Deuterated Ezlopitant | CYP3A4 | CYP2D6 |
---|---|---|
[d 1]Ezlopitant | 1.07 ± 0.04 | 1.39 ± 0.07 |
[d 3]Ezlopitant | 0.95 ± 0.05 | 0.92 ± 0.07 |
[d 4]Ezlopitant | 0.97 ± 0.05 | 0.94 ± 0.05 |
[d 6]Ezlopitant | 0.93 ± 0.04 | 0.96 ± 0.05 |
[d 7]Ezlopitant | 1.05 ± 0.07 | 1.53 ± 0.08 |
Each value represents the mean ± S.D. of n = 6 determinations.