Substrate | Inhibitor | Percentage Inhibition |
---|---|---|
Testosterone | Ketoconazole | |
1 μM | 0 | |
10 μM | 10 | |
5-MOP | ||
10 μM | 38 | |
50 μM | 84 | |
8-MOP | ||
2 μM | 60 | |
10 μM | 81 | |
Phenacetin | Furafylline | |
3 μM | 50 | |
30 μM | 55 | |
α-Naphthoflavone | ||
0.1 μM | 26 | |
5 μM | 94 | |
5-MOP | ||
10 μM | 95 | |
50 μM | 100 | |
8-MOP | ||
2 μM | 96 | |
10 μM | 100 | |
Chlorzoxazone | Diethyldithiocarbamate, 20 μM | 48 |
5-MOP | ||
10 μM | 58 | |
50 μM | 89 | |
8-MOP | ||
2 μM | 62 | |
10 μM | 87 | |
Dextromethorphan | Quinine | |
5 μM | 1 | |
10 μM | 23 | |
5-MOP | ||
10 μM | 79 | |
50 μM | 100 | |
8-MOP | ||
2 μM | 94 | |
| 10 μM | 100 |