DMD Bio-Rad Microplate Reader

Home Help [Feedback] [For Subscribers] [Archive] [Search] [Contents]
QUICK SEARCH:   [advanced]
Author:
Keyword(s):
Year:  Vol:  Page: 


Receive this page by email each issue: [Sign up for eTOCs]

Cover Caption
Other Issues:
May 2004; 32 (5)   [Index by Author]  [Cover Caption]
       Articles
       Short Communications
Find articles in this issue containing these words:
[Search ALL Issues]


To see an article, click its [Full Text] link. To review many abstracts, check the boxes to the left of the titles you want, and click the 'Get All Checked Abstract(s)' button. To see one abstract at a time, click its [Abstract] link.

Articles:

Yasuna Kobayashi, Naomi Ohshiro, Ayumi Tsuchiya, Noriko Kohyama, Masayuki Ohbayashi, and Toshinori Yamamoto
RENAL TRANSPORT OF ORGANIC COMPOUNDS MEDIATED BY MOUSE ORGANIC ANION TRANSPORTER 3 (MOAT3): FURTHER SUBSTRATE SPECIFICITY OF MOAT3
Drug Metab Dispos 2004 32: 479-483. [Abstract] [Full Text] [PDF]  

Mia Sandberg, Inger Johansson, Magnus Christensen, Anders Rane, and Erik Eliasson
THE IMPACT OF CYP2C9 GENETICS AND ORAL CONTRACEPTIVES ON CYTOCHROME P450 2C9 PHENOTYPE
Drug Metab Dispos 2004 32: 484-489. [Abstract] [Full Text] [PDF]  

Julianne L. Holleran, Julien Fourcade, Merrill J. Egorin, Julie L. Eiseman, Robert A. Parise, Steven M. Musser, Kevin D. White, Joseph M. Covey, Gerald L. Forrest, and Su-Shu Pan
IN VITRO METABOLISM OF THE PHOSPHATIDYLINOSITOL 3-KINASE INHIBITOR, WORTMANNIN, BY CARBONYL REDUCTASE
Drug Metab Dispos 2004 32: 490-496. [Abstract] [Full Text] [PDF]  

Mime Nagai, Allan H. Conney, and Bao Ting Zhu
STRONG INHIBITORY EFFECTS OF COMMON TEA CATECHINS AND BIOFLAVONOIDS ON THE O-METHYLATION OF CATECHOL ESTROGENS CATALYZED BY HUMAN LIVER CYTOSOLIC CATECHOL-O-METHYLTRANSFERASE
Drug Metab Dispos 2004 32: 497-504. [Abstract] [Full Text] [PDF]  

Sonal P. Sanghani, Sara K. Quinney, Tyler B. Fredenburg, Wilhelmina I. Davis, Daryl J. Murry, and William F. Bosron
HYDROLYSIS OF IRINOTECAN AND ITS OXIDATIVE METABOLITES, 7-ETHYL-10-[4-N-(5-AMINOPENTANOIC ACID)-1-PIPERIDINO] CARBONYLOXYCAMPTOTHECIN AND 7-ETHYL-10-[4-(1-PIPERIDINO)-1-AMINO]-CARBONYLOXYCAMPTOTHECIN, BY HUMAN CARBOXYLESTERASES CES1A1, CES2, AND A NEWLY EXPRESSED CARBOXYLESTERASE ISOENZYME, CES3
Drug Metab Dispos 2004 32: 505-511. [Abstract] [Full Text] [PDF]  

Bernard J. Komoroski, Shimin Zhang, Hongbo Cai, J. Matthew Hutzler, Reginald Frye, Timothy S. Tracy, Stephen C. Strom, Thomas Lehmann, Catharina Y. W. Ang, Yan Yan Cui, and Raman Venkataramanan
INDUCTION AND INHIBITION OF CYTOCHROMES P450 BY THE ST. JOHN'S WORT CONSTITUENT HYPERFORIN IN HUMAN HEPATOCYTE CULTURES
Drug Metab Dispos 2004 32: 512-518. [Abstract] [Full Text] [PDF]  

Naoki Ishiguro, Takashi Nozawa, Akiko Tsujihata, Asami Saito, Wataru Kishimoto, Kazutoshi Yokoyama, Takafumi Yotsumoto, Kenji Sakai, Takashi Igarashi, and Ikumi Tamai
INFLUX AND EFFLUX TRANSPORT OF H1-ANTAGONIST EPINASTINE ACROSS THE BLOOD-BRAIN BARRIER
Drug Metab Dispos 2004 32: 519-524. [Abstract] [Full Text] [PDF]  

