TSNA | Vmax | KM | Vmax/KM | Normalized Vmax/KM UGT2B10/UGT1A4 Ratioa | |
---|---|---|---|---|---|
pmol/min/mg total protein | mM | nl/min/mg total protein | |||
UGT1A4 | NNAL | 99 ± 27b | 22.79 ± 3.83 | 4.35 ± 0.96 | Referent |
NNN | 182 ± 43 | 26.24 ± 14.27 | 7.70 ± 2.13 | Referent | |
NAB | 166 ± 22 | 5.37 ± 1.61 | 32.1 ± 6.63 | Referent | |
NAT | 124 ± 4 | 3.31 ± 0.23 | 37.6 ± 2.31 | Referent | |
UGT2B10 | NNAL | 7.55 ± 0.37 | 3.62 ± 2.31 | 3.07 ± 2.13 | 3.0 |
NNN | 7.66 ± 1.63 | 1.18 ± 0.27 | 6.60 ± 1.08 | 3.6 | |
NAB | 41.09 ± 11.28 | 0.28 ± 0.00 | 147 ± 42.0 | 19 | |
NAT | 52.65 ± 14.99 | 0.22 ± 0.06 | 242 ± 2.86 | 27 | |
HLMc | NNAL | 259 ± 42 | 0.85 ± 0.42 | 348 ± 163 | |
NNN | 1400 ± 60 | 3.17 ± 0.37 | 446 ± 61 | ||
NAB | 2476 ± 621 | 0.20 ± 0.03 | 12,806 ± 5069 | ||
| NAT | 2593 ± 457 | 0.16 ± 0.01 | 16,227 ± 2852 |
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