TABLE 5
Inhibitory activity of temsirolimus metabolites against LNCaP cell proliferation
Sample
IC
50
nM
Temsirolimus
2
Seco-temsirolimus
∼5000
M8
∼1000
M9
∼100
M10
∼200
M11
∼200
M12
∼1000
M13
∼1000