Strain | Treatment Route | Tmax | Cmax | t1/2 | AUC0-∞ |
---|---|---|---|---|---|
h | nmol/ml | h | nmol · h/ml | ||
WT | Oral | 0.50 | 4.9 ± 1.2 | 1.38 ± 0.74 | 8.0 ± 0.5 |
IE-Cpr-null | Oral | 0.50 | 9.0 ± 2.5a | 0.91 ± 0.26 | 12.8 ± 2.3a |
WT | Intravenous | 0.17 | 6.6 ± 1.5 | 0.23 ± 0.02 | 3.6 ± 0.8 |
IE-Cpr-null | Intravenous | 0.17 | 6.6 ± 0.9 | 0.26 ± 0.05 | 3.8 ± 0.6 |
AUC, area under the concentration-time curve.
↵ a p < 0.01, as compared with similarly treated WT mice.