Metabolite | RT | Group 1 | Group 2 | ||||||
---|---|---|---|---|---|---|---|---|---|
Urine | Feces | Bile | Urine | Feces | |||||
min | % dose | ||||||||
M1 | 24.4 | 1.58 | 1.24 | 0.96 | 2.55 | 2.40 | |||
M2 | 28.6 | N.D. | 12.2 | 0.02 | N.D. | 5.09 | |||
M4 | 34.1 | N.D. | 0.37 | N.D. | N.D. | N.D. | |||
M7 | 27.6 | 1.46 | 3.70 | 0.32 | 1.85 | 2.76 | |||
M10 | 19.0 | N.D. | 0.09 | 0.24 | 0.46 | 0.26 | |||
M13 | 21.3 | N.D. | 3.07 | 0.06 | N.D. | 0.96 | |||
Apixaban | 48.9 | 21.5 | 34.0 | 0.84 | 23.9 | 34.5 | |||
Othersa | N.A. | N.A. | 1.30 | N.A. | N.A. | 0.73 | |||
Total | N.A. | 24.5 | 56.0 | 2.44 | 28.8 | 46.7 |
RT, retention time; N.D., not detected; N.A., not applicable.
↵ a Radioactivity distributed among many small peaks each representing ≤0.02%.