Inducer | Plasma | Hepatocytes | ||||
---|---|---|---|---|---|---|
Conc. | fu, p | Conc. | fu, hept | |||
μM | μM | |||||
BST | 1,10 | 0.0074 (0.003) | 1 | 0.189 (0.010) | ||
CMZ | 1,10 | 0.041 (0.002) | 20 | 0.520 (0.021) | ||
DEX | 1,10 | 0.300 (0.011) | 100 | 0.589 (0.043) | ||
EFA | 1,10 | 0.029 (0.004) | 5 | 0.063 (0.006) | ||
PB | 1,10 | 0.700 (0.092) | 250 | 1.000 (0.074) | ||
RIF | 1,10 | 0.175 (0.011) | 1 | 0.419 (0.052) |