Research ArticleArticle
Structure guided in-vitro to in-vivo pharmacokinetic optimization of propargyl-linked antifolates
Michael N Lombardo, Narendran G-Dayanandan, Santosh Keshipeddy, Wangda Zhou, Debjani Si, Stephanie M Reeve, Jeremy Alverson, Patrick Barney, Larissa Walker, John Hoody, Nigel Priestley, R. Scott Obach and Dennis L Wright
Drug Metabolism and Disposition June 14, 2019, dmd.119.086504; DOI: https://doi.org/10.1124/dmd.119.086504
Michael N Lombardo
1 University of Connecticut;
Narendran G-Dayanandan
1 University of Connecticut;
Santosh Keshipeddy
1 University of Connecticut;
Wangda Zhou
1 University of Connecticut;
Debjani Si
1 University of Connecticut;
Stephanie M Reeve
1 University of Connecticut;
Jeremy Alverson
2 University of Montana;
Patrick Barney
2 University of Montana;
Larissa Walker
2 University of Montana;
John Hoody
2 University of Montana;
Nigel Priestley
2 University of Montana;
R. Scott Obach
3 Pfizer
Dennis L Wright
1 University of Connecticut;
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Supplemental methods, 1 table, 16 figures.
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Research ArticleArticle
Structure guided in-vitro to in-vivo pharmacokinetic optimization of propargyl-linked antifolates
Michael N Lombardo, Narendran G-Dayanandan, Santosh Keshipeddy, Wangda Zhou, Debjani Si, Stephanie M Reeve, Jeremy Alverson, Patrick Barney, Larissa Walker, John Hoody, Nigel Priestley, R. Scott Obach and Dennis L Wright
Drug Metabolism and Disposition June 14, 2019, dmd.119.086504; DOI: https://doi.org/10.1124/dmd.119.086504
Research ArticleArticle
Structure guided in-vitro to in-vivo pharmacokinetic optimization of propargyl-linked antifolates
Michael N Lombardo, Narendran G-Dayanandan, Santosh Keshipeddy, Wangda Zhou, Debjani Si, Stephanie M Reeve, Jeremy Alverson, Patrick Barney, Larissa Walker, John Hoody, Nigel Priestley, R. Scott Obach and Dennis L Wright
Drug Metabolism and Disposition June 14, 2019, dmd.119.086504; DOI: https://doi.org/10.1124/dmd.119.086504
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