Form Dosed | Form Measured | Matrix | Time | KO | WT | ||||
---|---|---|---|---|---|---|---|---|---|
Conc. | Tissue/Plasma Ratio | Conc. | Tissue/Plasma Ratio | ||||||
h | ng/ml | ng/ml | |||||||
Acid | Acid | Plasma | 0.5 | 409 ± 200 | 388 ± 97 | ||||
Plasma | 1.5 | 131 ± 84 | 162 ± 38 | ||||||
Plasma | 3 | 56 ± 17 | 51 ± 24 | ||||||
Liver | 0.5 | 3391 ± 972 | 10 ± 6 | 2546 ± 380 | 6.7 ± 0.8 | ||||
Liver | 1.5 | 1338 ± 435 | 13 ± 5 | 1822 ± 563 | 9.1 ± 6.1 | ||||
|
| Liver | 3 | 559 ± 340 | 13 ± 11 | 881 ± 601 | 21 ± 14 |