Interaction | Mean AUCi/AUC | fmCYP3A4 | Reference | |
---|---|---|---|---|
Erythromycin | ||||
1 | + Alprazolam | 2.5 | 0.8 | Yasui et al. (1996) |
2 | + Buspirone | 5.9 | 0.99 | Kivisto et al. (1997) |
3 | + Carbamazepine | 1.4 | 0.6 | Barzaghi et al. (1987) |
4 | + Cerivastatin | 1.21 | 0.37 | Muck et al. (1998) |
5 | + Cyclosporinea | 2.15 | 0.71 | Gupta et al. (1989) |
6 | + Cyclosporinea | 2.22 | 0.71 | Freeman et al. (1987) |
7 | + Felodipine | 2.5 | 0.81 | Bailey et al. (1996) |
8 | + Loratadine | 1.5 | 0.6 | Brannan et al. (1995) |
9 | + Midazolam | 4.11 | 0.94 | Olkkola et al. (1993); Zimmermann et al. (1996) |
10 | + Nitrazepam | 1.25 | 0.6 | Luurila et al. (1995) |
11 | + Quinidine | 1.2 | 0.76 | Damkier et al. (1999a) |
12 | + Simvastatin | 6.2 | 0.99 | Kantola et al. (1998) |
13 | + Terfenadine | 2.1 | 0.74 | Honig et al. (1994) |
14 | + Triazolam | 2.06 | 0.92 | Phillips et al. (1986) |
15 | + Triazolam | 3.36 | 0.92 | Greenblatt et al. (1998) |
Clarithromycin | ||||
16 | + Cisapride | 3.16 | 0.95 | van Haarst et al. (1998) |
17 | + Midazolam | 3.6 | 0.94 | Yeates et al. (1996) |
18 | + Midazolam | 7 | 0.94 | Gorski et al. (1998) |
19 | + Pimozide | 2.12 | 0.4 | Desta et al. (1999) |
20 | + Terfenadine | 2.5 | 0.74 | Honig et al. (1994) |
21 | + Triazolam | 5.1 | 0.92 | Greenblatt et al. (1998) |
Azithromycin | ||||
22 | + Midazolam | 0.87 | 0.94 | Backman et al. (1995) |
23 | + Midazolam | 1.23 | 0.94 | Zimmermann et al. (1996) |
24 | + Triazolam | 1.03 | 0.92 | Greenblatt et al. (1998) |
Diltiazem | ||||
25 | + Cyclosporinea | 1.49 | 0.71 | Asberg et al. (1999) |
26 | + Cyclosporinea | 1.57 | 0.71 | Foradori et al. (1998) |
27 | + Cyclosporinea | 1.25 | 0.71 | Brockmoller et al. (1990) |
28 | + Lovastatin | 3.6 | 0.99 | Azie et al. (1998) |
29 | + Midazolam | 3.75 | 0.94 | Backman et al. (1994) |
30 | + Nifedipine | 2.22 | 0.71 | Tateishi et al. (1989) |
31 | + Nifedipine | 3.11 | 0.71 | Tateishi et al. (1989) |
32 | + Nifedipine | 2.39 | 0.71 | Ohashi et al. (1990) |
33 | + Simvastatin | 4.82 | 0.99 | Mousa et al. (2000) |
34 | + Triazolam | 3.38 | 0.92 | Varhe et al. (1996) |
35 | + Triazolam | 2.3 | 0.92 | Kosuge et al. (1997) |
36 | + Buspirone | 5.5 | 0.99 | Lamberg et al. (1998) |
37 | + Quinidine | 1.53 | 0.76 | Laganiere et al. (1996) |
↵ a fmCYP3A4 values obtained by regression analysis using eq. 1.