Efflux TransportXiaojie Zang, Guangji Wang, Qingyun Cai, Xiao Zheng, Jingwei Zhang, Qianying Chen, Baojin Wu, Xiong Zhu, Haiping Hao and Fang ZhouDrug Metabolism and Disposition May 2018, 46 (5) 542-551; DOI: https://doi.org/10.1124/dmd.117.079442
Cech, Nadja B.
- You have accessIdentification of Intestinal UDP-Glucuronosyltransferase Inhibitors in Green Tea (Camellia sinensis) Using a Biochemometric Approach: Application to Raloxifene as a Test Drug via In Vitro to In Vivo ExtrapolationDan-Dan Tian, Joshua J. Kellogg, Neşe Okut, Nicholas H. Oberlies, Nadja B. Cech, Danny D. Shen, Jeannine S. McCune and Mary F. PaineDrug Metabolism and Disposition May 2018, 46 (5) 552-560; DOI: https://doi.org/10.1124/dmd.117.079491
Chen, Kaiwen
- You have accessIdentification of a NFκB Inhibition Site on the Proximal Promoter Region of Human Organic Anion Transporting Polypeptide 1A2 Coding Gene SLCO1A2Zhaojian Xiang, Weike Li, Lixue Wang, Jicai Yi, Kaiwen Chen and Mei HongDrug Metabolism and Disposition May 2018, 46 (5) 643-651; DOI: https://doi.org/10.1124/dmd.117.078832
Chen, Qianying
- You have accessA Promising Microtubule Inhibitor Deoxypodophyllotoxin Exhibits Better Efficacy to Multidrug-Resistant Breast Cancer than Paclitaxel via Avoiding Efflux TransportXiaojie Zang, Guangji Wang, Qingyun Cai, Xiao Zheng, Jingwei Zhang, Qianying Chen, Baojin Wu, Xiong Zhu, Haiping Hao and Fang ZhouDrug Metabolism and Disposition May 2018, 46 (5) 542-551; DOI: https://doi.org/10.1124/dmd.117.079442
Chen, Yuan
- You have accessIntravital Multiphoton Microscopy with Fluorescent Bile Salts in Rats as an In Vivo Biomarker for Hepatobiliary Transport InhibitionJennifer Ryan, Ryan E. Morgan, Yuan Chen, Laurie P. Volak, Robert T. Dunn and Kenneth W. DunnDrug Metabolism and Disposition May 2018, 46 (5) 704-718; DOI: https://doi.org/10.1124/dmd.117.079277
Cook-Rostie, Nicholas
- You have accessBrain Distribution of a Novel MEK Inhibitor E6201: Implications in the Treatment of Melanoma Brain MetastasesGautham Gampa, Minjee Kim, Nicholas Cook-Rostie, Janice K. Laramy, Jann N. Sarkaria, Linda Paradiso, Louis DePalatis and William F. ElmquistDrug Metabolism and Disposition May 2018, 46 (5) 658-666; DOI: https://doi.org/10.1124/dmd.117.079194
Crawford, Rebecca R.
- You have accessBeyond Competitive Inhibition: Regulation of ABC Transporters by Kinases and Protein-Protein Interactions as Potential Mechanisms of Drug-Drug InteractionsRebecca R. Crawford, Praveen K. Potukuchi, Erin G. Schuetz and John D. SchuetzDrug Metabolism and Disposition May 2018, 46 (5) 567-580; DOI: https://doi.org/10.1124/dmd.118.080663
Cui, Julia Yue
- You have accessPhysiological Regulation of Drug Metabolism and Transport: Pregnancy, Microbiome, Inflammation, Infection, and FastingEdward T. Morgan, Joseph L. Dempsey, Sylvie M. Mimche, Tracey J. Lamb, Supriya Kulkarni, Julia Yue Cui, Hyunyoung Jeong and Angela L. SlittDrug Metabolism and Disposition May 2018, 46 (5) 503-513; DOI: https://doi.org/10.1124/dmd.117.079905
Cui, Yilong
- Open AccessA Clinical Quantitative Evaluation of Hepatobiliary Transport of [11C]Dehydropravastatin in Humans Using Positron Emission TomographyKen-ichi Kaneko, Masaaki Tanaka, Akira Ishii, Yumiko Katayama, Takayoshi Nakaoka, Satsuki Irie, Hideki Kawahata, Takashi Yamanaga, Yasuhiro Wada, Takeshi Miyake, Kota Toshimoto, Kazuya Maeda, Yilong Cui, Masaru Enomoto, Etsushi Kawamura, Norifumi Kawada, Joji Kawabe, Susumu Shiomi, Hiroyuki Kusuhara, Yuichi Sugiyama and Yasuyoshi WatanabeDrug Metabolism and Disposition May 2018, 46 (5) 719-728; DOI: https://doi.org/10.1124/dmd.118.080408
D
Dabaghie, Dina
- Open AccessExpression of Organic Anion Transporter 1 or 3 in Human Kidney Proximal Tubule Cells Reduces Cisplatin SensitivityTom T. G. Nieskens, Janny G. P. Peters, Dina Dabaghie, Daphne Korte, Katja Jansen, Alexander H. Van Asbeck, Neslihan N. Tavraz, Thomas Friedrich, Frans G. M. Russel, Rosalinde Masereeuw and Martijn J. WilmerDrug Metabolism and Disposition May 2018, 46 (5) 592-599; DOI: https://doi.org/10.1124/dmd.117.079384
Dempsey, Joseph L.
- You have accessPhysiological Regulation of Drug Metabolism and Transport: Pregnancy, Microbiome, Inflammation, Infection, and FastingEdward T. Morgan, Joseph L. Dempsey, Sylvie M. Mimche, Tracey J. Lamb, Supriya Kulkarni, Julia Yue Cui, Hyunyoung Jeong and Angela L. SlittDrug Metabolism and Disposition May 2018, 46 (5) 503-513; DOI: https://doi.org/10.1124/dmd.117.079905
DePalatis, Louis
- You have accessBrain Distribution of a Novel MEK Inhibitor E6201: Implications in the Treatment of Melanoma Brain MetastasesGautham Gampa, Minjee Kim, Nicholas Cook-Rostie, Janice K. Laramy, Jann N. Sarkaria, Linda Paradiso, Louis DePalatis and William F. ElmquistDrug Metabolism and Disposition May 2018, 46 (5) 658-666; DOI: https://doi.org/10.1124/dmd.117.079194
Dunn, Kenneth W.
- You have accessIntravital Multiphoton Microscopy with Fluorescent Bile Salts in Rats as an In Vivo Biomarker for Hepatobiliary Transport InhibitionJennifer Ryan, Ryan E. Morgan, Yuan Chen, Laurie P. Volak, Robert T. Dunn and Kenneth W. DunnDrug Metabolism and Disposition May 2018, 46 (5) 704-718; DOI: https://doi.org/10.1124/dmd.117.079277
Dunn, Robert T.
- You have accessIntravital Multiphoton Microscopy with Fluorescent Bile Salts in Rats as an In Vivo Biomarker for Hepatobiliary Transport InhibitionJennifer Ryan, Ryan E. Morgan, Yuan Chen, Laurie P. Volak, Robert T. Dunn and Kenneth W. DunnDrug Metabolism and Disposition May 2018, 46 (5) 704-718; DOI: https://doi.org/10.1124/dmd.117.079277
E
Eclov, Rachel J.
- You have accessRare Variants in the ABCG2 Promoter Modulate In Vivo ActivityRachel J. Eclov, Mee J. Kim, Robin Smith, Nadav Ahituv and Deanna L. KroetzDrug Metabolism and Disposition May 2018, 46 (5) 636-642; DOI: https://doi.org/10.1124/dmd.117.079541
El-Kattan, Ayman F.
- You have accessNavigating Transporter Sciences in Pharmacokinetics Characterization Using the Extended Clearance Classification SystemAyman F. El-Kattan and Manthena V. S. VarmaDrug Metabolism and Disposition May 2018, 46 (5) 729-739; DOI: https://doi.org/10.1124/dmd.117.080044
Elmquist, William F.
- You have accessBrain Distribution of a Novel MEK Inhibitor E6201: Implications in the Treatment of Melanoma Brain MetastasesGautham Gampa, Minjee Kim, Nicholas Cook-Rostie, Janice K. Laramy, Jann N. Sarkaria, Linda Paradiso, Louis DePalatis and William F. ElmquistDrug Metabolism and Disposition May 2018, 46 (5) 658-666; DOI: https://doi.org/10.1124/dmd.117.079194
Enomoto, Masaru
- Open AccessA Clinical Quantitative Evaluation of Hepatobiliary Transport of [11C]Dehydropravastatin in Humans Using Positron Emission TomographyKen-ichi Kaneko, Masaaki Tanaka, Akira Ishii, Yumiko Katayama, Takayoshi Nakaoka, Satsuki Irie, Hideki Kawahata, Takashi Yamanaga, Yasuhiro Wada, Takeshi Miyake, Kota Toshimoto, Kazuya Maeda, Yilong Cui, Masaru Enomoto, Etsushi Kawamura, Norifumi Kawada, Joji Kawabe, Susumu Shiomi, Hiroyuki Kusuhara, Yuichi Sugiyama and Yasuyoshi WatanabeDrug Metabolism and Disposition May 2018, 46 (5) 719-728; DOI: https://doi.org/10.1124/dmd.118.080408
Erickson, Brian K.
- You have accessComparison of Proteomic Quantification Approaches for Hepatic Drug Transporters: Multiplexed Global Quantitation Correlates with Targeted Proteomic QuantitationAnna Vildhede, Chuong Nguyen, Brian K. Erickson, Ryan C. Kunz, Richard Jones, Emi Kimoto, Francis Bourbonais, A. David Rodrigues and Manthena V.S. VarmaDrug Metabolism and Disposition May 2018, 46 (5) 692-696; DOI: https://doi.org/10.1124/dmd.117.079285
F
Fate, Gwendolyn D.
- You have accessBiosynthesis and Identification of Metabolites of Maraviroc and Their Use in Experiments to Delineate the Relative Contributions of Cytochrome P4503A4 versus 3A5Elaine Tseng, Gwendolyn D. Fate, Gregory S. Walker, Theunis C. Goosen and R. Scott ObachDrug Metabolism and Disposition May 2018, 46 (5) 493-502; DOI: https://doi.org/10.1124/dmd.117.079855
Follman, Kristin E.
- You have accessPrediction of the Effects of Renal Impairment on Clearance for Organic Cation Drugs that Undergo Renal Secretion: A Simulation-Based StudyKristin E. Follman and Marilyn E. MorrisDrug Metabolism and Disposition May 2018, 46 (5) 758-769; DOI: https://doi.org/10.1124/dmd.117.079558
Friedrich, Thomas
- Open AccessExpression of Organic Anion Transporter 1 or 3 in Human Kidney Proximal Tubule Cells Reduces Cisplatin SensitivityTom T. G. Nieskens, Janny G. P. Peters, Dina Dabaghie, Daphne Korte, Katja Jansen, Alexander H. Van Asbeck, Neslihan N. Tavraz, Thomas Friedrich, Frans G. M. Russel, Rosalinde Masereeuw and Martijn J. WilmerDrug Metabolism and Disposition May 2018, 46 (5) 592-599; DOI: https://doi.org/10.1124/dmd.117.079384
Fukuchi, Yukina
- You have accessSandwich-Cultured Hepatocytes for Mechanistic Understanding of Hepatic Disposition of Parent Drugs and Metabolites by Transporter–Enzyme InterplayNorikazu Matsunaga, Yukina Fukuchi, Haruo Imawaka and Ikumi TamaiDrug Metabolism and Disposition May 2018, 46 (5) 680-691; DOI: https://doi.org/10.1124/dmd.117.079236
Futatsugi, Azusa
- You have accessEvaluation of Alteration in Hepatic and Intestinal BCRP Function In Vivo from ABCG2 c.421C>A Polymorphism Based on PBPK Analysis of RosuvastatinAzusa Futatsugi, Kota Toshimoto, Takashi Yoshikado, Yuichi Sugiyama and Yukio KatoDrug Metabolism and Disposition May 2018, 46 (5) 749-757; DOI: https://doi.org/10.1124/dmd.117.078816
G
Gampa, Gautham
- You have accessBrain Distribution of a Novel MEK Inhibitor E6201: Implications in the Treatment of Melanoma Brain MetastasesGautham Gampa, Minjee Kim, Nicholas Cook-Rostie, Janice K. Laramy, Jann N. Sarkaria, Linda Paradiso, Louis DePalatis and William F. ElmquistDrug Metabolism and Disposition May 2018, 46 (5) 658-666; DOI: https://doi.org/10.1124/dmd.117.079194
Gao, Chunying
- You have accessHepatic Transport of 25-Hydroxyvitamin D3 Conjugates: A Mechanism of 25-Hydroxyvitamin D3 Delivery to the Intestinal TractChunying Gao, Michael Z. Liao, Lyrialle W. Han, Kenneth E. Thummel and Qingcheng MaoDrug Metabolism and Disposition May 2018, 46 (5) 581-591; DOI: https://doi.org/10.1124/dmd.117.078881
Gillen, Michael
- You have accessMetabolism and Disposition of Verinurad, a Uric Acid Reabsorption Inhibitor, in HumansCaroline A. Lee, Chun Yang, Vishal Shah, Zancong Shen, David M. Wilson, Traci M. Ostertag, Jean-Luc Girardet, Jesse Hall and Michael GillenDrug Metabolism and Disposition May 2018, 46 (5) 532-541; DOI: https://doi.org/10.1124/dmd.117.078220
Girardet, Jean-Luc
- You have accessMetabolism and Disposition of Verinurad, a Uric Acid Reabsorption Inhibitor, in HumansCaroline A. Lee, Chun Yang, Vishal Shah, Zancong Shen, David M. Wilson, Traci M. Ostertag, Jean-Luc Girardet, Jesse Hall and Michael GillenDrug Metabolism and Disposition May 2018, 46 (5) 532-541; DOI: https://doi.org/10.1124/dmd.117.078220
Goosen, Theunis C.
