Saquinavir Concentration | Percentage of Unbound | ||
---|---|---|---|
Plasma | Albumin | Alpha-1-Acid Glycoprotein | |
μg/ml | |||
0.1 | 2.2 ± 0.5 | 13.1 ± 1.2 | 1.5 ± 0.2 |
0.5 | 2.8 ± 0.6 | 12.0 ± 2.7 | 1.6 ± 0.3 |
1 | 2.7 ± 0.5 | 12.4 ± 1.2 | 1.5 ± 0.4 |
5 | 2.8 ± 0.4 | 12.3 ± 2.4 | 1.6 ± 0.6 |
10 | 3.2 ± 0.8 | 11.4 ± 3.4 | 1.5 ± 0.5 |
20 | 3.1 ± 1.0 | 9.4 ± 1.5 | 3.6 ± 0.8 |
30 | 3.1 ± 0.6 | 10.2 ± 1.4 | 3.2 ± 0.3 |
Data are expressed as the mean ± S.D.