Inhibitor (100 μM) | % CYP1A2 Activity Remaining | % CYP1A1 Activity Remaining | % CYP2B1 Activity Remaining |
---|---|---|---|
R-Deprenyl | 45 ± 21-a | 100 ± 2 | 2.8 ± 0.21-a |
Desmethyldeprenyl | 65 ± 21-a | 94 ± 11-a | 11.5 ± 0.51-a |
Pargyline | 56 ± 21-a | 96 ± 4 | 10.2 ± 1.11-a |
R-2HMP | 60 ± 11-a | 93 ± 2 | 8.5 ± 0.41-a |
R-2HPA | 56 ± 21-a | 100 ± 1 | 8.6 ± 0.41-a |
R-2HMA | 97 ± 2 | 96 ± 1 | 85.4 ± 4.91-a |
R-2HA | 107 ± 4 | 96 ± 1 | 46.9 ± 2.11-a |
R-2HPcAc | 95 ± 1 | 95 ± 1 | 106 ± 3.2 |
Values are mean ± S.E.M. (n = 6). Incubation time was 10 min.
↵1-a Value significantly different from respective control (p < 0.05).