UGT Source | Sites of Expression | n | Km | Absolute Vmax | RelativeaVmax | Clint | Kinetic Profile |
---|---|---|---|---|---|---|---|
μM | pmol/min/mg | pmol/min/mg | μl/min/mg | ||||
1A1b | L, GI | – | 185 ± 86 | 336 ± 37 | 24 ± 3 | 0.1 | H |
1A7b | – | – | 30 ± 1 | 370 ± 7 | 23 ± 0.4 | 0.8 | H |
1A8 | GI | S | |||||
*1 | 1.7 | 298 ± 82 | 32,570 ± 5742 | 25,252 ± 4452 | 43 | ||
*2 (A 173G) | 1.5 | 317 ± 69 | 26,858 ± 4760 | 24,461 ± 4335 | 41 | ||
*3 (C277Y) | 1.3 | 118 ± 56 | 1864 ± 614 | 5371 ± 1771c | 28 | ||
1A9 | L, K, GI | H | |||||
*1 | 291 ± 31 | 8380 ± 1506 | 8380 ± 1506 | 29 | |||
*2 (C3Y) | 224 ± 32 | 9873 ± 2865 | 10,703 ± 3105 | 48 | |||
*3 (M33T) | 720 ± 250c,d | 4416 ± 500 | 11,888 ± 1346 | 17 | |||
1A10b | GI | – | 119 ± 12 | 434 ± 37 | 10 ± 0.8 | 0.1 | H |