Inhibitor | IC50 | Inhibition (% of Control) at the Highest Concentration Used |
---|---|---|
μM | ||
Ticlopidine | 0.32 | 100 (1) |
ThioTEPA | 1.75 | 100 (100) |
Tranylcypromine | 3.1 | 90 (100) |
Ketoconazole | 3.5 | 70 (100) |
Metyrapone | 4.14 | 100(1000) |
Xanthate C8 | 6.93 | 100(1000) |
Benzyl-isothiocyanate | 8.59 | 100 (100) |
Retinol | 17.0 | 70 (100) |
Deramciclane | 63.5 | 58 (100) |
Troglitazone | 88.2 | 55 (100) |
Ethinylestradiol | 100 | 50 (100) |