DMD

Home Help [Feedback] [For Subscribers] [Archive] [Search] [Contents]
QUICK SEARCH:   [advanced]
Author:
Keyword(s):
Year:  Vol:  Page: 


Receive this page by email each issue: [Sign up for eTOCs]

Cover Caption
Other Issues:
April 2005; 33 (4)   [Index by Author]  [Cover Caption]
       Articles
       Commentaries
       Short Communications
Find articles in this issue containing these words:
[Search ALL Issues]


To see an article, click its [Full Text] link. To review many abstracts, check the boxes to the left of the titles you want, and click the 'Get All Checked Abstract(s)' button. To see one abstract at a time, click its [Abstract] link.

Articles:

Xiaochao Ma, Jeffrey R. Idle, Kristopher W. Krausz, and Frank J. Gonzalez
METABOLISM OF MELATONIN BY HUMAN CYTOCHROMES P450
Drug Metab Dispos 2005 33: 489-494. Published online December 22, 2004; 10.1124/dmd.104.002410 [Abstract] [Full Text] [PDF]  

Naoki Ishiguro, Asami Saito, Kazutoshi Yokoyama, Makoto Morikawa, Takashi Igarashi, and Ikumi Tamai
TRANSPORT OF THE DOPAMINE D2 AGONIST PRAMIPEXOLE BY RAT ORGANIC CATION TRANSPORTERS OCT1 AND OCT2 IN KIDNEY
Drug Metab Dispos 2005 33: 495-499. Published online January 7, 2005; 10.1124/dmd.104.002519 [Abstract] [Full Text] [PDF]  

Mingshe Zhu, Weiping Zhao, Humberto Jimenez, Donglu Zhang, Suresh Yeola, Renke Dai, Nimish Vachharajani, and James Mitroka
CYTOCHROME P450 3A-MEDIATED METABOLISM OF BUSPIRONE IN HUMAN LIVER MICROSOMES
Drug Metab Dispos 2005 33: 500-507. Published online January 7, 2005; 10.1124/dmd.104.000836 [Abstract] [Full Text] [PDF]  

Qiang Zhang, Peng Ma, Weiqun Wang, Richard B. Cole, and Guangdi Wang
IN VITRO METABOLISM OF DIARYLPYRAZOLES, A NOVEL GROUP OF CANNABINOID RECEPTOR LIGANDS
Drug Metab Dispos 2005 33: 508-517. Published online December 22, 2004; 10.1124/dmd.104.001974 [Abstract] [Full Text] [PDF]  

Hiroki Satoh, Fumiaki Yamashita, Masayuki Tsujimoto, Hideyasu Murakami, Noriko Koyabu, Hisakazu Ohtani, and Yasufumi Sawada
CITRUS JUICES INHIBIT THE FUNCTION OF HUMAN ORGANIC ANION-TRANSPORTING POLYPEPTIDE OATP-B
Drug Metab Dispos 2005 33: 518-523. Published online January 7, 2005; 10.1124/dmd.104.002337 [Abstract] [Full Text] [PDF]  

Dhanashri Kolwankar, Douglas D. Glover, Joseph A. Ware, and Timothy S. Tracy
EXPRESSION AND FUNCTION OF ABCB1 AND ABCG2 IN HUMAN PLACENTAL TISSUE
Drug Metab Dispos 2005 33: 524-529. Published online January 7, 2005; 10.1124/dmd.104.002261 [Abstract] [Full Text] [PDF]  

Christopher A. Reilly and Garold S. Yost
STRUCTURAL AND ENZYMATIC PARAMETERS THAT DETERMINE ALKYL DEHYDROGENATION/HYDROXYLATION OF CAPSAICINOIDS BY CYTOCHROME P450 ENZYMES
Drug Metab Dispos 2005 33: 530-536. Published online January 7, 2005; 10.1124/dmd.104.001214 [Abstract] [Full Text] [PDF]  

Cuiping Chen, Rouchelle J. Mireles, Scott D. Campbell, Jian Lin, Jessica B. Mills, Jinghai J. Xu, and Teresa A. Smolarek
DIFFERENTIAL INTERACTION OF 3-HYDROXY-3-METHYLGLUTARYL-COA REDUCTASE INHIBITORS WITH ABCB1, ABCC2, AND OATP1B1
Drug Metab Dispos 2005 33: 537-546. Published online December 22, 2004; 10.1124/dmd.104.002477 [Abstract] [Full Text] [PDF]  

Run Tian, Noriko Koyabu, Satoshi Morimoto, Yukihiro Shoyama, Hisakazu Ohtani, and Yasufumi Sawada
FUNCTIONAL INDUCTION AND DE-INDUCTION OF P-GLYCOPROTEIN BY ST. JOHN'S WORT AND ITS INGREDIENTS IN A HUMAN COLON ADENOCARCINOMA CELL LINE
Drug Metab Dispos 2005 33: 547-554. Published online January 7, 2005; 10.1124/dmd.104.002485 [Abstract] [Full Text] [PDF]  

