Microsomal Preparation | Apparent Km | Vmax | Intrinsic Clearance |
---|---|---|---|
μM | nmol Eq/min/mg | Vmax/Km | |
LV22 | 156 ± 16 | 12 ± 0.3 | 0.07 ± 0.02 |
LV35 | 141 ± 6 | 25 ± 0.3 | 0.18 ± 0.05 |
LV41 | 134 ± 12 | 26 ± 0.7 | 0.20 ± 0.06 |
UGT1A6 | 135 ± 36 | 8 ± 0.2 | 0.06 ± 0.01 |
UGT1A9 | 3674 ± 470 | 0.6 ± 0.0 | 0.0002 ± 0.0 |