Kinetic Parameters | Vmax | Km | Vmax/Km |
---|---|---|---|
pmol/min/mg protein | μM | μl/min/mg protein | |
Ebastine | |||
Dealkylation | 108.2 ± 29.6 | 17.5 ± 2.3 | 6.18 ± 1.16 |
Hydroxylation | 10.9 ± 3.0 | 5.1 ± 1.3 | 2.14 ± 0.48 |
Hydroxyebastine | |||
Dealkylation | 456.4 ± 69.1 | 13.7 ± 3.8 | 33.3 ± 9.0 |
Carboxylation | |||
Carebastine | 340.2 ± 64.1 | 8.9 ± 0.9 | 38.2 ± 6.5 |
Dealkylation | 94.1 ± 27.0 | 61 ± 6.1 | 1.54 ± 0.51 |