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Research ArticleArticle

In vitro interactions of epacadostat and its major metabolites with human efflux and uptake transporters: Implications for pharmacokinetics and drug interactions

Qiang Zhang, Yan Zhang, Jason Boer, Jack G Shi, Peidi Hu, Sharon Diamond and Swamy Yeleswaram
Drug Metabolism and Disposition March 10, 2017, dmd.116.074609; DOI: https://doi.org/10.1124/dmd.116.074609
Qiang Zhang
Incyte Corporation;
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  • For correspondence: qizhang@incyte.com
Yan Zhang
Incyte Corporation;
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Jason Boer
Incyte Corporation;
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Jack G Shi
Ultragenyx Pharmaceutical Company
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Peidi Hu
Incyte Corporation;
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Sharon Diamond
Incyte Corporation;
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Swamy Yeleswaram
Incyte Corporation;
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Drug Metabolism and Disposition: 46 (5)
Drug Metabolism and Disposition
Vol. 46, Issue 5
1 May 2018
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Research ArticleArticle

In vitro interactions of epacadostat and its major metabolites with human efflux and uptake transporters: Implications for pharmacokinetics and drug interactions

Qiang Zhang, Yan Zhang, Jason Boer, Jack G Shi, Peidi Hu, Sharon Diamond and Swamy Yeleswaram
Drug Metabolism and Disposition March 10, 2017, dmd.116.074609; DOI: https://doi.org/10.1124/dmd.116.074609

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Research ArticleArticle

In vitro interactions of epacadostat and its major metabolites with human efflux and uptake transporters: Implications for pharmacokinetics and drug interactions

Qiang Zhang, Yan Zhang, Jason Boer, Jack G Shi, Peidi Hu, Sharon Diamond and Swamy Yeleswaram
Drug Metabolism and Disposition March 10, 2017, dmd.116.074609; DOI: https://doi.org/10.1124/dmd.116.074609
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