Inhibitor | Ki Values | ||||||
---|---|---|---|---|---|---|---|
M1 | M2 | M3a | M3b | ||||
μM | |||||||
Ketoconazole (CYP3A4) | 1.33 ± 0.65 | 0.788 ± 0.063 | NI | 12.8 ± 4.09 | |||
Pentoxyresorufin (CYP2B6) | NI | NI | NI | NI | |||
Sulfaphenazole (CYP2C9) | 1.56 ± 0.97 | NI | 0.617 ± 0.195 | 1.04 ± 0.009 | |||
Tranylcypromine (CYP2C19) | NI | NI | NI | NI |
NI, not inhibited.