Low | Moderate | High | |
---|---|---|---|
CYP3A4-luc transgenic rats | Rifampicin pregnenolone | Phenobarbital nifedipine | Clotrimazole PCN dexamethasone |
CYP3A4-luc CD-1 Transgenic | Rifampicin pregnenolone | Phenobarbital nifedipine | Clotrimazole PCN dexamethasone |
CYP3A4-luc FVB/N transgenica | Rifampicin phenobarbital pregnenolone | Nifedipine | Clotrimazole PCN dexamethasone |
Mouse PXRb | Rifampicin phenobarbital clotrimazole | Dexamethasone pregnenolone | PCN nifedipine |
Rat PXRb | Rifampicin clotrimazole phenobarbital pregnenolone | Dexamethasone | PCN |
Human PXRb | PCN Dexamethasone | Pregnenolone phenobarbital nifedipine | Rifampicin clotrimazole |