- You have accessBiosynthesis and Identification of Metabolites of Maraviroc and Their Use in Experiments to Delineate the Relative Contributions of Cytochrome P4503A4 versus 3A5Elaine Tseng, Gwendolyn D. Fate, Gregory S. Walker, Theunis C. Goosen and R. Scott ObachDrug Metabolism and Disposition May 2018, 46 (5) 493-502; DOI: https://doi.org/10.1124/dmd.117.079855
Govindarajan, Rajgopal
- Open AccessIdentification of Structural and Molecular Features Involved in the Transport of 3′-Deoxy-Nucleoside Analogs by Human Equilibrative Nucleoside Transporter 3MD Fazlur Rahman, Radhika Raj and Rajgopal GovindarajanDrug Metabolism and Disposition May 2018, 46 (5) 600-609; DOI: https://doi.org/10.1124/dmd.117.079400
Guillemette, Chantal
- You have accessPost-transcriptional Regulation of UGT2B10 Hepatic Expression and Activity by Alternative SplicingAdrien Labriet, Eric P. Allain, Michèle Rouleau, Yannick Audet-Delage, Lyne Villeneuve and Chantal GuillemetteDrug Metabolism and Disposition May 2018, 46 (5) 514-524; DOI: https://doi.org/10.1124/dmd.117.079921
Guo, Dayong
- You have accessGeneration and Characterization of a CYP2C11-Null Rat Model by Using the CRISPR/Cas9 MethodYuan Wei, Li Yang, Xiaoyan Zhang, Danjuan Sui, Changsuo Wang, Kai Wang, Mangting Shan, Dayong Guo and Hongyu WangDrug Metabolism and Disposition May 2018, 46 (5) 525-531; DOI: https://doi.org/10.1124/dmd.117.078444
H
Hall, Jesse
- You have accessMetabolism and Disposition of Verinurad, a Uric Acid Reabsorption Inhibitor, in HumansCaroline A. Lee, Chun Yang, Vishal Shah, Zancong Shen, David M. Wilson, Traci M. Ostertag, Jean-Luc Girardet, Jesse Hall and Michael GillenDrug Metabolism and Disposition May 2018, 46 (5) 532-541; DOI: https://doi.org/10.1124/dmd.117.078220
Han, Lyrialle W.
- You have accessHepatic Transport of 25-Hydroxyvitamin D3 Conjugates: A Mechanism of 25-Hydroxyvitamin D3 Delivery to the Intestinal TractChunying Gao, Michael Z. Liao, Lyrialle W. Han, Kenneth E. Thummel and Qingcheng MaoDrug Metabolism and Disposition May 2018, 46 (5) 581-591; DOI: https://doi.org/10.1124/dmd.117.078881
Hao, Haiping
- You have accessA Promising Microtubule Inhibitor Deoxypodophyllotoxin Exhibits Better Efficacy to Multidrug-Resistant Breast Cancer than Paclitaxel via Avoiding Efflux TransportXiaojie Zang, Guangji Wang, Qingyun Cai, Xiao Zheng, Jingwei Zhang, Qianying Chen, Baojin Wu, Xiong Zhu, Haiping Hao and Fang ZhouDrug Metabolism and Disposition May 2018, 46 (5) 542-551; DOI: https://doi.org/10.1124/dmd.117.079442
Hirota, Takeshi
- You have accessInterindividual Differences in the Expression of ATP-Binding Cassette and Solute Carrier Family Transporters in Human Skin: DNA Methylation Regulates Transcriptional Activity of the Human ABCC3 GeneTomoki Takechi, Takeshi Hirota, Tatsuya Sakai, Natsumi Maeda, Daisuke Kobayashi and Ichiro IeiriDrug Metabolism and Disposition May 2018, 46 (5) 628-635; DOI: https://doi.org/10.1124/dmd.117.079061
Hisaka, Akihiro
- You have accessPhysiologically Based Pharmacokinetic Modeling of Bosentan Identifies the Saturable Hepatic Uptake As a Major Contributor to Its Nonlinear PharmacokineticsMasanobu Sato, Kota Toshimoto, Atsuko Tomaru, Takashi Yoshikado, Yuta Tanaka, Akihiro Hisaka, Wooin Lee and Yuichi SugiyamaDrug Metabolism and Disposition May 2018, 46 (5) 740-748; DOI: https://doi.org/10.1124/dmd.117.078972
Holmstock, Nico
- You have accessMRP2 Inhibition by HIV Protease Inhibitors in Rat and Human Hepatocytes: A Quantitative Confocal Microscopy StudyNico Holmstock, Marlies Oorts, Jan Snoeys and Pieter AnnaertDrug Metabolism and Disposition May 2018, 46 (5) 697-703; DOI: https://doi.org/10.1124/dmd.117.079467
Hong, Mei
- You have accessIdentification of a NFκB Inhibition Site on the Proximal Promoter Region of Human Organic Anion Transporting Polypeptide 1A2 Coding Gene SLCO1A2Zhaojian Xiang, Weike Li, Lixue Wang, Jicai Yi, Kaiwen Chen and Mei HongDrug Metabolism and Disposition May 2018, 46 (5) 643-651; DOI: https://doi.org/10.1124/dmd.117.078832
I
Ieiri, Ichiro
- You have accessInterindividual Differences in the Expression of ATP-Binding Cassette and Solute Carrier Family Transporters in Human Skin: DNA Methylation Regulates Transcriptional Activity of the Human ABCC3 GeneTomoki Takechi, Takeshi Hirota, Tatsuya Sakai, Natsumi Maeda, Daisuke Kobayashi and Ichiro IeiriDrug Metabolism and Disposition May 2018, 46 (5) 628-635; DOI: https://doi.org/10.1124/dmd.117.079061
Imaoka, Tomoki
- You have accessCurcumin as an In Vivo Selective Intestinal Breast Cancer Resistance Protein Inhibitor in Cynomolgus MonkeysTsuyoshi Karibe, Tomoki Imaoka, Koji Abe and Osamu AndoDrug Metabolism and Disposition May 2018, 46 (5) 667-679; DOI: https://doi.org/10.1124/dmd.117.078931
Imawaka, Haruo
- You have accessSandwich-Cultured Hepatocytes for Mechanistic Understanding of Hepatic Disposition of Parent Drugs and Metabolites by Transporter–Enzyme InterplayNorikazu Matsunaga, Yukina Fukuchi, Haruo Imawaka and Ikumi TamaiDrug Metabolism and Disposition May 2018, 46 (5) 680-691; DOI: https://doi.org/10.1124/dmd.117.079236
Irie, Satsuki
- Open AccessA Clinical Quantitative Evaluation of Hepatobiliary Transport of [11C]Dehydropravastatin in Humans Using Positron Emission TomographyKen-ichi Kaneko, Masaaki Tanaka, Akira Ishii, Yumiko Katayama, Takayoshi Nakaoka, Satsuki Irie, Hideki Kawahata, Takashi Yamanaga, Yasuhiro Wada, Takeshi Miyake, Kota Toshimoto, Kazuya Maeda, Yilong Cui, Masaru Enomoto, Etsushi Kawamura, Norifumi Kawada, Joji Kawabe, Susumu Shiomi, Hiroyuki Kusuhara, Yuichi Sugiyama and Yasuyoshi WatanabeDrug Metabolism and Disposition May 2018, 46 (5) 719-728; DOI: https://doi.org/10.1124/dmd.118.080408
Ishii, Akira
- Open AccessA Clinical Quantitative Evaluation of Hepatobiliary Transport of [11C]Dehydropravastatin in Humans Using Positron Emission TomographyKen-ichi Kaneko, Masaaki Tanaka, Akira Ishii, Yumiko Katayama, Takayoshi Nakaoka, Satsuki Irie, Hideki Kawahata, Takashi Yamanaga, Yasuhiro Wada, Takeshi Miyake, Kota Toshimoto, Kazuya Maeda, Yilong Cui, Masaru Enomoto, Etsushi Kawamura, Norifumi Kawada, Joji Kawabe, Susumu Shiomi, Hiroyuki Kusuhara, Yuichi Sugiyama and Yasuyoshi WatanabeDrug Metabolism and Disposition May 2018, 46 (5) 719-728; DOI: https://doi.org/10.1124/dmd.118.080408
J
Jansen, Katja
- Open AccessExpression of Organic Anion Transporter 1 or 3 in Human Kidney Proximal Tubule Cells Reduces Cisplatin SensitivityTom T. G. Nieskens, Janny G. P. Peters, Dina Dabaghie, Daphne Korte, Katja Jansen, Alexander H. Van Asbeck, Neslihan N. Tavraz, Thomas Friedrich, Frans G. M. Russel, Rosalinde Masereeuw and Martijn J. WilmerDrug Metabolism and Disposition May 2018, 46 (5) 592-599; DOI: https://doi.org/10.1124/dmd.117.079384
Jeong, Hyunyoung
- You have accessPhysiological Regulation of Drug Metabolism and Transport: Pregnancy, Microbiome, Inflammation, Infection, and FastingEdward T. Morgan, Joseph L. Dempsey, Sylvie M. Mimche, Tracey J. Lamb, Supriya Kulkarni, Julia Yue Cui, Hyunyoung Jeong and Angela L. SlittDrug Metabolism and Disposition May 2018, 46 (5) 503-513; DOI: https://doi.org/10.1124/dmd.117.079905
Jones, Richard
- You have accessComparison of Proteomic Quantification Approaches for Hepatic Drug Transporters: Multiplexed Global Quantitation Correlates with Targeted Proteomic QuantitationAnna Vildhede, Chuong Nguyen, Brian K. Erickson, Ryan C. Kunz, Richard Jones, Emi Kimoto, Francis Bourbonais, A. David Rodrigues and Manthena V.S. VarmaDrug Metabolism and Disposition May 2018, 46 (5) 692-696; DOI: https://doi.org/10.1124/dmd.117.079285
K
Kaneko, Ken-ichi
- Open AccessA Clinical Quantitative Evaluation of Hepatobiliary Transport of [11C]Dehydropravastatin in Humans Using Positron Emission TomographyKen-ichi Kaneko, Masaaki Tanaka, Akira Ishii, Yumiko Katayama, Takayoshi Nakaoka, Satsuki Irie, Hideki Kawahata, Takashi Yamanaga, Yasuhiro Wada, Takeshi Miyake, Kota Toshimoto, Kazuya Maeda, Yilong Cui, Masaru Enomoto, Etsushi Kawamura, Norifumi Kawada, Joji Kawabe, Susumu Shiomi, Hiroyuki Kusuhara, Yuichi Sugiyama and Yasuyoshi WatanabeDrug Metabolism and Disposition May 2018, 46 (5) 719-728; DOI: https://doi.org/10.1124/dmd.118.080408
Karibe, Tsuyoshi
- You have accessCurcumin as an In Vivo Selective Intestinal Breast Cancer Resistance Protein Inhibitor in Cynomolgus MonkeysTsuyoshi Karibe, Tomoki Imaoka, Koji Abe and Osamu AndoDrug Metabolism and Disposition May 2018, 46 (5) 667-679; DOI: https://doi.org/10.1124/dmd.117.078931
Kassam, Zahra
- You have accessApixaban and Rosuvastatin Pharmacokinetics in Nonalcoholic Fatty Liver DiseaseRommel G. Tirona, Zahra Kassam, Ruth Strapp, Mala Ramu, Catherine Zhu, Melissa Liu, Ute I. Schwarz, Richard B. Kim, Bandar Al-Judaibi and Melanie D. BeatonDrug Metabolism and Disposition May 2018, 46 (5) 485-492; DOI: https://doi.org/10.1124/dmd.117.079624
