Research ArticleArticle
Regional Proteomic Quantification of Clinically Relevant Non-Cytochrome P450 Enzymes along the Human Small Intestine
Haeyoung Zhang, Chris Wolford, Abdul Basit, Albert P. Li, Peter W. Fan, Bernard P. Murray, Ryan H. Takahashi, S. Cyrus Khojasteh, Bill J. Smith, Kenneth E. Thummel and Bhagwat Prasad
Drug Metabolism and Disposition July 2020, 48 (7) 528-536; DOI: https://doi.org/10.1124/dmd.120.090738
Haeyoung Zhang
Department of Pharmaceutics, University of Washington, Seattle, Washington (H.Z., C.W., A.B., K.E.T., B.P.); Department of Pharmaceutical Sciences, Washington State University, Spokane, Washington (A.B., B.P.); In Vitro ADMET Laboratories Inc., Columbia, Maryland (A.P.L.); Department of Pharmacokinetics, Pharmacodynamics and Drug Metabolism, Merck & Co., Inc., Boston, Massachusetts (P.W.F.); Genentech Inc., South San Francisco, California (R.H.T., S.C.K.); and Drug Metabolism Department, Gilead Sciences Inc., Foster City, California (B.J.S., B.P.M.)
Chris Wolford
Department of Pharmaceutics, University of Washington, Seattle, Washington (H.Z., C.W., A.B., K.E.T., B.P.); Department of Pharmaceutical Sciences, Washington State University, Spokane, Washington (A.B., B.P.); In Vitro ADMET Laboratories Inc., Columbia, Maryland (A.P.L.); Department of Pharmacokinetics, Pharmacodynamics and Drug Metabolism, Merck & Co., Inc., Boston, Massachusetts (P.W.F.); Genentech Inc., South San Francisco, California (R.H.T., S.C.K.); and Drug Metabolism Department, Gilead Sciences Inc., Foster City, California (B.J.S., B.P.M.)
Abdul Basit
Department of Pharmaceutics, University of Washington, Seattle, Washington (H.Z., C.W., A.B., K.E.T., B.P.); Department of Pharmaceutical Sciences, Washington State University, Spokane, Washington (A.B., B.P.); In Vitro ADMET Laboratories Inc., Columbia, Maryland (A.P.L.); Department of Pharmacokinetics, Pharmacodynamics and Drug Metabolism, Merck & Co., Inc., Boston, Massachusetts (P.W.F.); Genentech Inc., South San Francisco, California (R.H.T., S.C.K.); and Drug Metabolism Department, Gilead Sciences Inc., Foster City, California (B.J.S., B.P.M.)
Albert P. Li
Department of Pharmaceutics, University of Washington, Seattle, Washington (H.Z., C.W., A.B., K.E.T., B.P.); Department of Pharmaceutical Sciences, Washington State University, Spokane, Washington (A.B., B.P.); In Vitro ADMET Laboratories Inc., Columbia, Maryland (A.P.L.); Department of Pharmacokinetics, Pharmacodynamics and Drug Metabolism, Merck & Co., Inc., Boston, Massachusetts (P.W.F.); Genentech Inc., South San Francisco, California (R.H.T., S.C.K.); and Drug Metabolism Department, Gilead Sciences Inc., Foster City, California (B.J.S., B.P.M.)
Peter W. Fan
Department of Pharmaceutics, University of Washington, Seattle, Washington (H.Z., C.W., A.B., K.E.T., B.P.); Department of Pharmaceutical Sciences, Washington State University, Spokane, Washington (A.B., B.P.); In Vitro ADMET Laboratories Inc., Columbia, Maryland (A.P.L.); Department of Pharmacokinetics, Pharmacodynamics and Drug Metabolism, Merck & Co., Inc., Boston, Massachusetts (P.W.F.); Genentech Inc., South San Francisco, California (R.H.T., S.C.K.); and Drug Metabolism Department, Gilead Sciences Inc., Foster City, California (B.J.S., B.P.M.)
Bernard P. Murray
Department of Pharmaceutics, University of Washington, Seattle, Washington (H.Z., C.W., A.B., K.E.T., B.P.); Department of Pharmaceutical Sciences, Washington State University, Spokane, Washington (A.B., B.P.); In Vitro ADMET Laboratories Inc., Columbia, Maryland (A.P.L.); Department of Pharmacokinetics, Pharmacodynamics and Drug Metabolism, Merck & Co., Inc., Boston, Massachusetts (P.W.F.); Genentech Inc., South San Francisco, California (R.H.T., S.C.K.); and Drug Metabolism Department, Gilead Sciences Inc., Foster City, California (B.J.S., B.P.M.)
