Probe | IC50 Value | ||||||
---|---|---|---|---|---|---|---|
<5 | 5-15 | 15-50 | >50 | ||||
μM | |||||||
Calcein-AM | 918, CsA | K | V, Q, VB, P, A | ||||
Colchicine | 918, CsA | K | V, VB | Q, P, A, Dau | |||
Digoxin | 918, CsA, K | V, Q | VB | ||||
Prazosin | 918, CsA, K, V | Q | VB | Prop, A, I | |||
Vinblastine | 918 | CsA, K | V, Q | VB, A, Dau |
918, GF120918; A, amprenavir; CsA, cyclosporine A; Dau, daunorubicin; I, indinavir; K, ketoconazole; P, prazosin; Prop, propranolol; Q, quinidine; VB, vinblastine; V, verapamil.