P450 Isoenzyme | Rate of Formation (pmol/pmol P450 × min) | |
---|---|---|
5-HM | N-Dealkylated Tolterodine | |
1A1 | ND | ND |
1A2 | ND | ND |
2C8 | ND | ND |
2C9-Arg | ND | 0.25 ± 0.05 |
2C19 | ND | 1.51 ± 0.06 |
2D6 | 5.0 ± 0.35 | ND |
3A4 | ND | 0.23 ± 0.03 |
Data are mean ± SD of two experiments. ND, not detectable.