Katayama, Yumiko
- Open AccessA Clinical Quantitative Evaluation of Hepatobiliary Transport of [11C]Dehydropravastatin in Humans Using Positron Emission TomographyKen-ichi Kaneko, Masaaki Tanaka, Akira Ishii, Yumiko Katayama, Takayoshi Nakaoka, Satsuki Irie, Hideki Kawahata, Takashi Yamanaga, Yasuhiro Wada, Takeshi Miyake, Kota Toshimoto, Kazuya Maeda, Yilong Cui, Masaru Enomoto, Etsushi Kawamura, Norifumi Kawada, Joji Kawabe, Susumu Shiomi, Hiroyuki Kusuhara, Yuichi Sugiyama and Yasuyoshi WatanabeDrug Metabolism and Disposition May 2018, 46 (5) 719-728; DOI: https://doi.org/10.1124/dmd.118.080408
Kato, Yukio
- You have accessEvaluation of Alteration in Hepatic and Intestinal BCRP Function In Vivo from ABCG2 c.421C>A Polymorphism Based on PBPK Analysis of RosuvastatinAzusa Futatsugi, Kota Toshimoto, Takashi Yoshikado, Yuichi Sugiyama and Yukio KatoDrug Metabolism and Disposition May 2018, 46 (5) 749-757; DOI: https://doi.org/10.1124/dmd.117.078816
Kawabe, Joji
- Open AccessA Clinical Quantitative Evaluation of Hepatobiliary Transport of [11C]Dehydropravastatin in Humans Using Positron Emission TomographyKen-ichi Kaneko, Masaaki Tanaka, Akira Ishii, Yumiko Katayama, Takayoshi Nakaoka, Satsuki Irie, Hideki Kawahata, Takashi Yamanaga, Yasuhiro Wada, Takeshi Miyake, Kota Toshimoto, Kazuya Maeda, Yilong Cui, Masaru Enomoto, Etsushi Kawamura, Norifumi Kawada, Joji Kawabe, Susumu Shiomi, Hiroyuki Kusuhara, Yuichi Sugiyama and Yasuyoshi WatanabeDrug Metabolism and Disposition May 2018, 46 (5) 719-728; DOI: https://doi.org/10.1124/dmd.118.080408
Kawada, Norifumi
- Open AccessA Clinical Quantitative Evaluation of Hepatobiliary Transport of [11C]Dehydropravastatin in Humans Using Positron Emission TomographyKen-ichi Kaneko, Masaaki Tanaka, Akira Ishii, Yumiko Katayama, Takayoshi Nakaoka, Satsuki Irie, Hideki Kawahata, Takashi Yamanaga, Yasuhiro Wada, Takeshi Miyake, Kota Toshimoto, Kazuya Maeda, Yilong Cui, Masaru Enomoto, Etsushi Kawamura, Norifumi Kawada, Joji Kawabe, Susumu Shiomi, Hiroyuki Kusuhara, Yuichi Sugiyama and Yasuyoshi WatanabeDrug Metabolism and Disposition May 2018, 46 (5) 719-728; DOI: https://doi.org/10.1124/dmd.118.080408
Kawahata, Hideki
- Open AccessA Clinical Quantitative Evaluation of Hepatobiliary Transport of [11C]Dehydropravastatin in Humans Using Positron Emission TomographyKen-ichi Kaneko, Masaaki Tanaka, Akira Ishii, Yumiko Katayama, Takayoshi Nakaoka, Satsuki Irie, Hideki Kawahata, Takashi Yamanaga, Yasuhiro Wada, Takeshi Miyake, Kota Toshimoto, Kazuya Maeda, Yilong Cui, Masaru Enomoto, Etsushi Kawamura, Norifumi Kawada, Joji Kawabe, Susumu Shiomi, Hiroyuki Kusuhara, Yuichi Sugiyama and Yasuyoshi WatanabeDrug Metabolism and Disposition May 2018, 46 (5) 719-728; DOI: https://doi.org/10.1124/dmd.118.080408
Kawamura, Etsushi
- Open AccessA Clinical Quantitative Evaluation of Hepatobiliary Transport of [11C]Dehydropravastatin in Humans Using Positron Emission TomographyKen-ichi Kaneko, Masaaki Tanaka, Akira Ishii, Yumiko Katayama, Takayoshi Nakaoka, Satsuki Irie, Hideki Kawahata, Takashi Yamanaga, Yasuhiro Wada, Takeshi Miyake, Kota Toshimoto, Kazuya Maeda, Yilong Cui, Masaru Enomoto, Etsushi Kawamura, Norifumi Kawada, Joji Kawabe, Susumu Shiomi, Hiroyuki Kusuhara, Yuichi Sugiyama and Yasuyoshi WatanabeDrug Metabolism and Disposition May 2018, 46 (5) 719-728; DOI: https://doi.org/10.1124/dmd.118.080408
Kellogg, Joshua J.
- You have accessIdentification of Intestinal UDP-Glucuronosyltransferase Inhibitors in Green Tea (Camellia sinensis) Using a Biochemometric Approach: Application to Raloxifene as a Test Drug via In Vitro to In Vivo ExtrapolationDan-Dan Tian, Joshua J. Kellogg, Neşe Okut, Nicholas H. Oberlies, Nadja B. Cech, Danny D. Shen, Jeannine S. McCune and Mary F. PaineDrug Metabolism and Disposition May 2018, 46 (5) 552-560; DOI: https://doi.org/10.1124/dmd.117.079491
Kim, Mee J.
- You have accessRare Variants in the ABCG2 Promoter Modulate In Vivo ActivityRachel J. Eclov, Mee J. Kim, Robin Smith, Nadav Ahituv and Deanna L. KroetzDrug Metabolism and Disposition May 2018, 46 (5) 636-642; DOI: https://doi.org/10.1124/dmd.117.079541
Kim, Minjee
- You have accessBrain Distribution of a Novel MEK Inhibitor E6201: Implications in the Treatment of Melanoma Brain MetastasesGautham Gampa, Minjee Kim, Nicholas Cook-Rostie, Janice K. Laramy, Jann N. Sarkaria, Linda Paradiso, Louis DePalatis and William F. ElmquistDrug Metabolism and Disposition May 2018, 46 (5) 658-666; DOI: https://doi.org/10.1124/dmd.117.079194
Kim, Richard B.
- You have accessApixaban and Rosuvastatin Pharmacokinetics in Nonalcoholic Fatty Liver DiseaseRommel G. Tirona, Zahra Kassam, Ruth Strapp, Mala Ramu, Catherine Zhu, Melissa Liu, Ute I. Schwarz, Richard B. Kim, Bandar Al-Judaibi and Melanie D. BeatonDrug Metabolism and Disposition May 2018, 46 (5) 485-492; DOI: https://doi.org/10.1124/dmd.117.079624
Kimoto, Emi
- You have accessComparison of Proteomic Quantification Approaches for Hepatic Drug Transporters: Multiplexed Global Quantitation Correlates with Targeted Proteomic QuantitationAnna Vildhede, Chuong Nguyen, Brian K. Erickson, Ryan C. Kunz, Richard Jones, Emi Kimoto, Francis Bourbonais, A. David Rodrigues and Manthena V.S. VarmaDrug Metabolism and Disposition May 2018, 46 (5) 692-696; DOI: https://doi.org/10.1124/dmd.117.079285
Kobayashi, Daisuke
- You have accessInterindividual Differences in the Expression of ATP-Binding Cassette and Solute Carrier Family Transporters in Human Skin: DNA Methylation Regulates Transcriptional Activity of the Human ABCC3 GeneTomoki Takechi, Takeshi Hirota, Tatsuya Sakai, Natsumi Maeda, Daisuke Kobayashi and Ichiro IeiriDrug Metabolism and Disposition May 2018, 46 (5) 628-635; DOI: https://doi.org/10.1124/dmd.117.079061
Korte, Daphne
- Open AccessExpression of Organic Anion Transporter 1 or 3 in Human Kidney Proximal Tubule Cells Reduces Cisplatin SensitivityTom T. G. Nieskens, Janny G. P. Peters, Dina Dabaghie, Daphne Korte, Katja Jansen, Alexander H. Van Asbeck, Neslihan N. Tavraz, Thomas Friedrich, Frans G. M. Russel, Rosalinde Masereeuw and Martijn J. WilmerDrug Metabolism and Disposition May 2018, 46 (5) 592-599; DOI: https://doi.org/10.1124/dmd.117.079384
Kroetz, Deanna L.
- You have accessRare Variants in the ABCG2 Promoter Modulate In Vivo ActivityRachel J. Eclov, Mee J. Kim, Robin Smith, Nadav Ahituv and Deanna L. KroetzDrug Metabolism and Disposition May 2018, 46 (5) 636-642; DOI: https://doi.org/10.1124/dmd.117.079541
Kulkarni, Supriya
- You have accessPhysiological Regulation of Drug Metabolism and Transport: Pregnancy, Microbiome, Inflammation, Infection, and FastingEdward T. Morgan, Joseph L. Dempsey, Sylvie M. Mimche, Tracey J. Lamb, Supriya Kulkarni, Julia Yue Cui, Hyunyoung Jeong and Angela L. SlittDrug Metabolism and Disposition May 2018, 46 (5) 503-513; DOI: https://doi.org/10.1124/dmd.117.079905
Kunz, Ryan C.
- You have accessComparison of Proteomic Quantification Approaches for Hepatic Drug Transporters: Multiplexed Global Quantitation Correlates with Targeted Proteomic QuantitationAnna Vildhede, Chuong Nguyen, Brian K. Erickson, Ryan C. Kunz, Richard Jones, Emi Kimoto, Francis Bourbonais, A. David Rodrigues and Manthena V.S. VarmaDrug Metabolism and Disposition May 2018, 46 (5) 692-696; DOI: https://doi.org/10.1124/dmd.117.079285
Kusuhara, Hiroyuki
- Open AccessA Clinical Quantitative Evaluation of Hepatobiliary Transport of [11C]Dehydropravastatin in Humans Using Positron Emission TomographyKen-ichi Kaneko, Masaaki Tanaka, Akira Ishii, Yumiko Katayama, Takayoshi Nakaoka, Satsuki Irie, Hideki Kawahata, Takashi Yamanaga, Yasuhiro Wada, Takeshi Miyake, Kota Toshimoto, Kazuya Maeda, Yilong Cui, Masaru Enomoto, Etsushi Kawamura, Norifumi Kawada, Joji Kawabe, Susumu Shiomi, Hiroyuki Kusuhara, Yuichi Sugiyama and Yasuyoshi WatanabeDrug Metabolism and Disposition May 2018, 46 (5) 719-728; DOI: https://doi.org/10.1124/dmd.118.080408
- You have accessOrganic Anion Transporting Polypeptide 1a4 is Responsible for the Hepatic Uptake of Cardiac Glycosides in MiceJunichi Takano, Kazuya Maeda, Hiroyuki Kusuhara and Yuichi SugiyamaDrug Metabolism and Disposition May 2018, 46 (5) 652-657; DOI: https://doi.org/10.1124/dmd.117.079483
L
Labriet, Adrien
- You have accessPost-transcriptional Regulation of UGT2B10 Hepatic Expression and Activity by Alternative SplicingAdrien Labriet, Eric P. Allain, Michèle Rouleau, Yannick Audet-Delage, Lyne Villeneuve and Chantal GuillemetteDrug Metabolism and Disposition May 2018, 46 (5) 514-524; DOI: https://doi.org/10.1124/dmd.117.079921
Lai, Yurong
- You have accessDrug Transporters in Xenobiotic Disposition and Pharmacokinetic PredictionQingcheng Mao, Yurong Lai and Joanne WangDrug Metabolism and Disposition May 2018, 46 (5) 561-566; DOI: https://doi.org/10.1124/dmd.118.081356
Lamb, Tracey J.