Liang Cui, Feng Qiu, and Xinsheng Yao
ISOLATION AND IDENTIFICATION OF SEVEN GLUCURONIDE CONJUGATES OF ANDROGRAPHOLIDE IN HUMAN URINE
Drug Metab Dispos 2005 33: 555-562. Published online January 11, 2005; 10.1124/dmd.104.001958 [Abstract] [Full Text] [PDF]  

Sonia Chalbot and Robert Morfin
HUMAN LIVER S9 FRACTIONS: METABOLISM OF DEHYDROEPIANDROSTERONE, EPIANDROSTERONE, AND RELATED 7-HYDROXYLATED DERIVATIVES
Drug Metab Dispos 2005 33: 563-569. Published online January 13, 2005; 10.1124/dmd.104.003004 [Abstract] [Full Text] [PDF]  

Susanne Andersson, Yvonne Hofmann, Åsa Nordling, Xue-qing Li, Sabina Nivelius, Tommy B. Andersson, Magnus Ingelman-Sundberg, and Inger Johansson
CHARACTERIZATION AND PARTIAL PURIFICATION OF THE RAT AND HUMAN ENZYME SYSTEMS ACTIVE IN THE REDUCTION OF N-HYDROXYMELAGATRAN AND BENZAMIDOXIME
Drug Metab Dispos 2005 33: 570-578. Published online January 7, 2005; 10.1124/dmd.104.002972 [Abstract] [Full Text] [PDF]  

Spencer Ling and Fakhreddin Jamali
EFFECT OF EARLY PHASE ADJUVANT ARTHRITIS ON HEPATIC P450 ENZYMES AND PHARMACOKINETICS OF VERAPAMIL: AN ALTERNATIVE APPROACH TO THE USE OF AN ANIMAL MODEL OF INFLAMMATION FOR PHARMACOKINETIC STUDIES
Drug Metab Dispos 2005 33: 579-586. Published online January 19, 2005; 10.1124/dmd.104.002360 [Abstract] [Full Text] [PDF]  

Don K. Walker, Samantha Abel, Pierre Comby, Gary J. Muirhead, Angus N. R. Nedderman, and Dennis A. Smith
SPECIES DIFFERENCES IN THE DISPOSITION OF THE CCR5 ANTAGONIST, UK-427,857, A NEW POTENTIAL TREATMENT FOR HIV
Drug Metab Dispos 2005 33: 587-595. Published online January 13, 2005; 10.1124/dmd.104.002626 [Abstract] [Full Text] [PDF]  

Norito Takamura, Toru Maruyama, Etsuo Chosa, Keiichi Kawai, Yasuhiro Tsutsumi, Yukie Uryu, Keishi Yamasaki, Tsuneo Deguchi, and Masaki Otagiri
BUCOLOME, A POTENT BINDING INHIBITOR FOR FUROSEMIDE, ALTERS THE PHARMACOKINETICS AND DIURETIC EFFECT OF FUROSEMIDE: POTENTIAL FOR USE OF BUCOLOME TO RESTORE DIURETIC RESPONSE IN NEPHROTIC SYNDROME
Drug Metab Dispos 2005 33: 596-602. Published online January 7, 2005; 10.1124/dmd.104.002782 [Abstract] [Full Text] [PDF]  

Commentaries:

John Schenkman
Commentary: David Kupfer, Ph.D., 1925–2004
Drug Metab Dispos 2005 33: 483. [Full Text] [PDF]  

Short Communications:

Li J. Yu, Yue Chen, Michael P. Deninno, Thomas N. O'Connell, and Cornelis E. C. A. Hop
IDENTIFICATION OF A NOVEL GLUTATHIONE ADDUCT OF DICLOFENAC, 4'-HYDROXY-2'-GLUTATHION-DESCHLORO-DICLOFENAC, UPON INCUBATION WITH HUMAN LIVER MICROSOMES
Drug Metab Dispos 2005 33: 484-488. Published online January 7, 2005; 10.1124/dmd.104.002840 [Abstract] [Full Text] [PDF]  

To see an article, click its [Full Text] link. To review many abstracts, check the boxes to the left of the titles you want, and click the 'Get All Checked Abstract(s)' button. To see one abstract at a time, click its [Abstract] link.


Cover Caption:

14-deoxy-12-hydroxy-andrographolide-19-O--D-glucuronide(A), metabolite M-5, 14 deoxy-12(13)-en-andrographolide-19-O--D-glucuronide (B), metabolite M-6, 14 deoxyandrographolide-19-O--D-glucuronide (C), and metabolite M-7, 3-oxoandrogarapholide-19-O--D-glucuronide (D). See the article by Cui et al. on page 555 of this issue.



Home Help [Feedback] [For Subscribers] [Archive] [Search] [Contents]
All ASPET Journals Molecular Pharmacology Pharmacological Reviews
The Journal of Pharmacology and Experimental 
Therapeutics Molecular Interventions Drug Metabolism and Disposition

Copyright © 2005 by the American Society for Pharmacology and Experimental Therapeutics.