Research ArticleArticle
The phenomenon of "albumin-mediated" hepatic uptake of organic anion transport polypeptide substrates: Prediction of the in vivo uptake clearance from the in vitro uptake by isolated hepatocytes using a "facilitated-dissociation" model
SEIJI MIYAUCHI, Masayuki Masuda, Soo-Jin Kim, Yuudai Tanaka, Kyeong Ryoon Lee, Shouko Iwakado, Momoko Nemoto, Shotaro Sasaki, Kazumi Shimono, Yoshio Tanaka and Yuichi Sugiyama
Drug Metabolism and Disposition January 3, 2018, dmd.117.077115; DOI: https://doi.org/10.1124/dmd.117.077115
SEIJI MIYAUCHI
1 Toho University Faculty of Pharmaceutical Sciences;
Masayuki Masuda
1 Toho University Faculty of Pharmaceutical Sciences;
Soo-Jin Kim
2 RIKEN, RIKEN Innovation Center
Yuudai Tanaka
1 Toho University Faculty of Pharmaceutical Sciences;
Kyeong Ryoon Lee
2 RIKEN, RIKEN Innovation Center
Shouko Iwakado
1 Toho University Faculty of Pharmaceutical Sciences;
Momoko Nemoto
1 Toho University Faculty of Pharmaceutical Sciences;
Shotaro Sasaki
1 Toho University Faculty of Pharmaceutical Sciences;
Kazumi Shimono
1 Toho University Faculty of Pharmaceutical Sciences;
Yoshio Tanaka
1 Toho University Faculty of Pharmaceutical Sciences;
Yuichi Sugiyama
2 RIKEN, RIKEN Innovation Center
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Research ArticleArticle
The phenomenon of "albumin-mediated" hepatic uptake of organic anion transport polypeptide substrates: Prediction of the in vivo uptake clearance from the in vitro uptake by isolated hepatocytes using a "facilitated-dissociation" model
SEIJI MIYAUCHI, Masayuki Masuda, Soo-Jin Kim, Yuudai Tanaka, Kyeong Ryoon Lee, Shouko Iwakado, Momoko Nemoto, Shotaro Sasaki, Kazumi Shimono, Yoshio Tanaka and Yuichi Sugiyama
Drug Metabolism and Disposition January 3, 2018, dmd.117.077115; DOI: https://doi.org/10.1124/dmd.117.077115
Research ArticleArticle
The phenomenon of "albumin-mediated" hepatic uptake of organic anion transport polypeptide substrates: Prediction of the in vivo uptake clearance from the in vitro uptake by isolated hepatocytes using a "facilitated-dissociation" model
SEIJI MIYAUCHI, Masayuki Masuda, Soo-Jin Kim, Yuudai Tanaka, Kyeong Ryoon Lee, Shouko Iwakado, Momoko Nemoto, Shotaro Sasaki, Kazumi Shimono, Yoshio Tanaka and Yuichi Sugiyama
Drug Metabolism and Disposition January 3, 2018, dmd.117.077115; DOI: https://doi.org/10.1124/dmd.117.077115
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