- You have accessPhysiological Regulation of Drug Metabolism and Transport: Pregnancy, Microbiome, Inflammation, Infection, and FastingEdward T. Morgan, Joseph L. Dempsey, Sylvie M. Mimche, Tracey J. Lamb, Supriya Kulkarni, Julia Yue Cui, Hyunyoung Jeong and Angela L. SlittDrug Metabolism and Disposition May 2018, 46 (5) 503-513; DOI: https://doi.org/10.1124/dmd.117.079905
Laramy, Janice K.
- You have accessBrain Distribution of a Novel MEK Inhibitor E6201: Implications in the Treatment of Melanoma Brain MetastasesGautham Gampa, Minjee Kim, Nicholas Cook-Rostie, Janice K. Laramy, Jann N. Sarkaria, Linda Paradiso, Louis DePalatis and William F. ElmquistDrug Metabolism and Disposition May 2018, 46 (5) 658-666; DOI: https://doi.org/10.1124/dmd.117.079194
Lee, Caroline A.
- You have accessMetabolism and Disposition of Verinurad, a Uric Acid Reabsorption Inhibitor, in HumansCaroline A. Lee, Chun Yang, Vishal Shah, Zancong Shen, David M. Wilson, Traci M. Ostertag, Jean-Luc Girardet, Jesse Hall and Michael GillenDrug Metabolism and Disposition May 2018, 46 (5) 532-541; DOI: https://doi.org/10.1124/dmd.117.078220
Lee, Wooin
- You have accessPhysiologically Based Pharmacokinetic Modeling of Bosentan Identifies the Saturable Hepatic Uptake As a Major Contributor to Its Nonlinear PharmacokineticsMasanobu Sato, Kota Toshimoto, Atsuko Tomaru, Takashi Yoshikado, Yuta Tanaka, Akihiro Hisaka, Wooin Lee and Yuichi SugiyamaDrug Metabolism and Disposition May 2018, 46 (5) 740-748; DOI: https://doi.org/10.1124/dmd.117.078972
Li, Weike
- You have accessIdentification of a NFκB Inhibition Site on the Proximal Promoter Region of Human Organic Anion Transporting Polypeptide 1A2 Coding Gene SLCO1A2Zhaojian Xiang, Weike Li, Lixue Wang, Jicai Yi, Kaiwen Chen and Mei HongDrug Metabolism and Disposition May 2018, 46 (5) 643-651; DOI: https://doi.org/10.1124/dmd.117.078832
Liao, Michael Z.
- You have accessHepatic Transport of 25-Hydroxyvitamin D3 Conjugates: A Mechanism of 25-Hydroxyvitamin D3 Delivery to the Intestinal TractChunying Gao, Michael Z. Liao, Lyrialle W. Han, Kenneth E. Thummel and Qingcheng MaoDrug Metabolism and Disposition May 2018, 46 (5) 581-591; DOI: https://doi.org/10.1124/dmd.117.078881
Liu, Melissa
- You have accessApixaban and Rosuvastatin Pharmacokinetics in Nonalcoholic Fatty Liver DiseaseRommel G. Tirona, Zahra Kassam, Ruth Strapp, Mala Ramu, Catherine Zhu, Melissa Liu, Ute I. Schwarz, Richard B. Kim, Bandar Al-Judaibi and Melanie D. BeatonDrug Metabolism and Disposition May 2018, 46 (5) 485-492; DOI: https://doi.org/10.1124/dmd.117.079624
M
Maeda, Kazuya
- Open AccessA Clinical Quantitative Evaluation of Hepatobiliary Transport of [11C]Dehydropravastatin in Humans Using Positron Emission TomographyKen-ichi Kaneko, Masaaki Tanaka, Akira Ishii, Yumiko Katayama, Takayoshi Nakaoka, Satsuki Irie, Hideki Kawahata, Takashi Yamanaga, Yasuhiro Wada, Takeshi Miyake, Kota Toshimoto, Kazuya Maeda, Yilong Cui, Masaru Enomoto, Etsushi Kawamura, Norifumi Kawada, Joji Kawabe, Susumu Shiomi, Hiroyuki Kusuhara, Yuichi Sugiyama and Yasuyoshi WatanabeDrug Metabolism and Disposition May 2018, 46 (5) 719-728; DOI: https://doi.org/10.1124/dmd.118.080408
- You have accessOrganic Anion Transporting Polypeptide 1a4 is Responsible for the Hepatic Uptake of Cardiac Glycosides in MiceJunichi Takano, Kazuya Maeda, Hiroyuki Kusuhara and Yuichi SugiyamaDrug Metabolism and Disposition May 2018, 46 (5) 652-657; DOI: https://doi.org/10.1124/dmd.117.079483
Maeda, Natsumi
- You have accessInterindividual Differences in the Expression of ATP-Binding Cassette and Solute Carrier Family Transporters in Human Skin: DNA Methylation Regulates Transcriptional Activity of the Human ABCC3 GeneTomoki Takechi, Takeshi Hirota, Tatsuya Sakai, Natsumi Maeda, Daisuke Kobayashi and Ichiro IeiriDrug Metabolism and Disposition May 2018, 46 (5) 628-635; DOI: https://doi.org/10.1124/dmd.117.079061
Mao, Qingcheng
- You have accessHepatic Transport of 25-Hydroxyvitamin D3 Conjugates: A Mechanism of 25-Hydroxyvitamin D3 Delivery to the Intestinal TractChunying Gao, Michael Z. Liao, Lyrialle W. Han, Kenneth E. Thummel and Qingcheng MaoDrug Metabolism and Disposition May 2018, 46 (5) 581-591; DOI: https://doi.org/10.1124/dmd.117.078881
- You have accessDrug Transporters in Xenobiotic Disposition and Pharmacokinetic PredictionQingcheng Mao, Yurong Lai and Joanne WangDrug Metabolism and Disposition May 2018, 46 (5) 561-566; DOI: https://doi.org/10.1124/dmd.118.081356
Masereeuw, Rosalinde
- Open AccessExpression of Organic Anion Transporter 1 or 3 in Human Kidney Proximal Tubule Cells Reduces Cisplatin SensitivityTom T. G. Nieskens, Janny G. P. Peters, Dina Dabaghie, Daphne Korte, Katja Jansen, Alexander H. Van Asbeck, Neslihan N. Tavraz, Thomas Friedrich, Frans G. M. Russel, Rosalinde Masereeuw and Martijn J. WilmerDrug Metabolism and Disposition May 2018, 46 (5) 592-599; DOI: https://doi.org/10.1124/dmd.117.079384
Matsunaga, Norikazu
- You have accessSandwich-Cultured Hepatocytes for Mechanistic Understanding of Hepatic Disposition of Parent Drugs and Metabolites by Transporter–Enzyme InterplayNorikazu Matsunaga, Yukina Fukuchi, Haruo Imawaka and Ikumi TamaiDrug Metabolism and Disposition May 2018, 46 (5) 680-691; DOI: https://doi.org/10.1124/dmd.117.079236
McCune, Jeannine S.
- You have accessIdentification of Intestinal UDP-Glucuronosyltransferase Inhibitors in Green Tea (Camellia sinensis) Using a Biochemometric Approach: Application to Raloxifene as a Test Drug via In Vitro to In Vivo ExtrapolationDan-Dan Tian, Joshua J. Kellogg, Neşe Okut, Nicholas H. Oberlies, Nadja B. Cech, Danny D. Shen, Jeannine S. McCune and Mary F. PaineDrug Metabolism and Disposition May 2018, 46 (5) 552-560; DOI: https://doi.org/10.1124/dmd.117.079491
Memon, Naureen
- You have accessInterindividual Regulation of the Breast Cancer Resistance Protein/ABCG2 Transporter in Term Human PlacentasKristin M. Bircsak, Jamie E. Moscovitz, Xia Wen, Faith Archer, Poi Yu Sofia Yuen, Moiz Mohammed, Naureen Memon, Barry I. Weinberger, Laura M. Saba, Anna M. Vetrano and Lauren M. AleksunesDrug Metabolism and Disposition May 2018, 46 (5) 619-627; DOI: https://doi.org/10.1124/dmd.117.079228
Mimche, Sylvie M.
- You have accessPhysiological Regulation of Drug Metabolism and Transport: Pregnancy, Microbiome, Inflammation, Infection, and FastingEdward T. Morgan, Joseph L. Dempsey, Sylvie M. Mimche, Tracey J. Lamb, Supriya Kulkarni, Julia Yue Cui, Hyunyoung Jeong and Angela L. SlittDrug Metabolism and Disposition May 2018, 46 (5) 503-513; DOI: https://doi.org/10.1124/dmd.117.079905
Miyake, Takeshi
- Open AccessA Clinical Quantitative Evaluation of Hepatobiliary Transport of [11C]Dehydropravastatin in Humans Using Positron Emission TomographyKen-ichi Kaneko, Masaaki Tanaka, Akira Ishii, Yumiko Katayama, Takayoshi Nakaoka, Satsuki Irie, Hideki Kawahata, Takashi Yamanaga, Yasuhiro Wada, Takeshi Miyake, Kota Toshimoto, Kazuya Maeda, Yilong Cui, Masaru Enomoto, Etsushi Kawamura, Norifumi Kawada, Joji Kawabe, Susumu Shiomi, Hiroyuki Kusuhara, Yuichi Sugiyama and Yasuyoshi WatanabeDrug Metabolism and Disposition May 2018, 46 (5) 719-728; DOI: https://doi.org/10.1124/dmd.118.080408
Mohammed, Moiz
- You have accessInterindividual Regulation of the Breast Cancer Resistance Protein/ABCG2 Transporter in Term Human PlacentasKristin M. Bircsak, Jamie E. Moscovitz, Xia Wen, Faith Archer, Poi Yu Sofia Yuen, Moiz Mohammed, Naureen Memon, Barry I. Weinberger, Laura M. Saba, Anna M. Vetrano and Lauren M. AleksunesDrug Metabolism and Disposition May 2018, 46 (5) 619-627; DOI: https://doi.org/10.1124/dmd.117.079228
Morgan, Edward T.
- You have accessPhysiological Regulation of Drug Metabolism and Transport: Pregnancy, Microbiome, Inflammation, Infection, and FastingEdward T. Morgan, Joseph L. Dempsey, Sylvie M. Mimche, Tracey J. Lamb, Supriya Kulkarni, Julia Yue Cui, Hyunyoung Jeong and Angela L. SlittDrug Metabolism and Disposition May 2018, 46 (5) 503-513; DOI: https://doi.org/10.1124/dmd.117.079905
Morgan, Ryan E.
- You have accessIntravital Multiphoton Microscopy with Fluorescent Bile Salts in Rats as an In Vivo Biomarker for Hepatobiliary Transport InhibitionJennifer Ryan, Ryan E. Morgan, Yuan Chen, Laurie P. Volak, Robert T. Dunn and Kenneth W. DunnDrug Metabolism and Disposition May 2018, 46 (5) 704-718; DOI: https://doi.org/10.1124/dmd.117.079277
Morris, Marilyn E.
- You have accessPrediction of the Effects of Renal Impairment on Clearance for Organic Cation Drugs that Undergo Renal Secretion: A Simulation-Based StudyKristin E. Follman and Marilyn E. MorrisDrug Metabolism and Disposition May 2018, 46 (5) 758-769; DOI: https://doi.org/10.1124/dmd.117.079558
Moscovitz, Jamie E.
- You have accessInterindividual Regulation of the Breast Cancer Resistance Protein/ABCG2 Transporter in Term Human PlacentasKristin M. Bircsak, Jamie E. Moscovitz, Xia Wen, Faith Archer, Poi Yu Sofia Yuen, Moiz Mohammed, Naureen Memon, Barry I. Weinberger, Laura M. Saba, Anna M. Vetrano and Lauren M. AleksunesDrug Metabolism and Disposition May 2018, 46 (5) 619-627; DOI: https://doi.org/10.1124/dmd.117.079228
N
Nakaoka, Takayoshi
- Open AccessA Clinical Quantitative Evaluation of Hepatobiliary Transport of [11C]Dehydropravastatin in Humans Using Positron Emission TomographyKen-ichi Kaneko, Masaaki Tanaka, Akira Ishii, Yumiko Katayama, Takayoshi Nakaoka, Satsuki Irie, Hideki Kawahata, Takashi Yamanaga, Yasuhiro Wada, Takeshi Miyake, Kota Toshimoto, Kazuya Maeda, Yilong Cui, Masaru Enomoto, Etsushi Kawamura, Norifumi Kawada, Joji Kawabe, Susumu Shiomi, Hiroyuki Kusuhara, Yuichi Sugiyama and Yasuyoshi WatanabeDrug Metabolism and Disposition May 2018, 46 (5) 719-728; DOI: https://doi.org/10.1124/dmd.118.080408
Nguyen, Chuong
- You have accessComparison of Proteomic Quantification Approaches for Hepatic Drug Transporters: Multiplexed Global Quantitation Correlates with Targeted Proteomic QuantitationAnna Vildhede, Chuong Nguyen, Brian K. Erickson, Ryan C. Kunz, Richard Jones, Emi Kimoto, Francis Bourbonais, A. David Rodrigues and Manthena V.S. VarmaDrug Metabolism and Disposition May 2018, 46 (5) 692-696; DOI: https://doi.org/10.1124/dmd.117.079285
Nieskens, Tom T. G.
