NSAIDs | rOat1a | rOat2 | rOat3a | hOat2b |
---|---|---|---|---|
μM | μM | μM | μM | |
Salicylate | 2110 ± 190 | 399 ± 133 | 519 ± 132 | N.D. |
Diclofenac | 4.56 ± 1.24 | 107 ± 29 | 3.17 ± 0.43 | 14.3 |
Sulindac | 99.9 ± 18.6 | 537 ± 282 | 7.72 ± 1.32 | 440 |
Indomethacin | 7.44 ± 3.88 | 1.25 ± 0.40 | 1.29 ± 0.46 | 64.1 |
Etodolac | >100 | 344 ± 99 | 9.98 ± 1.48 | N.D. |
Tolmetin | 15.4 ± 3.2 | 288 ± 118 | 8.78 ± 2.32 | N.D. |
Ibuprofen | 4.33 ± 0.40 | 346 ± 100 | 3.57 ± 1.09 | 692 |
Ketoprofen | 6.11 ± 1.66 | 3.31 ± 0.18* | 4.31 ± 1.28 | 400 |
Naproxen | 5.54 ± 0.89 | >1000 | 19.1 ± 6.9 | 486 |
Phenylbutazone | 47.9 ± 9.2 | 387 ± 129 | 8.48 ± 0.78 | N.D. |