TABLE 1

Michaelis-Menten parameters (Vmax and KM) of BNX-G and FLX-G formation in human liver microsomes

DonorBNX
FLX
VmaxKMVmax/KMVmaxKMVmax/KM
nmol/mg/minmMμl/min/mgnmol/mg/minmMμl/min/mg
10.8650.3222.690.2230.1361.64
21.240.3963.130.1900.3690.515
30.0490.2860.171