- Open AccessExpression of Organic Anion Transporter 1 or 3 in Human Kidney Proximal Tubule Cells Reduces Cisplatin SensitivityTom T. G. Nieskens, Janny G. P. Peters, Dina Dabaghie, Daphne Korte, Katja Jansen, Alexander H. Van Asbeck, Neslihan N. Tavraz, Thomas Friedrich, Frans G. M. Russel, Rosalinde Masereeuw and Martijn J. WilmerDrug Metabolism and Disposition May 2018, 46 (5) 592-599; DOI: https://doi.org/10.1124/dmd.117.079384
O
Obach, R. Scott
- You have accessBiosynthesis and Identification of Metabolites of Maraviroc and Their Use in Experiments to Delineate the Relative Contributions of Cytochrome P4503A4 versus 3A5Elaine Tseng, Gwendolyn D. Fate, Gregory S. Walker, Theunis C. Goosen and R. Scott ObachDrug Metabolism and Disposition May 2018, 46 (5) 493-502; DOI: https://doi.org/10.1124/dmd.117.079855
Oberlies, Nicholas H.
- You have accessIdentification of Intestinal UDP-Glucuronosyltransferase Inhibitors in Green Tea (Camellia sinensis) Using a Biochemometric Approach: Application to Raloxifene as a Test Drug via In Vitro to In Vivo ExtrapolationDan-Dan Tian, Joshua J. Kellogg, Neşe Okut, Nicholas H. Oberlies, Nadja B. Cech, Danny D. Shen, Jeannine S. McCune and Mary F. PaineDrug Metabolism and Disposition May 2018, 46 (5) 552-560; DOI: https://doi.org/10.1124/dmd.117.079491
Okut, Neşe
- You have accessIdentification of Intestinal UDP-Glucuronosyltransferase Inhibitors in Green Tea (Camellia sinensis) Using a Biochemometric Approach: Application to Raloxifene as a Test Drug via In Vitro to In Vivo ExtrapolationDan-Dan Tian, Joshua J. Kellogg, Neşe Okut, Nicholas H. Oberlies, Nadja B. Cech, Danny D. Shen, Jeannine S. McCune and Mary F. PaineDrug Metabolism and Disposition May 2018, 46 (5) 552-560; DOI: https://doi.org/10.1124/dmd.117.079491
Oorts, Marlies
- You have accessMRP2 Inhibition by HIV Protease Inhibitors in Rat and Human Hepatocytes: A Quantitative Confocal Microscopy StudyNico Holmstock, Marlies Oorts, Jan Snoeys and Pieter AnnaertDrug Metabolism and Disposition May 2018, 46 (5) 697-703; DOI: https://doi.org/10.1124/dmd.117.079467
Ostertag, Traci M.
- You have accessMetabolism and Disposition of Verinurad, a Uric Acid Reabsorption Inhibitor, in HumansCaroline A. Lee, Chun Yang, Vishal Shah, Zancong Shen, David M. Wilson, Traci M. Ostertag, Jean-Luc Girardet, Jesse Hall and Michael GillenDrug Metabolism and Disposition May 2018, 46 (5) 532-541; DOI: https://doi.org/10.1124/dmd.117.078220
P
Paine, Mary F.
- You have accessIdentification of Intestinal UDP-Glucuronosyltransferase Inhibitors in Green Tea (Camellia sinensis) Using a Biochemometric Approach: Application to Raloxifene as a Test Drug via In Vitro to In Vivo ExtrapolationDan-Dan Tian, Joshua J. Kellogg, Neşe Okut, Nicholas H. Oberlies, Nadja B. Cech, Danny D. Shen, Jeannine S. McCune and Mary F. PaineDrug Metabolism and Disposition May 2018, 46 (5) 552-560; DOI: https://doi.org/10.1124/dmd.117.079491
Paradiso, Linda
- You have accessBrain Distribution of a Novel MEK Inhibitor E6201: Implications in the Treatment of Melanoma Brain MetastasesGautham Gampa, Minjee Kim, Nicholas Cook-Rostie, Janice K. Laramy, Jann N. Sarkaria, Linda Paradiso, Louis DePalatis and William F. ElmquistDrug Metabolism and Disposition May 2018, 46 (5) 658-666; DOI: https://doi.org/10.1124/dmd.117.079194
Peters, Janny G. P.
- Open AccessExpression of Organic Anion Transporter 1 or 3 in Human Kidney Proximal Tubule Cells Reduces Cisplatin SensitivityTom T. G. Nieskens, Janny G. P. Peters, Dina Dabaghie, Daphne Korte, Katja Jansen, Alexander H. Van Asbeck, Neslihan N. Tavraz, Thomas Friedrich, Frans G. M. Russel, Rosalinde Masereeuw and Martijn J. WilmerDrug Metabolism and Disposition May 2018, 46 (5) 592-599; DOI: https://doi.org/10.1124/dmd.117.079384
Potukuchi, Praveen K.
- You have accessBeyond Competitive Inhibition: Regulation of ABC Transporters by Kinases and Protein-Protein Interactions as Potential Mechanisms of Drug-Drug InteractionsRebecca R. Crawford, Praveen K. Potukuchi, Erin G. Schuetz and John D. SchuetzDrug Metabolism and Disposition May 2018, 46 (5) 567-580; DOI: https://doi.org/10.1124/dmd.118.080663
R
Rahman, MD Fazlur
- Open AccessIdentification of Structural and Molecular Features Involved in the Transport of 3′-Deoxy-Nucleoside Analogs by Human Equilibrative Nucleoside Transporter 3MD Fazlur Rahman, Radhika Raj and Rajgopal GovindarajanDrug Metabolism and Disposition May 2018, 46 (5) 600-609; DOI: https://doi.org/10.1124/dmd.117.079400
Raj, Radhika
- Open AccessIdentification of Structural and Molecular Features Involved in the Transport of 3′-Deoxy-Nucleoside Analogs by Human Equilibrative Nucleoside Transporter 3MD Fazlur Rahman, Radhika Raj and Rajgopal GovindarajanDrug Metabolism and Disposition May 2018, 46 (5) 600-609; DOI: https://doi.org/10.1124/dmd.117.079400
Ramu, Mala
- You have accessApixaban and Rosuvastatin Pharmacokinetics in Nonalcoholic Fatty Liver DiseaseRommel G. Tirona, Zahra Kassam, Ruth Strapp, Mala Ramu, Catherine Zhu, Melissa Liu, Ute I. Schwarz, Richard B. Kim, Bandar Al-Judaibi and Melanie D. BeatonDrug Metabolism and Disposition May 2018, 46 (5) 485-492; DOI: https://doi.org/10.1124/dmd.117.079624
Rodrigues, A. David
- You have accessComparison of Proteomic Quantification Approaches for Hepatic Drug Transporters: Multiplexed Global Quantitation Correlates with Targeted Proteomic QuantitationAnna Vildhede, Chuong Nguyen, Brian K. Erickson, Ryan C. Kunz, Richard Jones, Emi Kimoto, Francis Bourbonais, A. David Rodrigues and Manthena V.S. VarmaDrug Metabolism and Disposition May 2018, 46 (5) 692-696; DOI: https://doi.org/10.1124/dmd.117.079285
Rouleau, Michèle
- You have accessPost-transcriptional Regulation of UGT2B10 Hepatic Expression and Activity by Alternative SplicingAdrien Labriet, Eric P. Allain, Michèle Rouleau, Yannick Audet-Delage, Lyne Villeneuve and Chantal GuillemetteDrug Metabolism and Disposition May 2018, 46 (5) 514-524; DOI: https://doi.org/10.1124/dmd.117.079921
Russel, Frans G. M.
- Open AccessExpression of Organic Anion Transporter 1 or 3 in Human Kidney Proximal Tubule Cells Reduces Cisplatin SensitivityTom T. G. Nieskens, Janny G. P. Peters, Dina Dabaghie, Daphne Korte, Katja Jansen, Alexander H. Van Asbeck, Neslihan N. Tavraz, Thomas Friedrich, Frans G. M. Russel, Rosalinde Masereeuw and Martijn J. WilmerDrug Metabolism and Disposition May 2018, 46 (5) 592-599; DOI: https://doi.org/10.1124/dmd.117.079384
Ryan, Jennifer
- You have accessIntravital Multiphoton Microscopy with Fluorescent Bile Salts in Rats as an In Vivo Biomarker for Hepatobiliary Transport InhibitionJennifer Ryan, Ryan E. Morgan, Yuan Chen, Laurie P. Volak, Robert T. Dunn and Kenneth W. DunnDrug Metabolism and Disposition May 2018, 46 (5) 704-718; DOI: https://doi.org/10.1124/dmd.117.079277
S
Saba, Laura M.
- You have accessInterindividual Regulation of the Breast Cancer Resistance Protein/ABCG2 Transporter in Term Human PlacentasKristin M. Bircsak, Jamie E. Moscovitz, Xia Wen, Faith Archer, Poi Yu Sofia Yuen, Moiz Mohammed, Naureen Memon, Barry I. Weinberger, Laura M. Saba, Anna M. Vetrano and Lauren M. AleksunesDrug Metabolism and Disposition May 2018, 46 (5) 619-627; DOI: https://doi.org/10.1124/dmd.117.079228
Saigusa, Daisuke
- You have accessLiver Zonation Index of Drug Transporter and Metabolizing Enzyme Protein Expressions in Mouse Liver AcinusMasanori Tachikawa, Yuna Sumiyoshiya, Daisuke Saigusa, Kazunari Sasaki, Michitoshi Watanabe, Yasuo Uchida and Tetsuya TerasakiDrug Metabolism and Disposition May 2018, 46 (5) 610-618; DOI: https://doi.org/10.1124/dmd.117.079244
Sakai, Tatsuya
- You have accessInterindividual Differences in the Expression of ATP-Binding Cassette and Solute Carrier Family Transporters in Human Skin: DNA Methylation Regulates Transcriptional Activity of the Human ABCC3 GeneTomoki Takechi, Takeshi Hirota, Tatsuya Sakai, Natsumi Maeda, Daisuke Kobayashi and Ichiro IeiriDrug Metabolism and Disposition May 2018, 46 (5) 628-635; DOI: https://doi.org/10.1124/dmd.117.079061
Sarkaria, Jann N.
- You have accessBrain Distribution of a Novel MEK Inhibitor E6201: Implications in the Treatment of Melanoma Brain MetastasesGautham Gampa, Minjee Kim, Nicholas Cook-Rostie, Janice K. Laramy, Jann N. Sarkaria, Linda Paradiso, Louis DePalatis and William F. ElmquistDrug Metabolism and Disposition May 2018, 46 (5) 658-666; DOI: https://doi.org/10.1124/dmd.117.079194
Sasaki, Kazunari
- You have accessLiver Zonation Index of Drug Transporter and Metabolizing Enzyme Protein Expressions in Mouse Liver AcinusMasanori Tachikawa, Yuna Sumiyoshiya, Daisuke Saigusa, Kazunari Sasaki, Michitoshi Watanabe, Yasuo Uchida and Tetsuya TerasakiDrug Metabolism and Disposition May 2018, 46 (5) 610-618; DOI: https://doi.org/10.1124/dmd.117.079244
Sato, Masanobu
- You have accessPhysiologically Based Pharmacokinetic Modeling of Bosentan Identifies the Saturable Hepatic Uptake As a Major Contributor to Its Nonlinear PharmacokineticsMasanobu Sato, Kota Toshimoto, Atsuko Tomaru, Takashi Yoshikado, Yuta Tanaka, Akihiro Hisaka, Wooin Lee and Yuichi SugiyamaDrug Metabolism and Disposition May 2018, 46 (5) 740-748; DOI: https://doi.org/10.1124/dmd.117.078972
Schuetz, Erin G.
