UGT Enzyme | Vmax | Km | Clint |
---|---|---|---|
nmol/min/mg | mM | μl/min/mg | |
UGT1A1 | N.A. | N.A. | |
UGT1A3 | 0.6 ± 0.3 | 6.4 ± 0.76 | 0.09 |
UGT1A4 | 0.4 ± 0.1 | 3.1 ± 0.32 | 0.13 |
UGT1A6 | 0.70 ± 0.44a | 3.2 ± 0.53a | 0.22a |
UGT1A8 | 0.87 ± 0.5 | 5.9 ± 0.76 | 0.14 |
UGT1A9 | 0.96 ± 0.5 | 6.3 ± 0.75 | 0.15 |
0.98 ± 0.06a | 5.2 ± 0.84a | 0.19a | |
UGT1A10 | 0.88 ± 0.3 | 5.5 ± 0.39 | 0.16 |
UGT2B7 | 1.2 ± 0.15 | 1.4 ± 0.09 | 0.86 |
| 0.66 ± 0.44a | 2.1 ± 0.35a | 0.31a |
N.A., no activity.
↵ a Denotes literature-reported values (Ethell et al., 2003).