Km | Vmax | CLint = Vmax/Km | |
---|---|---|---|
μM | ml/min/g | ||
Homogeneous hepatocytes (S9 metabolism) | 1308 ± 419 | 8 ± 3 nmol/min/mg S9 protein or 800 nmol/min/g livera | 0.61 |
Homogeneous hepatocytes (transport) | 344 to 361 | 11.0 to 11.6 nmol/min/106 cells or 1,425 nmol/min/g liverb | 4.00 |
Transport/metabolism |
|
|
6.56
|
↵ a Based on 100 mg of protein per g of liver.
↵ b Based on 130 × 106 cells per g of liver (Zahlten and Stratman, 1974).