- You have accessBeyond Competitive Inhibition: Regulation of ABC Transporters by Kinases and Protein-Protein Interactions as Potential Mechanisms of Drug-Drug InteractionsRebecca R. Crawford, Praveen K. Potukuchi, Erin G. Schuetz and John D. SchuetzDrug Metabolism and Disposition May 2018, 46 (5) 567-580; DOI: https://doi.org/10.1124/dmd.118.080663
Schuetz, John D.
- You have accessBeyond Competitive Inhibition: Regulation of ABC Transporters by Kinases and Protein-Protein Interactions as Potential Mechanisms of Drug-Drug InteractionsRebecca R. Crawford, Praveen K. Potukuchi, Erin G. Schuetz and John D. SchuetzDrug Metabolism and Disposition May 2018, 46 (5) 567-580; DOI: https://doi.org/10.1124/dmd.118.080663
Schwarz, Ute I.
- You have accessApixaban and Rosuvastatin Pharmacokinetics in Nonalcoholic Fatty Liver DiseaseRommel G. Tirona, Zahra Kassam, Ruth Strapp, Mala Ramu, Catherine Zhu, Melissa Liu, Ute I. Schwarz, Richard B. Kim, Bandar Al-Judaibi and Melanie D. BeatonDrug Metabolism and Disposition May 2018, 46 (5) 485-492; DOI: https://doi.org/10.1124/dmd.117.079624
Shah, Vishal
- You have accessMetabolism and Disposition of Verinurad, a Uric Acid Reabsorption Inhibitor, in HumansCaroline A. Lee, Chun Yang, Vishal Shah, Zancong Shen, David M. Wilson, Traci M. Ostertag, Jean-Luc Girardet, Jesse Hall and Michael GillenDrug Metabolism and Disposition May 2018, 46 (5) 532-541; DOI: https://doi.org/10.1124/dmd.117.078220
Shan, Mangting
- You have accessGeneration and Characterization of a CYP2C11-Null Rat Model by Using the CRISPR/Cas9 MethodYuan Wei, Li Yang, Xiaoyan Zhang, Danjuan Sui, Changsuo Wang, Kai Wang, Mangting Shan, Dayong Guo and Hongyu WangDrug Metabolism and Disposition May 2018, 46 (5) 525-531; DOI: https://doi.org/10.1124/dmd.117.078444
Shen, Danny D.
- You have accessIdentification of Intestinal UDP-Glucuronosyltransferase Inhibitors in Green Tea (Camellia sinensis) Using a Biochemometric Approach: Application to Raloxifene as a Test Drug via In Vitro to In Vivo ExtrapolationDan-Dan Tian, Joshua J. Kellogg, Neşe Okut, Nicholas H. Oberlies, Nadja B. Cech, Danny D. Shen, Jeannine S. McCune and Mary F. PaineDrug Metabolism and Disposition May 2018, 46 (5) 552-560; DOI: https://doi.org/10.1124/dmd.117.079491
Shen, Zancong
- You have accessMetabolism and Disposition of Verinurad, a Uric Acid Reabsorption Inhibitor, in HumansCaroline A. Lee, Chun Yang, Vishal Shah, Zancong Shen, David M. Wilson, Traci M. Ostertag, Jean-Luc Girardet, Jesse Hall and Michael GillenDrug Metabolism and Disposition May 2018, 46 (5) 532-541; DOI: https://doi.org/10.1124/dmd.117.078220
Shiomi, Susumu
- Open AccessA Clinical Quantitative Evaluation of Hepatobiliary Transport of [11C]Dehydropravastatin in Humans Using Positron Emission TomographyKen-ichi Kaneko, Masaaki Tanaka, Akira Ishii, Yumiko Katayama, Takayoshi Nakaoka, Satsuki Irie, Hideki Kawahata, Takashi Yamanaga, Yasuhiro Wada, Takeshi Miyake, Kota Toshimoto, Kazuya Maeda, Yilong Cui, Masaru Enomoto, Etsushi Kawamura, Norifumi Kawada, Joji Kawabe, Susumu Shiomi, Hiroyuki Kusuhara, Yuichi Sugiyama and Yasuyoshi WatanabeDrug Metabolism and Disposition May 2018, 46 (5) 719-728; DOI: https://doi.org/10.1124/dmd.118.080408
Slitt, Angela L.
- You have accessPhysiological Regulation of Drug Metabolism and Transport: Pregnancy, Microbiome, Inflammation, Infection, and FastingEdward T. Morgan, Joseph L. Dempsey, Sylvie M. Mimche, Tracey J. Lamb, Supriya Kulkarni, Julia Yue Cui, Hyunyoung Jeong and Angela L. SlittDrug Metabolism and Disposition May 2018, 46 (5) 503-513; DOI: https://doi.org/10.1124/dmd.117.079905
Smith, Robin
- You have accessRare Variants in the ABCG2 Promoter Modulate In Vivo ActivityRachel J. Eclov, Mee J. Kim, Robin Smith, Nadav Ahituv and Deanna L. KroetzDrug Metabolism and Disposition May 2018, 46 (5) 636-642; DOI: https://doi.org/10.1124/dmd.117.079541
Snoeys, Jan
- You have accessMRP2 Inhibition by HIV Protease Inhibitors in Rat and Human Hepatocytes: A Quantitative Confocal Microscopy StudyNico Holmstock, Marlies Oorts, Jan Snoeys and Pieter AnnaertDrug Metabolism and Disposition May 2018, 46 (5) 697-703; DOI: https://doi.org/10.1124/dmd.117.079467
Strapp, Ruth
- You have accessApixaban and Rosuvastatin Pharmacokinetics in Nonalcoholic Fatty Liver DiseaseRommel G. Tirona, Zahra Kassam, Ruth Strapp, Mala Ramu, Catherine Zhu, Melissa Liu, Ute I. Schwarz, Richard B. Kim, Bandar Al-Judaibi and Melanie D. BeatonDrug Metabolism and Disposition May 2018, 46 (5) 485-492; DOI: https://doi.org/10.1124/dmd.117.079624
Sugiyama, Yuichi
- Open AccessA Clinical Quantitative Evaluation of Hepatobiliary Transport of [11C]Dehydropravastatin in Humans Using Positron Emission TomographyKen-ichi Kaneko, Masaaki Tanaka, Akira Ishii, Yumiko Katayama, Takayoshi Nakaoka, Satsuki Irie, Hideki Kawahata, Takashi Yamanaga, Yasuhiro Wada, Takeshi Miyake, Kota Toshimoto, Kazuya Maeda, Yilong Cui, Masaru Enomoto, Etsushi Kawamura, Norifumi Kawada, Joji Kawabe, Susumu Shiomi, Hiroyuki Kusuhara, Yuichi Sugiyama and Yasuyoshi WatanabeDrug Metabolism and Disposition May 2018, 46 (5) 719-728; DOI: https://doi.org/10.1124/dmd.118.080408
- You have accessOrganic Anion Transporting Polypeptide 1a4 is Responsible for the Hepatic Uptake of Cardiac Glycosides in MiceJunichi Takano, Kazuya Maeda, Hiroyuki Kusuhara and Yuichi SugiyamaDrug Metabolism and Disposition May 2018, 46 (5) 652-657; DOI: https://doi.org/10.1124/dmd.117.079483
- You have accessEvaluation of Alteration in Hepatic and Intestinal BCRP Function In Vivo from ABCG2 c.421C>A Polymorphism Based on PBPK Analysis of RosuvastatinAzusa Futatsugi, Kota Toshimoto, Takashi Yoshikado, Yuichi Sugiyama and Yukio KatoDrug Metabolism and Disposition May 2018, 46 (5) 749-757; DOI: https://doi.org/10.1124/dmd.117.078816
- You have accessPhysiologically Based Pharmacokinetic Modeling of Bosentan Identifies the Saturable Hepatic Uptake As a Major Contributor to Its Nonlinear PharmacokineticsMasanobu Sato, Kota Toshimoto, Atsuko Tomaru, Takashi Yoshikado, Yuta Tanaka, Akihiro Hisaka, Wooin Lee and Yuichi SugiyamaDrug Metabolism and Disposition May 2018, 46 (5) 740-748; DOI: https://doi.org/10.1124/dmd.117.078972
Sui, Danjuan
- You have accessGeneration and Characterization of a CYP2C11-Null Rat Model by Using the CRISPR/Cas9 MethodYuan Wei, Li Yang, Xiaoyan Zhang, Danjuan Sui, Changsuo Wang, Kai Wang, Mangting Shan, Dayong Guo and Hongyu WangDrug Metabolism and Disposition May 2018, 46 (5) 525-531; DOI: https://doi.org/10.1124/dmd.117.078444
Sumiyoshiya, Yuna
- You have accessLiver Zonation Index of Drug Transporter and Metabolizing Enzyme Protein Expressions in Mouse Liver AcinusMasanori Tachikawa, Yuna Sumiyoshiya, Daisuke Saigusa, Kazunari Sasaki, Michitoshi Watanabe, Yasuo Uchida and Tetsuya TerasakiDrug Metabolism and Disposition May 2018, 46 (5) 610-618; DOI: https://doi.org/10.1124/dmd.117.079244
T
Tachikawa, Masanori
- You have accessLiver Zonation Index of Drug Transporter and Metabolizing Enzyme Protein Expressions in Mouse Liver AcinusMasanori Tachikawa, Yuna Sumiyoshiya, Daisuke Saigusa, Kazunari Sasaki, Michitoshi Watanabe, Yasuo Uchida and Tetsuya TerasakiDrug Metabolism and Disposition May 2018, 46 (5) 610-618; DOI: https://doi.org/10.1124/dmd.117.079244
Takano, Junichi
- You have accessOrganic Anion Transporting Polypeptide 1a4 is Responsible for the Hepatic Uptake of Cardiac Glycosides in MiceJunichi Takano, Kazuya Maeda, Hiroyuki Kusuhara and Yuichi SugiyamaDrug Metabolism and Disposition May 2018, 46 (5) 652-657; DOI: https://doi.org/10.1124/dmd.117.079483
Takechi, Tomoki
- You have accessInterindividual Differences in the Expression of ATP-Binding Cassette and Solute Carrier Family Transporters in Human Skin: DNA Methylation Regulates Transcriptional Activity of the Human ABCC3 GeneTomoki Takechi, Takeshi Hirota, Tatsuya Sakai, Natsumi Maeda, Daisuke Kobayashi and Ichiro IeiriDrug Metabolism and Disposition May 2018, 46 (5) 628-635; DOI: https://doi.org/10.1124/dmd.117.079061
Tamai, Ikumi
- You have accessSandwich-Cultured Hepatocytes for Mechanistic Understanding of Hepatic Disposition of Parent Drugs and Metabolites by Transporter–Enzyme InterplayNorikazu Matsunaga, Yukina Fukuchi, Haruo Imawaka and Ikumi TamaiDrug Metabolism and Disposition May 2018, 46 (5) 680-691; DOI: https://doi.org/10.1124/dmd.117.079236
Tanaka, Masaaki
- Open AccessA Clinical Quantitative Evaluation of Hepatobiliary Transport of [11C]Dehydropravastatin in Humans Using Positron Emission TomographyKen-ichi Kaneko, Masaaki Tanaka, Akira Ishii, Yumiko Katayama, Takayoshi Nakaoka, Satsuki Irie, Hideki Kawahata, Takashi Yamanaga, Yasuhiro Wada, Takeshi Miyake, Kota Toshimoto, Kazuya Maeda, Yilong Cui, Masaru Enomoto, Etsushi Kawamura, Norifumi Kawada, Joji Kawabe, Susumu Shiomi, Hiroyuki Kusuhara, Yuichi Sugiyama and Yasuyoshi WatanabeDrug Metabolism and Disposition May 2018, 46 (5) 719-728; DOI: https://doi.org/10.1124/dmd.118.080408
Tanaka, Yuta
- You have accessPhysiologically Based Pharmacokinetic Modeling of Bosentan Identifies the Saturable Hepatic Uptake As a Major Contributor to Its Nonlinear PharmacokineticsMasanobu Sato, Kota Toshimoto, Atsuko Tomaru, Takashi Yoshikado, Yuta Tanaka, Akihiro Hisaka, Wooin Lee and Yuichi SugiyamaDrug Metabolism and Disposition May 2018, 46 (5) 740-748; DOI: https://doi.org/10.1124/dmd.117.078972
Tavraz, Neslihan N.
