Inhibition of CD10604 reduction in human liver cytosol
| Inhibitor | Inhibitor Concentration | Mean Turnover Rate | Inhibition |
|---|---|---|---|
| μM | pmol/min/mg protein | % | |
| Phenolphthalein | 0 | 1197 | 0 |
| 0.5 | 874 | 27 | |
| 5 | 459 | 62 | |
| Flufenamic acid | 0 | 941 | 0 |
| 1 | 717 | 24 | |
| 10 | 556 | 41 | |
| Rutin hydrate | 0 | 930 | 0 |
| 10 | 924 | 1 | |
| 100 | 797 | 14 | |
| Dexamethasone | 0 | 877 | 0 |
| 5 | 896 | 0 | |
| 50 | 570 | 35 | |
| Menadione | 0 | 877 | 0 |
| 10 | 754 | 14 | |
| 100 | 428 | 51 | |
| Quercitrin | 0 | 899 | 0 |
| 10 | 860 | 4 | |
| 100 | 808 | 10 | |
| Medroxyprogesterone acetate | 0 | 912 | 0 |
| 0.2 | 860 | 6 | |
| 2 | 554 | 39 |