TABLE 1

Km,app and scaled CLINT values for deltamethrin and esfenvalerate in rats and humans

Data are mean ± S.D. (n = 3).




Km,app

Clearance
μM ml/min/kg body wt.
Deltamethrin
    Rat microsomes 39 89.0 ± 23.7
    Human microsomes 75 162.1 ± 32.7
Esfenvalerate
    Rat microsomes 22 108.2 ± 2.2
    Human microsomes
21
37.3 ± 10.3