- Open AccessExpression of Organic Anion Transporter 1 or 3 in Human Kidney Proximal Tubule Cells Reduces Cisplatin SensitivityTom T. G. Nieskens, Janny G. P. Peters, Dina Dabaghie, Daphne Korte, Katja Jansen, Alexander H. Van Asbeck, Neslihan N. Tavraz, Thomas Friedrich, Frans G. M. Russel, Rosalinde Masereeuw and Martijn J. WilmerDrug Metabolism and Disposition May 2018, 46 (5) 592-599; DOI: https://doi.org/10.1124/dmd.117.079384
Terasaki, Tetsuya
- You have accessLiver Zonation Index of Drug Transporter and Metabolizing Enzyme Protein Expressions in Mouse Liver AcinusMasanori Tachikawa, Yuna Sumiyoshiya, Daisuke Saigusa, Kazunari Sasaki, Michitoshi Watanabe, Yasuo Uchida and Tetsuya TerasakiDrug Metabolism and Disposition May 2018, 46 (5) 610-618; DOI: https://doi.org/10.1124/dmd.117.079244
Thummel, Kenneth E.
- You have accessHepatic Transport of 25-Hydroxyvitamin D3 Conjugates: A Mechanism of 25-Hydroxyvitamin D3 Delivery to the Intestinal TractChunying Gao, Michael Z. Liao, Lyrialle W. Han, Kenneth E. Thummel and Qingcheng MaoDrug Metabolism and Disposition May 2018, 46 (5) 581-591; DOI: https://doi.org/10.1124/dmd.117.078881
Tian, Dan-Dan
- You have accessIdentification of Intestinal UDP-Glucuronosyltransferase Inhibitors in Green Tea (Camellia sinensis) Using a Biochemometric Approach: Application to Raloxifene as a Test Drug via In Vitro to In Vivo ExtrapolationDan-Dan Tian, Joshua J. Kellogg, Neşe Okut, Nicholas H. Oberlies, Nadja B. Cech, Danny D. Shen, Jeannine S. McCune and Mary F. PaineDrug Metabolism and Disposition May 2018, 46 (5) 552-560; DOI: https://doi.org/10.1124/dmd.117.079491
Tirona, Rommel G.
- You have accessApixaban and Rosuvastatin Pharmacokinetics in Nonalcoholic Fatty Liver DiseaseRommel G. Tirona, Zahra Kassam, Ruth Strapp, Mala Ramu, Catherine Zhu, Melissa Liu, Ute I. Schwarz, Richard B. Kim, Bandar Al-Judaibi and Melanie D. BeatonDrug Metabolism and Disposition May 2018, 46 (5) 485-492; DOI: https://doi.org/10.1124/dmd.117.079624
Tomaru, Atsuko
- You have accessPhysiologically Based Pharmacokinetic Modeling of Bosentan Identifies the Saturable Hepatic Uptake As a Major Contributor to Its Nonlinear PharmacokineticsMasanobu Sato, Kota Toshimoto, Atsuko Tomaru, Takashi Yoshikado, Yuta Tanaka, Akihiro Hisaka, Wooin Lee and Yuichi SugiyamaDrug Metabolism and Disposition May 2018, 46 (5) 740-748; DOI: https://doi.org/10.1124/dmd.117.078972
Toshimoto, Kota
- Open AccessA Clinical Quantitative Evaluation of Hepatobiliary Transport of [11C]Dehydropravastatin in Humans Using Positron Emission TomographyKen-ichi Kaneko, Masaaki Tanaka, Akira Ishii, Yumiko Katayama, Takayoshi Nakaoka, Satsuki Irie, Hideki Kawahata, Takashi Yamanaga, Yasuhiro Wada, Takeshi Miyake, Kota Toshimoto, Kazuya Maeda, Yilong Cui, Masaru Enomoto, Etsushi Kawamura, Norifumi Kawada, Joji Kawabe, Susumu Shiomi, Hiroyuki Kusuhara, Yuichi Sugiyama and Yasuyoshi WatanabeDrug Metabolism and Disposition May 2018, 46 (5) 719-728; DOI: https://doi.org/10.1124/dmd.118.080408
- You have accessEvaluation of Alteration in Hepatic and Intestinal BCRP Function In Vivo from ABCG2 c.421C>A Polymorphism Based on PBPK Analysis of RosuvastatinAzusa Futatsugi, Kota Toshimoto, Takashi Yoshikado, Yuichi Sugiyama and Yukio KatoDrug Metabolism and Disposition May 2018, 46 (5) 749-757; DOI: https://doi.org/10.1124/dmd.117.078816
- You have accessPhysiologically Based Pharmacokinetic Modeling of Bosentan Identifies the Saturable Hepatic Uptake As a Major Contributor to Its Nonlinear PharmacokineticsMasanobu Sato, Kota Toshimoto, Atsuko Tomaru, Takashi Yoshikado, Yuta Tanaka, Akihiro Hisaka, Wooin Lee and Yuichi SugiyamaDrug Metabolism and Disposition May 2018, 46 (5) 740-748; DOI: https://doi.org/10.1124/dmd.117.078972
Tseng, Elaine
- You have accessBiosynthesis and Identification of Metabolites of Maraviroc and Their Use in Experiments to Delineate the Relative Contributions of Cytochrome P4503A4 versus 3A5Elaine Tseng, Gwendolyn D. Fate, Gregory S. Walker, Theunis C. Goosen and R. Scott ObachDrug Metabolism and Disposition May 2018, 46 (5) 493-502; DOI: https://doi.org/10.1124/dmd.117.079855
U
Uchida, Yasuo
- You have accessLiver Zonation Index of Drug Transporter and Metabolizing Enzyme Protein Expressions in Mouse Liver AcinusMasanori Tachikawa, Yuna Sumiyoshiya, Daisuke Saigusa, Kazunari Sasaki, Michitoshi Watanabe, Yasuo Uchida and Tetsuya TerasakiDrug Metabolism and Disposition May 2018, 46 (5) 610-618; DOI: https://doi.org/10.1124/dmd.117.079244
V
Van Asbeck, Alexander H.
- Open AccessExpression of Organic Anion Transporter 1 or 3 in Human Kidney Proximal Tubule Cells Reduces Cisplatin SensitivityTom T. G. Nieskens, Janny G. P. Peters, Dina Dabaghie, Daphne Korte, Katja Jansen, Alexander H. Van Asbeck, Neslihan N. Tavraz, Thomas Friedrich, Frans G. M. Russel, Rosalinde Masereeuw and Martijn J. WilmerDrug Metabolism and Disposition May 2018, 46 (5) 592-599; DOI: https://doi.org/10.1124/dmd.117.079384
Varma, Manthena V. S.
- You have accessNavigating Transporter Sciences in Pharmacokinetics Characterization Using the Extended Clearance Classification SystemAyman F. El-Kattan and Manthena V. S. VarmaDrug Metabolism and Disposition May 2018, 46 (5) 729-739; DOI: https://doi.org/10.1124/dmd.117.080044
Varma, Manthena V.S.
- You have accessComparison of Proteomic Quantification Approaches for Hepatic Drug Transporters: Multiplexed Global Quantitation Correlates with Targeted Proteomic QuantitationAnna Vildhede, Chuong Nguyen, Brian K. Erickson, Ryan C. Kunz, Richard Jones, Emi Kimoto, Francis Bourbonais, A. David Rodrigues and Manthena V.S. VarmaDrug Metabolism and Disposition May 2018, 46 (5) 692-696; DOI: https://doi.org/10.1124/dmd.117.079285
Vetrano, Anna M.
- You have accessInterindividual Regulation of the Breast Cancer Resistance Protein/ABCG2 Transporter in Term Human PlacentasKristin M. Bircsak, Jamie E. Moscovitz, Xia Wen, Faith Archer, Poi Yu Sofia Yuen, Moiz Mohammed, Naureen Memon, Barry I. Weinberger, Laura M. Saba, Anna M. Vetrano and Lauren M. AleksunesDrug Metabolism and Disposition May 2018, 46 (5) 619-627; DOI: https://doi.org/10.1124/dmd.117.079228
Vildhede, Anna
- You have accessComparison of Proteomic Quantification Approaches for Hepatic Drug Transporters: Multiplexed Global Quantitation Correlates with Targeted Proteomic QuantitationAnna Vildhede, Chuong Nguyen, Brian K. Erickson, Ryan C. Kunz, Richard Jones, Emi Kimoto, Francis Bourbonais, A. David Rodrigues and Manthena V.S. VarmaDrug Metabolism and Disposition May 2018, 46 (5) 692-696; DOI: https://doi.org/10.1124/dmd.117.079285
Villeneuve, Lyne
- You have accessPost-transcriptional Regulation of UGT2B10 Hepatic Expression and Activity by Alternative SplicingAdrien Labriet, Eric P. Allain, Michèle Rouleau, Yannick Audet-Delage, Lyne Villeneuve and Chantal GuillemetteDrug Metabolism and Disposition May 2018, 46 (5) 514-524; DOI: https://doi.org/10.1124/dmd.117.079921
Volak, Laurie P.
- You have accessIntravital Multiphoton Microscopy with Fluorescent Bile Salts in Rats as an In Vivo Biomarker for Hepatobiliary Transport InhibitionJennifer Ryan, Ryan E. Morgan, Yuan Chen, Laurie P. Volak, Robert T. Dunn and Kenneth W. DunnDrug Metabolism and Disposition May 2018, 46 (5) 704-718; DOI: https://doi.org/10.1124/dmd.117.079277
W
Wada, Yasuhiro
- Open AccessA Clinical Quantitative Evaluation of Hepatobiliary Transport of [11C]Dehydropravastatin in Humans Using Positron Emission TomographyKen-ichi Kaneko, Masaaki Tanaka, Akira Ishii, Yumiko Katayama, Takayoshi Nakaoka, Satsuki Irie, Hideki Kawahata, Takashi Yamanaga, Yasuhiro Wada, Takeshi Miyake, Kota Toshimoto, Kazuya Maeda, Yilong Cui, Masaru Enomoto, Etsushi Kawamura, Norifumi Kawada, Joji Kawabe, Susumu Shiomi, Hiroyuki Kusuhara, Yuichi Sugiyama and Yasuyoshi WatanabeDrug Metabolism and Disposition May 2018, 46 (5) 719-728; DOI: https://doi.org/10.1124/dmd.118.080408
Walker, Gregory S.
