BBB Model | Km | Vmax | Vmax/Km |
---|---|---|---|
μM | pmol · min–1 · mg protein–1 | μl · min–1 · mg protein–1 | |
BBM | 1448.2 ± 183.1 | 624.9 ± 38.2 | 0.447 ± 0.083 |
MDCKII-MDR1 | 178.4 ± 12.4 | 92.5 ± 3.6 | 0.521 ± 0.023 |
BBMEC | 474.3 ± 98.1 | 122.8 ± 22.9 | 0.262 ± 0.015 |
BBMEC + indomethacin | 1299.6 ± 94.2 | 181.1 ± 4.5 | 0.141 ± 0.014 |
Values represent mean ± S.E.M. (n = 9) from three separate studies