TABLE 4

Clint values for CYP2J2 substrates

CompoundMean ClintS.D.
μl/min/pmol CYP2J2
Terfenadinea3.981.39
Astemizolea1.140.10
Amiodarone0.490.04
Albendazole0.360.02
Danazol0.290.02
Thioridazine0.270.04
Tamoxifen0.190.004
Cyclosporin A0.120.03
Nabumetone0.110.001
Mesoridazine0.060.007
  • a Previously identified substrates serve as positive controls.