- You have accessBiosynthesis and Identification of Metabolites of Maraviroc and Their Use in Experiments to Delineate the Relative Contributions of Cytochrome P4503A4 versus 3A5Elaine Tseng, Gwendolyn D. Fate, Gregory S. Walker, Theunis C. Goosen and R. Scott ObachDrug Metabolism and Disposition May 2018, 46 (5) 493-502; DOI: https://doi.org/10.1124/dmd.117.079855
Wang, Changsuo
- You have accessGeneration and Characterization of a CYP2C11-Null Rat Model by Using the CRISPR/Cas9 MethodYuan Wei, Li Yang, Xiaoyan Zhang, Danjuan Sui, Changsuo Wang, Kai Wang, Mangting Shan, Dayong Guo and Hongyu WangDrug Metabolism and Disposition May 2018, 46 (5) 525-531; DOI: https://doi.org/10.1124/dmd.117.078444
Wang, Guangji
- You have accessA Promising Microtubule Inhibitor Deoxypodophyllotoxin Exhibits Better Efficacy to Multidrug-Resistant Breast Cancer than Paclitaxel via Avoiding Efflux TransportXiaojie Zang, Guangji Wang, Qingyun Cai, Xiao Zheng, Jingwei Zhang, Qianying Chen, Baojin Wu, Xiong Zhu, Haiping Hao and Fang ZhouDrug Metabolism and Disposition May 2018, 46 (5) 542-551; DOI: https://doi.org/10.1124/dmd.117.079442
Wang, Hongyu
- You have accessGeneration and Characterization of a CYP2C11-Null Rat Model by Using the CRISPR/Cas9 MethodYuan Wei, Li Yang, Xiaoyan Zhang, Danjuan Sui, Changsuo Wang, Kai Wang, Mangting Shan, Dayong Guo and Hongyu WangDrug Metabolism and Disposition May 2018, 46 (5) 525-531; DOI: https://doi.org/10.1124/dmd.117.078444
Wang, Joanne
- You have accessDrug Transporters in Xenobiotic Disposition and Pharmacokinetic PredictionQingcheng Mao, Yurong Lai and Joanne WangDrug Metabolism and Disposition May 2018, 46 (5) 561-566; DOI: https://doi.org/10.1124/dmd.118.081356
Wang, Kai
- You have accessGeneration and Characterization of a CYP2C11-Null Rat Model by Using the CRISPR/Cas9 MethodYuan Wei, Li Yang, Xiaoyan Zhang, Danjuan Sui, Changsuo Wang, Kai Wang, Mangting Shan, Dayong Guo and Hongyu WangDrug Metabolism and Disposition May 2018, 46 (5) 525-531; DOI: https://doi.org/10.1124/dmd.117.078444
Wang, Lixue
- You have accessIdentification of a NFκB Inhibition Site on the Proximal Promoter Region of Human Organic Anion Transporting Polypeptide 1A2 Coding Gene SLCO1A2Zhaojian Xiang, Weike Li, Lixue Wang, Jicai Yi, Kaiwen Chen and Mei HongDrug Metabolism and Disposition May 2018, 46 (5) 643-651; DOI: https://doi.org/10.1124/dmd.117.078832
Watanabe, Michitoshi
- You have accessLiver Zonation Index of Drug Transporter and Metabolizing Enzyme Protein Expressions in Mouse Liver AcinusMasanori Tachikawa, Yuna Sumiyoshiya, Daisuke Saigusa, Kazunari Sasaki, Michitoshi Watanabe, Yasuo Uchida and Tetsuya TerasakiDrug Metabolism and Disposition May 2018, 46 (5) 610-618; DOI: https://doi.org/10.1124/dmd.117.079244
Watanabe, Yasuyoshi
- Open AccessA Clinical Quantitative Evaluation of Hepatobiliary Transport of [11C]Dehydropravastatin in Humans Using Positron Emission TomographyKen-ichi Kaneko, Masaaki Tanaka, Akira Ishii, Yumiko Katayama, Takayoshi Nakaoka, Satsuki Irie, Hideki Kawahata, Takashi Yamanaga, Yasuhiro Wada, Takeshi Miyake, Kota Toshimoto, Kazuya Maeda, Yilong Cui, Masaru Enomoto, Etsushi Kawamura, Norifumi Kawada, Joji Kawabe, Susumu Shiomi, Hiroyuki Kusuhara, Yuichi Sugiyama and Yasuyoshi WatanabeDrug Metabolism and Disposition May 2018, 46 (5) 719-728; DOI: https://doi.org/10.1124/dmd.118.080408
Wei, Yuan
- You have accessGeneration and Characterization of a CYP2C11-Null Rat Model by Using the CRISPR/Cas9 MethodYuan Wei, Li Yang, Xiaoyan Zhang, Danjuan Sui, Changsuo Wang, Kai Wang, Mangting Shan, Dayong Guo and Hongyu WangDrug Metabolism and Disposition May 2018, 46 (5) 525-531; DOI: https://doi.org/10.1124/dmd.117.078444
Weinberger, Barry I.
- You have accessInterindividual Regulation of the Breast Cancer Resistance Protein/ABCG2 Transporter in Term Human PlacentasKristin M. Bircsak, Jamie E. Moscovitz, Xia Wen, Faith Archer, Poi Yu Sofia Yuen, Moiz Mohammed, Naureen Memon, Barry I. Weinberger, Laura M. Saba, Anna M. Vetrano and Lauren M. AleksunesDrug Metabolism and Disposition May 2018, 46 (5) 619-627; DOI: https://doi.org/10.1124/dmd.117.079228
Wen, Xia
- You have accessInterindividual Regulation of the Breast Cancer Resistance Protein/ABCG2 Transporter in Term Human PlacentasKristin M. Bircsak, Jamie E. Moscovitz, Xia Wen, Faith Archer, Poi Yu Sofia Yuen, Moiz Mohammed, Naureen Memon, Barry I. Weinberger, Laura M. Saba, Anna M. Vetrano and Lauren M. AleksunesDrug Metabolism and Disposition May 2018, 46 (5) 619-627; DOI: https://doi.org/10.1124/dmd.117.079228
Wilmer, Martijn J.
- Open AccessExpression of Organic Anion Transporter 1 or 3 in Human Kidney Proximal Tubule Cells Reduces Cisplatin SensitivityTom T. G. Nieskens, Janny G. P. Peters, Dina Dabaghie, Daphne Korte, Katja Jansen, Alexander H. Van Asbeck, Neslihan N. Tavraz, Thomas Friedrich, Frans G. M. Russel, Rosalinde Masereeuw and Martijn J. WilmerDrug Metabolism and Disposition May 2018, 46 (5) 592-599; DOI: https://doi.org/10.1124/dmd.117.079384
Wilson, David M.
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Wu, Baojin
- You have accessA Promising Microtubule Inhibitor Deoxypodophyllotoxin Exhibits Better Efficacy to Multidrug-Resistant Breast Cancer than Paclitaxel via Avoiding Efflux TransportXiaojie Zang, Guangji Wang, Qingyun Cai, Xiao Zheng, Jingwei Zhang, Qianying Chen, Baojin Wu, Xiong Zhu, Haiping Hao and Fang ZhouDrug Metabolism and Disposition May 2018, 46 (5) 542-551; DOI: https://doi.org/10.1124/dmd.117.079442
X
Xiang, Zhaojian
- You have accessIdentification of a NFκB Inhibition Site on the Proximal Promoter Region of Human Organic Anion Transporting Polypeptide 1A2 Coding Gene SLCO1A2Zhaojian Xiang, Weike Li, Lixue Wang, Jicai Yi, Kaiwen Chen and Mei HongDrug Metabolism and Disposition May 2018, 46 (5) 643-651; DOI: https://doi.org/10.1124/dmd.117.078832
Y
Yamanaga, Takashi
- Open AccessA Clinical Quantitative Evaluation of Hepatobiliary Transport of [11C]Dehydropravastatin in Humans Using Positron Emission TomographyKen-ichi Kaneko, Masaaki Tanaka, Akira Ishii, Yumiko Katayama, Takayoshi Nakaoka, Satsuki Irie, Hideki Kawahata, Takashi Yamanaga, Yasuhiro Wada, Takeshi Miyake, Kota Toshimoto, Kazuya Maeda, Yilong Cui, Masaru Enomoto, Etsushi Kawamura, Norifumi Kawada, Joji Kawabe, Susumu Shiomi, Hiroyuki Kusuhara, Yuichi Sugiyama and Yasuyoshi WatanabeDrug Metabolism and Disposition May 2018, 46 (5) 719-728; DOI: https://doi.org/10.1124/dmd.118.080408
Yang, Chun
- You have accessMetabolism and Disposition of Verinurad, a Uric Acid Reabsorption Inhibitor, in HumansCaroline A. Lee, Chun Yang, Vishal Shah, Zancong Shen, David M. Wilson, Traci M. Ostertag, Jean-Luc Girardet, Jesse Hall and Michael GillenDrug Metabolism and Disposition May 2018, 46 (5) 532-541; DOI: https://doi.org/10.1124/dmd.117.078220
Yang, Li
- You have accessGeneration and Characterization of a CYP2C11-Null Rat Model by Using the CRISPR/Cas9 MethodYuan Wei, Li Yang, Xiaoyan Zhang, Danjuan Sui, Changsuo Wang, Kai Wang, Mangting Shan, Dayong Guo and Hongyu WangDrug Metabolism and Disposition May 2018, 46 (5) 525-531; DOI: https://doi.org/10.1124/dmd.117.078444
Yi, Jicai
- You have accessIdentification of a NFκB Inhibition Site on the Proximal Promoter Region of Human Organic Anion Transporting Polypeptide 1A2 Coding Gene SLCO1A2Zhaojian Xiang, Weike Li, Lixue Wang, Jicai Yi, Kaiwen Chen and Mei HongDrug Metabolism and Disposition May 2018, 46 (5) 643-651; DOI: https://doi.org/10.1124/dmd.117.078832
Yoshikado, Takashi
- You have accessEvaluation of Alteration in Hepatic and Intestinal BCRP Function In Vivo from ABCG2 c.421C>A Polymorphism Based on PBPK Analysis of RosuvastatinAzusa Futatsugi, Kota Toshimoto, Takashi Yoshikado, Yuichi Sugiyama and Yukio KatoDrug Metabolism and Disposition May 2018, 46 (5) 749-757; DOI: https://doi.org/10.1124/dmd.117.078816
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Yuen, Poi Yu Sofia
- You have accessInterindividual Regulation of the Breast Cancer Resistance Protein/ABCG2 Transporter in Term Human PlacentasKristin M. Bircsak, Jamie E. Moscovitz, Xia Wen, Faith Archer, Poi Yu Sofia Yuen, Moiz Mohammed, Naureen Memon, Barry I. Weinberger, Laura M. Saba, Anna M. Vetrano and Lauren M. AleksunesDrug Metabolism and Disposition May 2018, 46 (5) 619-627; DOI: https://doi.org/10.1124/dmd.117.079228
Z
Zang, Xiaojie
- You have accessA Promising Microtubule Inhibitor Deoxypodophyllotoxin Exhibits Better Efficacy to Multidrug-Resistant Breast Cancer than Paclitaxel via Avoiding Efflux TransportXiaojie Zang, Guangji Wang, Qingyun Cai, Xiao Zheng, Jingwei Zhang, Qianying Chen, Baojin Wu, Xiong Zhu, Haiping Hao and Fang ZhouDrug Metabolism and Disposition May 2018, 46 (5) 542-551; DOI: https://doi.org/10.1124/dmd.117.079442
Zhang, Jingwei
- You have accessA Promising Microtubule Inhibitor Deoxypodophyllotoxin Exhibits Better Efficacy to Multidrug-Resistant Breast Cancer than Paclitaxel via Avoiding Efflux TransportXiaojie Zang, Guangji Wang, Qingyun Cai, Xiao Zheng, Jingwei Zhang, Qianying Chen, Baojin Wu, Xiong Zhu, Haiping Hao and Fang ZhouDrug Metabolism and Disposition May 2018, 46 (5) 542-551; DOI: https://doi.org/10.1124/dmd.117.079442
Zhang, Xiaoyan
- You have accessGeneration and Characterization of a CYP2C11-Null Rat Model by Using the CRISPR/Cas9 MethodYuan Wei, Li Yang, Xiaoyan Zhang, Danjuan Sui, Changsuo Wang, Kai Wang, Mangting Shan, Dayong Guo and Hongyu WangDrug Metabolism and Disposition May 2018, 46 (5) 525-531; DOI: https://doi.org/10.1124/dmd.117.078444
Zheng, Xiao
- You have accessA Promising Microtubule Inhibitor Deoxypodophyllotoxin Exhibits Better Efficacy to Multidrug-Resistant Breast Cancer than Paclitaxel via Avoiding Efflux TransportXiaojie Zang, Guangji Wang, Qingyun Cai, Xiao Zheng, Jingwei Zhang, Qianying Chen, Baojin Wu, Xiong Zhu, Haiping Hao and Fang ZhouDrug Metabolism and Disposition May 2018, 46 (5) 542-551; DOI: https://doi.org/10.1124/dmd.117.079442
Zhou, Fang
- You have accessA Promising Microtubule Inhibitor Deoxypodophyllotoxin Exhibits Better Efficacy to Multidrug-Resistant Breast Cancer than Paclitaxel via Avoiding Efflux TransportXiaojie Zang, Guangji Wang, Qingyun Cai, Xiao Zheng, Jingwei Zhang, Qianying Chen, Baojin Wu, Xiong Zhu, Haiping Hao and Fang ZhouDrug Metabolism and Disposition May 2018, 46 (5) 542-551; DOI: https://doi.org/10.1124/dmd.117.079442
Zhu, Catherine
- You have accessApixaban and Rosuvastatin Pharmacokinetics in Nonalcoholic Fatty Liver DiseaseRommel G. Tirona, Zahra Kassam, Ruth Strapp, Mala Ramu, Catherine Zhu, Melissa Liu, Ute I. Schwarz, Richard B. Kim, Bandar Al-Judaibi and Melanie D. BeatonDrug Metabolism and Disposition May 2018, 46 (5) 485-492; DOI: https://doi.org/10.1124/dmd.117.079624
Zhu, Xiong
- You have accessA Promising Microtubule Inhibitor Deoxypodophyllotoxin Exhibits Better Efficacy to Multidrug-Resistant Breast Cancer than Paclitaxel via Avoiding Efflux TransportXiaojie Zang, Guangji Wang, Qingyun Cai, Xiao Zheng, Jingwei Zhang, Qianying Chen, Baojin Wu, Xiong Zhu, Haiping Hao and Fang ZhouDrug Metabolism and Disposition May 2018, 46 (5) 542-551; DOI: https://doi.org/10.1124/dmd.117.079442
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