Reaction | HLM | Recombinant UGT1A9 | ||||||||
---|---|---|---|---|---|---|---|---|---|---|
Km | Vmax | Vmax/Km | Km | Vmax | Vmax/Km | |||||
μM | pmol/min/mg protein | μl/min/mg protein | μM | pmol/min/mg protein | μl/min/mg protein | |||||
N1-Glucuronidation | 64.1 | 87.5 | 1.37 | 13.2 | 207.3 | 15.7 | ||||
N2-Glucuronidation | 72.7 | 46.5 | 0.64 | 12.9 | 80.4 | 6.2 |