Table 1

Pharmacokinetic parameters of CP117 after a single intravenous bolus administration of CP117 (450 μmol/kg) (N = 6)

Pharmacokinetic ParametersMean ± SDUnits
AUC43.2  ± 9.1μmol/liter · hr
AUMC6.4  ± 2.8μmol/liter · hr2
MRT0.14  ± 0.05hr
CL 10.9  ± 3.0liters · kg · hr−1
Vd ss 1.54  ± 0.52liters · kg−1
AUC (CP102)425  ± 9.0μmol/liter · hr