Protein Concentration in Perfusate (%) | Unbound Fraction in Perfusatea | Initial Free Drug Concentration in Perfusate | Radioactivity in Liver at End of Perfusion |
---|---|---|---|
% | μg/ml | % of dose | |
0.1 | 26.7 | 2.67 | 43.3 ± 4.5 |
0.5 | 8.3 | 0.83 | 18.9 ± 2.0 |
4.0 | 2.9 | 0.29 | 4.9 ± 0.5 |
↵ a Unbound fraction in perfusate values are an average of two determinations.