CYP2D6 Substrate | Number of Studies Predicted | fmCYP2D6 | References | ||
---|---|---|---|---|---|
From PM Dataa | From Regression Analysisb | ||||
Desipramine | 11(5)c | 0.877 | 0.799 | Brosen and Gram (1988) | |
Encainide | 2 | 0.857 | 0.814 | Funck-Brentano et al. (1989) | |
Flecainide | 1 | 0.412 | 0.748 | Mikus et al. (1989) | |
Imipramine | 7 | 0.457 | 0.549 | Brosen and Gram (1988) | |
Metoprolol | 12 | 0.828 | 0.695 | Silas et al. (1985) | |
Mexiletine | 1 | 0.493 | 0.247 | Turgeon et al. (1991) | |
Propafenone | 2 | 0.763 | 0.540 | Siddoway et al. (1987) | |
Propranolol | 9 | 0.367 | 0.579 | Raghuram et al. (1984) | |
Tolterodine | 1 | 0.942 | 0.891 | Brynne et al. (1998) |