FK1706 Conc. during Preincubation | Midazolam 1′-Hydroxylase Activity | |||
---|---|---|---|---|
Before Dialysis | After Dialysis | |||
NADPH (+) | NADPH (−) | NADPH (+) | NADPH (−) | |
pmol/min/mg protein | ||||
0 μM (control) | 150 ± 10 | 114 ± 9 | 54.1 ± 2.9 | 51.9 ± 2.9 |
2 μM | 9.94 ± 0.18 (6.6) | 60.9 ± 5.7 (53.5) | 3.48 ± 0.59 (6.4) | 50.3 ± 2.8 (96.9) |