Inhibitor | Inhibition at Inhibitor Concentration [μM] | IC50a | ||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
0.52 | 2.06 | 4.13 | 8.25 | 16.5 | 33 | 100 | ||||||||
% | % | % | % | % | % | % | μM | |||||||
SKF-Acid | 102 | 342 | 483 | 642 | 861 | 941 | ∼4 | |||||||
SKF-Alcohol | 32 | 54 | 160 | 521 | 841 | ∼33 | ||||||||
SKF26754 | 152 | 384 | 451 | 743 | 33–100 | |||||||||
SKF8742 | 171 | 202 | 443 | >100 | ||||||||||
SKF525A |
|
|
|
| 130 | 254 | 444 | >100 |
↵ a The IC50 value was estimated by interpolation