Cell Lines | Substrate | Inhibitor | Km | IC50 |
---|---|---|---|---|
μM | μM | |||
Mock-HEK293 | YM758 | 135 | ||
rOct1-HEK293 | MPP | YM758 | 23.8 | |
rOct1-HEK293 | Metformin | YM758 | <10.0 | |
hOCT1-HEK293 | MPP | YM758 | 40.5 | |
OATP1B1-HEK293 | E217βG | YM758 | 13.0 | |
LLC-MDR1 | YM758 | 20.9 | ||
Human hepatocyte | YM758 | 87.9 | ||
Human hepatocyte | YM758 | Quinidine |
| 147 |