Table 1

Excretion of radioactivity (mean ± SD, N = 6) after a single 50 mg oral dose of [14C]CZ

ExcretaTime interval (hr)Per cent of Dose
Urine0–34.01  ± 1.18
3–65.11  ± 1.66
6–95.07  ± 2.65
9–123.57  ± 0.57
12–2411.00  ± 1.72
24–365.89  ± 1.54
36–484.69  ± 1.16
48–725.79  ± 1.24
72–962.08  ± 0.55
96–1201.15  ± 0.38
120–144 0.67  ± 0.17
Total excreted in urine0–14448.98  ± 4.69
Feces0–241.06  ± 2.58
24–4811.50  ± 7.41
48–729.90  ± 6.38
72–964.80  ± 3.06
96–1201.59  ± 1.55
120–144 0.80  ± 0.79
Total excreted in feces0–14429.64  ± 2.64
Total (urine + feces)0–14478.61  ± 5.23