Vincent Bombail, Kevin Taylor, G. Gordon Gibson, and Nick Plant
ROLE OF Sp1, C/EBP{alpha}, HNF3, AND PXR IN THE BASAL- AND XENOBIOTIC-MEDIATED REGULATION OF THE CYP3A4 GENE
Drug Metab Dispos 2004 32: 525-535. [Abstract] [Full Text] [PDF]  

G. Virkel, A. Lifschitz, J. Sallovitz, A. Pis, and C. Lanusse
COMPARATIVE HEPATIC AND EXTRAHEPATIC ENANTIOSELECTIVE SULFOXIDATION OF ALBENDAZOLE AND FENBENDAZOLE IN SHEEP AND CATTLE
Drug Metab Dispos 2004 32: 536-544. [Abstract] [Full Text] [PDF]  

Donglu Zhang, Weiping Zhao, Vikram A. Roongta, James G. Mitroka, Lewis J. Klunk, and Mingshe Zhu
AMIDE N-GLUCURONIDATION OF MAXIPOST CATALYZED BY UDP-GLUCURONOSYLTRANSFERASE 2B7 IN HUMANS
Drug Metab Dispos 2004 32: 545-551. [Abstract] [Full Text] [PDF]  

Sarah J. Griffin and J. Brian Houston
COMPARISON OF FRESH AND CRYOPRESERVED RAT HEPATOCYTE SUSPENSIONS FOR THE PREDICTION OF IN VITRO INTRINSIC CLEARANCE
Drug Metab Dispos 2004 32: 552-558. [Abstract] [Full Text] [PDF]  

Jonathan J. Sheng, Atmaja Saxena, and Michael W. Duffel
INFLUENCE OF PHENYLALANINES 77 AND 138 ON THE STEREOSPECIFICITY OF ARYL SULFOTRANSFERASE IV
Drug Metab Dispos 2004 32: 559-565. [Abstract] [Full Text] [PDF]  

James B. Mangold, Helen Gu, Lolita C. Rodriguez, Johanne Bonner, Janet Dickson, and Christiane Rordorf
PHARMACOKINETICS AND METABOLISM OF LUMIRACOXIB IN HEALTHY MALE SUBJECTS
Drug Metab Dispos 2004 32: 566-571. [Abstract] [Full Text] [PDF]  

Hannah M. Jones, David Hallifax, and J. Brian Houston
QUANTITATIVE PREDICTION OF THE IN VIVO INHIBITION OF DIAZEPAM METABOLISM BY OMEPRAZOLE USING RAT LIVER MICROSOMES AND HEPATOCYTES
Drug Metab Dispos 2004 32: 572-580. [Abstract] [Full Text] [PDF]  

Short Communications:

Bennett Ma, Raju Subramanian, Michael L. Schrag, A. David Rodrigues, and Cuyue Tang
CYTOCHROME P450 2C8 (CYP2C8)-MEDIATED HYDROXYLATION OF AN ENDOTHELIN ETA RECEPTOR ANTAGONIST IN HUMAN LIVER MICROSOMES
Drug Metab Dispos 2004 32: 473-478. [Abstract] [Full Text] [PDF]  

To see an article, click its [Full Text] link. To review many abstracts, check the boxes to the left of the titles you want, and click the 'Get All Checked Abstract(s)' button. To see one abstract at a time, click its [Abstract] link.


Cover Caption:

A molecule of (R)-(--)-1,2,3,4-tetrahydro-1-naphthol [(R)-(--)-THN] (A) is shown docked into the homology model of the active site of AST IV; and the proximity of the side chains of Phe77, Phe138, and Tyr236 to the position of (R)-(--)-THN in A is highlighted (B). See the article by Sheng et al. on page 559 of this issue.



Home Help [Feedback] [For Subscribers] [Archive] [Search] [Contents]
All ASPET Journals Molecular Pharmacology Pharmacological Reviews
The Journal of Pharmacology and Experimental 
Therapeutics Molecular Interventions Drug Metabolism and Disposition

Copyright © 2004 by the American Society for Pharmacology and Experimental Therapeutics.