Compound | Mean Clint | S.D. |
---|---|---|
μl/min/pmol CYP2J2 | ||
Terfenadinea | 3.98 | 1.39 |
Astemizolea | 1.14 | 0.10 |
Amiodarone | 0.49 | 0.04 |
Albendazole | 0.36 | 0.02 |
Danazol | 0.29 | 0.02 |
Thioridazine | 0.27 | 0.04 |
Tamoxifen | 0.19 | 0.004 |
Cyclosporin A | 0.12 | 0.03 |
Nabumetone | 0.11 | 0.001 |
Mesoridazine | 0.06 | 0.007 |
↵a Previously identified substrates serve as positive controls.