Compound | PAMPA Retention Factor (Rf) | PAMPA Papp | A > B Papp in MDCK |
---|---|---|---|
× 10-6 cm/s | × 10-6 cm/s | ||
Buspirone | 0.5 ± 0.04 | 27.1 ± 19.95 | 23.3 ± 3.91 |
Caffeine | N.D. | N.D. | 30.6 ± 2.47 |
Carbamazepine | 0.2 ± 0.05 | 17.3 ± 2.38 | 29.4 ± 2.46 |
Carisoprodol | 0.2 ± 0.06 | 16.2 ± 2.57 | 25.6 ± 2.86 |
Chlorpromazine | 0.9 ± 0.03 | 6.1 ± 1.64 | 4.1 ± 0.44 |
Citalopram | 0.5 ± 0.04 | 14.5 ± 3.74 | 18.3 ± 3.76 |
Cyclobenzaprine | 0.8 ± 0.04 | 13.0 ± 2.49 | 12.2 ± 0.34 |
Diazepam | 0.5 ± 0.03 | 17.4 ± 3.18 | 27.7 ± 2.45 |
Ethosuximide | 0.1 ± 0.12 | 10.0 ± 1.24 | 26.8 ± 2.59 |
Fluoxetine | 0.3 ± 0.08 | 0.1 ± 0.03 | 6.3 ± 0.61 |
Fluvoxamine | 0.8 ± 0.06 | 10.0 ± 0.35 | 13.0 ± 2.69 |
Haloperidol | 0.8 ± 0.04 | 8.6 ± 1.30 | 12.3 ± 3.31 |
Hydrocodone | 0.2 ± 0.08 | 11.9 ± 0.25 | 20.0 ± 1.77 |
Hydroxyzine | 0.6 ± 0.01 | 12.5 ± 0.56 | 16.1 ± 3.25 |
Lamotrigine | N.D. | N.D. | 22.9 ± 0.97 |
Methylphenidate | 0.3 ± 0.04 | 23.2 ± 6.53 | 24.7 ± 2.03 |
Metoclopramide | 0.4 ± 0.05 | 11.0 ± 1.27 | 17.7 ± 2.61 |
Midazolam | 0.5 ± 0.02 | 13.1 ± 1.28 | 22.5 ± 2.08 |
Morphine | 0.2 ± 0.05 | 4.8 ± 0.78 | 1.8 ± 0.07 |
Nortriptyline | 0.8 ± 0.06 | 10.1 ± 2.51 | 9.1 ± 0.16 |
Paroxetine | 0.9 ± 0.01 | 5.7 ± 1.08 | 6.1 ± 0.29 |
Phenytoin | 0.3 ± 0.03 | 15.2 ± 0.63 | 24.0 ± 1.80 |
Propoxyphene | 0.6 ± 0.04 | 13.1 ± 1.08 | 21.9 ± 4.65 |
Risperidone | 0.5 ± 0.05 | 13.8 ± 0.50 | 19.8 ± 3.24 |
9-Hydroxyrisperidone | N.D. | N.D. | 16.8 ± 1.04 |
Selegiline | 0.6 ± 0.04 | 26.1 ± 11.91 | 23.2 ± 1.46 |
Sertraline | 0.9 ± 0.02 | 2.8 ± 0.50 | 1.9 ± 0.37 |
Sulpiride | 0.01 ± 0.01 | 0.03 ± 0.03 | 0.9 ± 0.47 |
Thiopental | 0.5 ± 0.02 | 21.1 ± 6.39 | 25.2 ± 1.15 |
Trazodone | 0.5 ± 0.03 | 13.6 ± 1.07 | 19.7 ± 0.64 |
Venlafaxine | N.D. | N.D. | 22.1 ± 0.77 |
Zolpidem | 0.4 ± 0.03 | 15.7 ± 1.45 | 23.4 ± 0.76 |
N.D., no data were generated.