Compound | pBCECs | ||
---|---|---|---|
f2 | IC50 | ||
μM | |||
GG918 | 0.001 ± 0.0003 | 0.002 ± 0.0006 | |
LY335979 | 0.003 ± 0.0007 | 0.007 ± 0.001 | |
SDZ-PSC833 | 0.006 ± 0.003 | 0.02 ± 0.01 | |
Itraconazole | 0.02 ± 0.01 | 0.05 ± 0.01 | |
Loperamide | 0.79 ± 0.11 | 1.86 ± 0.41 | |
Desmethylloperamide | 0.96 ± 0.29 | 2.35 ± 0.60 | |
Verapamil | 0.60 ± 0.20 | 3.22 ± 0.82 | |
Quinidine | 1.12 ± 0.42 | 7.19 ± 1.60 | |
Amprenavir | 8.61 ± 0.83 | 19.7 ± 6.78 |