Ryan H. Takahashi
Department of Pharmaceutics, University of Washington, Seattle, Washington (H.Z., C.W., A.B., K.E.T., B.P.); Department of Pharmaceutical Sciences, Washington State University, Spokane, Washington (A.B., B.P.); In Vitro ADMET Laboratories Inc., Columbia, Maryland (A.P.L.); Department of Pharmacokinetics, Pharmacodynamics and Drug Metabolism, Merck & Co., Inc., Boston, Massachusetts (P.W.F.); Genentech Inc., South San Francisco, California (R.H.T., S.C.K.); and Drug Metabolism Department, Gilead Sciences Inc., Foster City, California (B.J.S., B.P.M.)
S. Cyrus Khojasteh
Department of Pharmaceutics, University of Washington, Seattle, Washington (H.Z., C.W., A.B., K.E.T., B.P.); Department of Pharmaceutical Sciences, Washington State University, Spokane, Washington (A.B., B.P.); In Vitro ADMET Laboratories Inc., Columbia, Maryland (A.P.L.); Department of Pharmacokinetics, Pharmacodynamics and Drug Metabolism, Merck & Co., Inc., Boston, Massachusetts (P.W.F.); Genentech Inc., South San Francisco, California (R.H.T., S.C.K.); and Drug Metabolism Department, Gilead Sciences Inc., Foster City, California (B.J.S., B.P.M.)
Bill J. Smith
Department of Pharmaceutics, University of Washington, Seattle, Washington (H.Z., C.W., A.B., K.E.T., B.P.); Department of Pharmaceutical Sciences, Washington State University, Spokane, Washington (A.B., B.P.); In Vitro ADMET Laboratories Inc., Columbia, Maryland (A.P.L.); Department of Pharmacokinetics, Pharmacodynamics and Drug Metabolism, Merck & Co., Inc., Boston, Massachusetts (P.W.F.); Genentech Inc., South San Francisco, California (R.H.T., S.C.K.); and Drug Metabolism Department, Gilead Sciences Inc., Foster City, California (B.J.S., B.P.M.)
Kenneth E. Thummel
Department of Pharmaceutics, University of Washington, Seattle, Washington (H.Z., C.W., A.B., K.E.T., B.P.); Department of Pharmaceutical Sciences, Washington State University, Spokane, Washington (A.B., B.P.); In Vitro ADMET Laboratories Inc., Columbia, Maryland (A.P.L.); Department of Pharmacokinetics, Pharmacodynamics and Drug Metabolism, Merck & Co., Inc., Boston, Massachusetts (P.W.F.); Genentech Inc., South San Francisco, California (R.H.T., S.C.K.); and Drug Metabolism Department, Gilead Sciences Inc., Foster City, California (B.J.S., B.P.M.)
Bhagwat Prasad
Department of Pharmaceutics, University of Washington, Seattle, Washington (H.Z., C.W., A.B., K.E.T., B.P.); Department of Pharmaceutical Sciences, Washington State University, Spokane, Washington (A.B., B.P.); In Vitro ADMET Laboratories Inc., Columbia, Maryland (A.P.L.); Department of Pharmacokinetics, Pharmacodynamics and Drug Metabolism, Merck & Co., Inc., Boston, Massachusetts (P.W.F.); Genentech Inc., South San Francisco, California (R.H.T., S.C.K.); and Drug Metabolism Department, Gilead Sciences Inc., Foster City, California (B.J.S., B.P.M.)
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Research ArticleArticle
Non–Cytochrome P450 Enzyme Quantification in Small Intestine
Haeyoung Zhang, Chris Wolford, Abdul Basit, Albert P. Li, Peter W. Fan, Bernard P. Murray, Ryan H. Takahashi, S. Cyrus Khojasteh, Bill J. Smith, Kenneth E. Thummel and Bhagwat Prasad
Drug Metabolism and Disposition July 1, 2020, 48 (7) 528-536; DOI: https://doi.org/10.1124/dmd.120.090738
Research ArticleArticle
Non–Cytochrome P450 Enzyme Quantification in Small Intestine
Haeyoung Zhang, Chris Wolford, Abdul Basit, Albert P. Li, Peter W. Fan, Bernard P. Murray, Ryan H. Takahashi, S. Cyrus Khojasteh, Bill J. Smith, Kenneth E. Thummel and Bhagwat Prasad
Drug Metabolism and Disposition July 1, 2020, 48 (7) 528-536; DOI: https://doi.org/10.1124/dmd.120.090738
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